JP2021527650A5 - - Google Patents

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Publication number
JP2021527650A5
JP2021527650A5 JP2020569890A JP2020569890A JP2021527650A5 JP 2021527650 A5 JP2021527650 A5 JP 2021527650A5 JP 2020569890 A JP2020569890 A JP 2020569890A JP 2020569890 A JP2020569890 A JP 2020569890A JP 2021527650 A5 JP2021527650 A5 JP 2021527650A5
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JP
Japan
Prior art keywords
arenediyl
alkyl
cycloalkyl
aryl
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020569890A
Other languages
English (en)
Japanese (ja)
Other versions
JP7498122B2 (ja
JP2021527650A (ja
Filing date
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Application filed filed Critical
Priority claimed from PCT/US2019/037543 external-priority patent/WO2019241796A1/en
Publication of JP2021527650A publication Critical patent/JP2021527650A/ja
Publication of JP2021527650A5 publication Critical patent/JP2021527650A5/ja
Application granted granted Critical
Publication of JP7498122B2 publication Critical patent/JP7498122B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020569890A 2018-06-15 2019-06-17 IL-17およびRORγの阻害用のピラゾール化合物およびイミダゾール化合物 Active JP7498122B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862685742P 2018-06-15 2018-06-15
US62/685,742 2018-06-15
US201862687602P 2018-06-20 2018-06-20
US62/687,602 2018-06-20
PCT/US2019/037543 WO2019241796A1 (en) 2018-06-15 2019-06-17 Pyrazole and imidazole compounds for inhibition of il-17 and rorgamma

Publications (3)

Publication Number Publication Date
JP2021527650A JP2021527650A (ja) 2021-10-14
JP2021527650A5 true JP2021527650A5 (enExample) 2022-06-22
JP7498122B2 JP7498122B2 (ja) 2024-06-11

Family

ID=67482968

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020569890A Active JP7498122B2 (ja) 2018-06-15 2019-06-17 IL-17およびRORγの阻害用のピラゾール化合物およびイミダゾール化合物

Country Status (11)

Country Link
US (2) US11993574B2 (enExample)
EP (1) EP3807265A1 (enExample)
JP (1) JP7498122B2 (enExample)
KR (1) KR102887518B1 (enExample)
CN (2) CN112654610B (enExample)
AU (1) AU2019286531B2 (enExample)
BR (1) BR112020025605A2 (enExample)
CO (1) CO2021000229A2 (enExample)
IL (2) IL322405A (enExample)
MX (1) MX2020013692A (enExample)
WO (1) WO2019241796A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI831738B (zh) 2016-12-16 2024-02-11 美商瑞塔醫藥有限責任公司 用於抑制RORγ及其他用途的嘧啶三環烯酮衍生物
CN115867348B (zh) * 2020-04-30 2025-05-06 詹森药业有限公司 作为il-17调节剂的咪唑并嘧啶
CN114409724A (zh) * 2022-01-10 2022-04-29 南京联智医药科技有限公司 一种新的达那唑制备方法
CN118852108B (zh) * 2024-07-15 2025-09-26 南京林业大学 一种用于检测有机磷农药敌敌畏和敌百虫的新型樟脑基荧光探针及其制备方法与应用

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