JP2020508300A5 - - Google Patents

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JP2020508300A5
JP2020508300A5 JP2019544606A JP2019544606A JP2020508300A5 JP 2020508300 A5 JP2020508300 A5 JP 2020508300A5 JP 2019544606 A JP2019544606 A JP 2019544606A JP 2019544606 A JP2019544606 A JP 2019544606A JP 2020508300 A5 JP2020508300 A5 JP 2020508300A5
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Japan
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optionally substituted
substituted
alkyl
pharmaceutically acceptable
acceptable salt
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JP2019544606A
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JP7316216B2 (ja
JP2020508300A (ja
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Priority claimed from PCT/US2018/018312 external-priority patent/WO2018152293A1/en
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JP2019544606A 2017-02-17 2018-02-15 5員アザ複素環を含有するデルタ-オピオイド受容体調節化合物、その使用方法及び製造方法 Active JP7316216B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762460407P 2017-02-17 2017-02-17
US62/460,407 2017-02-17
PCT/US2018/018312 WO2018152293A1 (en) 2017-02-17 2018-02-15 5-membered aza-heterocyclic containing delta-opioid receptor modulating compounds, methods of using and making the same

Publications (3)

Publication Number Publication Date
JP2020508300A JP2020508300A (ja) 2020-03-19
JP2020508300A5 true JP2020508300A5 (https=) 2021-03-25
JP7316216B2 JP7316216B2 (ja) 2023-07-27

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JP2019544606A Active JP7316216B2 (ja) 2017-02-17 2018-02-15 5員アザ複素環を含有するデルタ-オピオイド受容体調節化合物、その使用方法及び製造方法

Country Status (10)

Country Link
US (1) US11702408B2 (https=)
EP (1) EP3582779B1 (https=)
JP (1) JP7316216B2 (https=)
KR (1) KR20190129867A (https=)
CN (1) CN110520129A (https=)
AU (1) AU2018221148B2 (https=)
BR (1) BR112019016827A2 (https=)
CA (1) CA3052480A1 (https=)
IL (1) IL268414A (https=)
WO (1) WO2018152293A1 (https=)

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BR112019016827A2 (pt) 2017-02-17 2020-04-07 Trevena Inc compostos moduladores de receptor delta-opioide contendo aza-heterocíclico com 5 membros, métodos de uso e produção dos mesmos
WO2020113094A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
CN110117245B (zh) * 2019-06-21 2021-03-02 浙江师范大学 一种jak抑制剂中间体的合成方法
BR112022016941A2 (pt) * 2020-02-25 2022-10-25 Tes Pharma S R L Compostos heterocíclicos para a modulação de nr2f6

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