JP2021512953A5 - - Google Patents

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Publication number
JP2021512953A5
JP2021512953A5 JP2020564037A JP2020564037A JP2021512953A5 JP 2021512953 A5 JP2021512953 A5 JP 2021512953A5 JP 2020564037 A JP2020564037 A JP 2020564037A JP 2020564037 A JP2020564037 A JP 2020564037A JP 2021512953 A5 JP2021512953 A5 JP 2021512953A5
Authority
JP
Japan
Prior art keywords
substituted
pharmaceutically acceptable
amide
compound according
ester
Prior art date
Application number
JP2020564037A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2019152955A5 (https=
JP2021512953A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/016557 external-priority patent/WO2019152955A1/en
Publication of JP2021512953A publication Critical patent/JP2021512953A/ja
Publication of JP2021512953A5 publication Critical patent/JP2021512953A5/ja
Publication of JPWO2019152955A5 publication Critical patent/JPWO2019152955A5/ja
Priority to JP2024007282A priority Critical patent/JP2024054873A/ja
Pending legal-status Critical Current

Links

JP2020564037A 2018-02-02 2019-02-04 ゲムシタビンモノホスフェートの小分子薬物コンジュゲート Pending JP2021512953A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024007282A JP2024054873A (ja) 2018-02-02 2024-01-22 ゲムシタビンモノホスフェートの小分子薬物コンジュゲート

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862625820P 2018-02-02 2018-02-02
US62/625,820 2018-02-02
PCT/US2019/016557 WO2019152955A1 (en) 2018-02-02 2019-02-04 Small molecule drug conjugates of gemcitabine monophosphate

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024007282A Division JP2024054873A (ja) 2018-02-02 2024-01-22 ゲムシタビンモノホスフェートの小分子薬物コンジュゲート

Publications (3)

Publication Number Publication Date
JP2021512953A JP2021512953A (ja) 2021-05-20
JP2021512953A5 true JP2021512953A5 (https=) 2022-02-14
JPWO2019152955A5 JPWO2019152955A5 (https=) 2022-02-14

Family

ID=65494554

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020564037A Pending JP2021512953A (ja) 2018-02-02 2019-02-04 ゲムシタビンモノホスフェートの小分子薬物コンジュゲート
JP2024007282A Pending JP2024054873A (ja) 2018-02-02 2024-01-22 ゲムシタビンモノホスフェートの小分子薬物コンジュゲート

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024007282A Pending JP2024054873A (ja) 2018-02-02 2024-01-22 ゲムシタビンモノホスフェートの小分子薬物コンジュゲート

Country Status (17)

Country Link
US (1) US11760773B2 (https=)
EP (1) EP3746134A1 (https=)
JP (2) JP2021512953A (https=)
KR (1) KR20200118827A (https=)
CN (1) CN112135634A (https=)
AU (1) AU2019216531A1 (https=)
BR (1) BR112020015745A2 (https=)
CA (1) CA3091027A1 (https=)
CL (1) CL2020002022A1 (https=)
CO (1) CO2020010970A2 (https=)
EA (1) EA202091856A1 (https=)
IL (1) IL276436A (https=)
MX (1) MX2020008188A (https=)
PE (1) PE20210367A1 (https=)
PH (1) PH12020551182A1 (https=)
SG (1) SG11202007386RA (https=)
WO (1) WO2019152955A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20210367A1 (es) * 2018-02-02 2021-02-26 Maverix Oncology Inc Conjugados de farmacos de molecula pequena de monofosfato de gemcitabina

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