JP2021515015A5 - - Google Patents

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Publication number
JP2021515015A5
JP2021515015A5 JP2020546378A JP2020546378A JP2021515015A5 JP 2021515015 A5 JP2021515015 A5 JP 2021515015A5 JP 2020546378 A JP2020546378 A JP 2020546378A JP 2020546378 A JP2020546378 A JP 2020546378A JP 2021515015 A5 JP2021515015 A5 JP 2021515015A5
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JP
Japan
Prior art keywords
ray powder
powder diffraction
diffraction peaks
angles
crystal form
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020546378A
Other languages
English (en)
Japanese (ja)
Other versions
JP7423539B2 (ja
JP2021515015A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/021080 external-priority patent/WO2019173551A1/en
Publication of JP2021515015A publication Critical patent/JP2021515015A/ja
Publication of JP2021515015A5 publication Critical patent/JP2021515015A5/ja
Application granted granted Critical
Publication of JP7423539B2 publication Critical patent/JP7423539B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020546378A 2018-03-07 2019-03-07 Sgc刺激因子の結晶形態 Active JP7423539B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862639846P 2018-03-07 2018-03-07
US62/639,846 2018-03-07
PCT/US2019/021080 WO2019173551A1 (en) 2018-03-07 2019-03-07 Crystalline forms of an sgc stimulator

Publications (3)

Publication Number Publication Date
JP2021515015A JP2021515015A (ja) 2021-06-17
JP2021515015A5 true JP2021515015A5 (https=) 2022-03-14
JP7423539B2 JP7423539B2 (ja) 2024-01-29

Family

ID=65818696

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020546378A Active JP7423539B2 (ja) 2018-03-07 2019-03-07 Sgc刺激因子の結晶形態

Country Status (21)

Country Link
US (3) US11466015B2 (https=)
EP (1) EP3762389B1 (https=)
JP (1) JP7423539B2 (https=)
KR (1) KR102782810B1 (https=)
CN (1) CN111836812A (https=)
AU (1) AU2019231724B2 (https=)
BR (1) BR112020018212A2 (https=)
CA (1) CA3092683A1 (https=)
CL (5) CL2020002284A1 (https=)
CO (1) CO2020012493A2 (https=)
CR (1) CR20200458A (https=)
EA (1) EA202092109A1 (https=)
ES (1) ES2980256T3 (https=)
IL (1) IL276853B1 (https=)
MA (1) MA54638A (https=)
MX (5) MX2023004857A (https=)
PE (1) PE20210124A1 (https=)
PH (1) PH12020551394A1 (https=)
SG (1) SG11202008641WA (https=)
TW (1) TWI823903B (https=)
WO (1) WO2019173551A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019231724B2 (en) 2018-03-07 2024-06-27 Tisento Therapeutics Inc. Crystalline forms of an sGC stimulator
KR20250141845A (ko) * 2018-07-11 2025-09-29 티센토 쎄라퓨틱스 인크. 미토콘드리아 장애의 치료를 위한 sGC 자극제의 용도
US20230130739A1 (en) * 2020-03-26 2023-04-27 Cyclerion Therapeutics, Inc. DEUTERATED sGC STIMULATORS
CN118221651A (zh) * 2022-12-21 2024-06-21 广东东阳光药业股份有限公司 氟取代的吲唑化合物的晶型及其用途
AU2023412228A1 (en) * 2022-12-21 2025-07-03 Sunshine Lake Pharma Co., Ltd. Crystal form of fluorine-substituted indazole compound and use thereof

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DE19744026A1 (de) 1997-10-06 1999-04-08 Hoechst Marion Roussel De Gmbh Pyrazol-Derivate, ihre Herstellung und ihre Verwendung in Arzneimitteln
CZ302691B6 (cs) 1998-07-08 2011-09-07 Sanofi - Aventis Deutschland GmbH N-Arylamidová sloucenina, zpusob její prípravy, farmaceutický prostredek tuto slouceninu obsahující, tato sloucenina pro použití jako aktivátor a pro použití k terapii nebo profylaxi
DE19830430A1 (de) 1998-07-08 2000-01-13 Hoechst Marion Roussel De Gmbh Schwefelsubstituierte Sulfonylamino-carbonsäure-N-arylamide, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate
DE19834044A1 (de) 1998-07-29 2000-02-03 Bayer Ag Neue substituierte Pyrazolderivate
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GB9824310D0 (en) 1998-11-05 1998-12-30 Univ London Activators of soluble guanylate cyclase
DE19942809A1 (de) 1999-09-08 2001-03-15 Bayer Ag Verfahren zur Herstellung substituierter Pyrimidinderivate
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SI3507291T1 (sl) * 2016-09-02 2021-11-30 Cyclerion Therapeutics, Inc. Kondenzirani biciklični SGS stimulatorji
AU2019231724B2 (en) 2018-03-07 2024-06-27 Tisento Therapeutics Inc. Crystalline forms of an sGC stimulator

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