JP2022525759A5 - - Google Patents

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Publication number
JP2022525759A5
JP2022525759A5 JP2021555545A JP2021555545A JP2022525759A5 JP 2022525759 A5 JP2022525759 A5 JP 2022525759A5 JP 2021555545 A JP2021555545 A JP 2021555545A JP 2021555545 A JP2021555545 A JP 2021555545A JP 2022525759 A5 JP2022525759 A5 JP 2022525759A5
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JP
Japan
Prior art keywords
powder
crystal morphology
ray diffraction
morphology
angles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021555545A
Other languages
English (en)
Japanese (ja)
Other versions
JP7738482B2 (ja
JP2022525759A (ja
Filing date
Publication date
Priority claimed from PCT/CN2019/081985 external-priority patent/WO2020206623A1/en
Application filed filed Critical
Publication of JP2022525759A publication Critical patent/JP2022525759A/ja
Publication of JP2022525759A5 publication Critical patent/JP2022525759A5/ja
Priority to JP2025144862A priority Critical patent/JP2026004294A/ja
Application granted granted Critical
Publication of JP7738482B2 publication Critical patent/JP7738482B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021555545A 2019-04-10 2020-04-10 ピリダジノンtrpc阻害剤の結晶形態 Active JP7738482B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025144862A JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
PCT/CN2019/081985 WO2020206623A1 (en) 2019-04-10 2019-04-10 Crystal forms
CNPCT/CN2019/081985 2019-04-10
PCT/US2020/027689 WO2020210639A1 (en) 2019-04-10 2020-04-10 Crystal forms of a pyridazinone trpc inhibitor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025144862A Division JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Publications (3)

Publication Number Publication Date
JP2022525759A JP2022525759A (ja) 2022-05-19
JP2022525759A5 true JP2022525759A5 (https=) 2023-07-07
JP7738482B2 JP7738482B2 (ja) 2025-09-12

Family

ID=70482847

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021555545A Active JP7738482B2 (ja) 2019-04-10 2020-04-10 ピリダジノンtrpc阻害剤の結晶形態
JP2025144862A Pending JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025144862A Pending JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Country Status (10)

Country Link
US (1) US20220177455A1 (https=)
EP (1) EP3953352A1 (https=)
JP (2) JP7738482B2 (https=)
CN (2) CN114502552B (https=)
AU (1) AU2026201003A1 (https=)
BR (1) BR112021018221A2 (https=)
CA (1) CA3136652A1 (https=)
MA (1) MA55614A (https=)
MX (2) MX2021012313A (https=)
WO (2) WO2020206623A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3684364A4 (en) 2017-09-18 2021-06-02 Goldfinch Bio, Inc. PYRIDAZINONE AND METHOD OF USE THEREOF
MA71645A (fr) * 2018-09-18 2025-05-30 Goldfinch Bio, Inc. Pyridazinones et leurs procédés d'utilisation
US12576033B2 (en) * 2019-04-11 2026-03-17 Gfb (Abc), Llc Spray-dried formulation of a pyridazinone TRPC5 inhibitor
JP2022551580A (ja) * 2019-10-04 2022-12-12 ゴールドフィンチ バイオ,インク. 巣状分節性糸球体硬化症および糖尿病性腎症のバイオマーカーに基づく処置
JP7539545B2 (ja) * 2020-07-03 2024-08-23 武漢朗来科技発展有限公司 複素環化合物及びその使用
US20250122190A1 (en) * 2021-09-10 2025-04-17 Medshine Discovery Inc. Halogen-substituted pyridazinone compound and application thereof
US20250082655A1 (en) * 2022-01-27 2025-03-13 Wuhan Createrna Science And Technology Co., Ltd. Use of heterocyclic compound
WO2024027752A1 (zh) * 2022-08-05 2024-02-08 武汉朗来科技发展有限公司 包含杂环化合物的药物组合物及其制备方法和应用
WO2025250920A1 (en) 2024-05-31 2025-12-04 Gfb (Abc), Llc Pyridazinone phosphate compounds, pharmaceutical compositions, and medical uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP310798A0 (en) * 1998-04-22 1998-05-14 Soltec Research Pty Ltd Vehicle system for a composition comprising a piperidinopyrimidine derivative
US8633233B2 (en) * 2008-08-06 2014-01-21 Hydra Biosciences, Inc. Methods and compositions for treating anxiety
WO2016023830A1 (en) * 2014-08-11 2016-02-18 Hydra Biosciences, Inc. Pyrido[2,3-d]pyrimidine-2,4(1h,3h)-dione derivatives
EP3684364A4 (en) * 2017-09-18 2021-06-02 Goldfinch Bio, Inc. PYRIDAZINONE AND METHOD OF USE THEREOF
MA71645A (fr) * 2018-09-18 2025-05-30 Goldfinch Bio, Inc. Pyridazinones et leurs procédés d'utilisation

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