JP2023159197A5 - - Google Patents

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JP2023159197A5
JP2023159197A5 JP2023129305A JP2023129305A JP2023159197A5 JP 2023159197 A5 JP2023159197 A5 JP 2023159197A5 JP 2023129305 A JP2023129305 A JP 2023129305A JP 2023129305 A JP2023129305 A JP 2023129305A JP 2023159197 A5 JP2023159197 A5 JP 2023159197A5
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JP7651203B2 (ja
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JP2023129305A 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用 Active JP7651203B2 (ja)

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JP2025035562A JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

Applications Claiming Priority (4)

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US201862660729P 2018-04-20 2018-04-20
US62/660,729 2018-04-20
JP2020557178A JP7329260B2 (ja) 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用
PCT/US2019/027844 WO2019204419A1 (en) 2018-04-20 2019-04-17 Boronic acid derivatives and therapeutic uses thereof

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JP2020557178A Division JP7329260B2 (ja) 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用

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JP2023159197A JP2023159197A (ja) 2023-10-31
JP2023159197A5 true JP2023159197A5 (enExample) 2023-11-24
JP7651203B2 JP7651203B2 (ja) 2025-03-26

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JP2020557178A Active JP7329260B2 (ja) 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用
JP2023129305A Active JP7651203B2 (ja) 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用
JP2025035562A Pending JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

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US (2) US12016868B2 (enExample)
EP (1) EP3781576B1 (enExample)
JP (3) JP7329260B2 (enExample)
CN (1) CN112424209A (enExample)
AU (1) AU2019256351B2 (enExample)
CA (1) CA3097127A1 (enExample)
TW (1) TW201945005A (enExample)
WO (1) WO2019204419A1 (enExample)
ZA (1) ZA202006377B (enExample)

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Publication number Priority date Publication date Assignee Title
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CN113880871B (zh) * 2020-10-16 2022-08-23 中国科学院兰州化学物理研究所 一种饱和单硼类化合物的制备方法
EP4304581A1 (en) 2021-03-08 2024-01-17 Eli Lilly And Co. Use of mevidalen and other d1 positive allosteric modulators in the treatment of hallucinations and dementia-related psychosis
BR112023018196A2 (pt) 2021-03-09 2023-12-12 Lilly Co Eli Uso de mevidalen e outros moduladores alostéricos positivos d1 para retardar a progressão da doença de parkinson
TW202404610A (zh) * 2022-06-24 2024-02-01 大陸商瑞石生物醫藥有限公司 一種硼酸酯衍生物的結晶、其製備方法及用途
US20250099495A1 (en) * 2023-09-22 2025-03-27 City University Of Hong Kong Methods of inhibiting klebsiella pneumoniae carbapenemase-2
WO2025119216A1 (zh) * 2023-12-04 2025-06-12 珠海联邦制药股份有限公司 硼酸类β-内酰胺酶抑制剂及其制备方法和应用
CN119119096B (zh) * 2024-09-09 2025-09-16 郑州药领医药科技有限公司 一种4-((4,4,5,5-四甲基-1,3,2-二氧硼杂环戊烷-2-基)甲基)哌啶-1-甲酸叔丁酯的合成方法

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