JP2021522167A5 - - Google Patents

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JP2021522167A5
JP2021522167A5 JP2020557178A JP2020557178A JP2021522167A5 JP 2021522167 A5 JP2021522167 A5 JP 2021522167A5 JP 2020557178 A JP2020557178 A JP 2020557178A JP 2020557178 A JP2020557178 A JP 2020557178A JP 2021522167 A5 JP2021522167 A5 JP 2021522167A5
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JP7329260B2 (ja
JP2021522167A (ja
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Priority claimed from PCT/US2019/027844 external-priority patent/WO2019204419A1/en
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Priority to JP2025035562A priority patent/JP2025083398A/ja
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JP2020557178A 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用 Active JP7329260B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2023129305A JP7651203B2 (ja) 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用
JP2025035562A JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

Applications Claiming Priority (3)

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US201862660729P 2018-04-20 2018-04-20
US62/660,729 2018-04-20
PCT/US2019/027844 WO2019204419A1 (en) 2018-04-20 2019-04-17 Boronic acid derivatives and therapeutic uses thereof

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JP2023129305A Division JP7651203B2 (ja) 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用

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JP2021522167A JP2021522167A (ja) 2021-08-30
JP2021522167A5 true JP2021522167A5 (enExample) 2022-04-08
JP7329260B2 JP7329260B2 (ja) 2023-08-18

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JP2020557178A Active JP7329260B2 (ja) 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用
JP2023129305A Active JP7651203B2 (ja) 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用
JP2025035562A Pending JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

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JP2023129305A Active JP7651203B2 (ja) 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用
JP2025035562A Pending JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

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US (2) US12016868B2 (enExample)
EP (1) EP3781576B1 (enExample)
JP (3) JP7329260B2 (enExample)
CN (1) CN112424209A (enExample)
AU (1) AU2019256351B2 (enExample)
CA (1) CA3097127A1 (enExample)
TW (1) TW201945005A (enExample)
WO (1) WO2019204419A1 (enExample)
ZA (1) ZA202006377B (enExample)

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US12637481B2 (en) 2020-03-18 2026-05-26 Qpex Biopharma, Inc. Boronic acid derivatives and therapeutic uses thereof
IL297458A (en) 2020-05-05 2022-12-01 Qpex Biopharma Inc Boronic acid derivatives and their synthesis, polymorphic forms and medicinal uses
CN113880871B (zh) * 2020-10-16 2022-08-23 中国科学院兰州化学物理研究所 一种饱和单硼类化合物的制备方法
US20240299375A1 (en) 2021-03-08 2024-09-12 Eli Lilly And Company Use of mevidalen and other d1 positive allosteric modulators in the treatment of hallucinations and dementia-related psychosis
CN117337173A (zh) 2021-03-09 2024-01-02 伊莱利利公司 美维达林和其他d1正向别构调节剂用于减缓帕金森氏病进展的用途
TW202404610A (zh) * 2022-06-24 2024-02-01 大陸商瑞石生物醫藥有限公司 一種硼酸酯衍生物的結晶、其製備方法及用途
US12642808B2 (en) * 2023-09-22 2026-06-02 City University Of Hong Kong Methods of inhibiting Klebsiella pneumoniae carbapenemase-2
CN122374319A (zh) * 2023-12-04 2026-07-10 珠海联邦制药股份有限公司 硼酸类β-内酰胺酶抑制剂及其制备方法和应用
CN119119096B (zh) * 2024-09-09 2025-09-16 郑州药领医药科技有限公司 一种4-((4,4,5,5-四甲基-1,3,2-二氧硼杂环戊烷-2-基)甲基)哌啶-1-甲酸叔丁酯的合成方法

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