JP2021512889A5 - - Google Patents
Info
- Publication number
- JP2021512889A5 JP2021512889A5 JP2020542437A JP2020542437A JP2021512889A5 JP 2021512889 A5 JP2021512889 A5 JP 2021512889A5 JP 2020542437 A JP2020542437 A JP 2020542437A JP 2020542437 A JP2020542437 A JP 2020542437A JP 2021512889 A5 JP2021512889 A5 JP 2021512889A5
- Authority
- JP
- Japan
- Prior art keywords
- pyridine
- benzodiazole
- fluoro
- substituted
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862629377P | 2018-02-12 | 2018-02-12 | |
| US62/629,377 | 2018-02-12 | ||
| US201862673042P | 2018-05-17 | 2018-05-17 | |
| US62/673,042 | 2018-05-17 | ||
| US201862724421P | 2018-08-29 | 2018-08-29 | |
| US62/724,421 | 2018-08-29 | ||
| PCT/US2019/017529 WO2019157458A1 (en) | 2018-02-12 | 2019-02-11 | Somatostatin modulators and uses thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021512889A JP2021512889A (ja) | 2021-05-20 |
| JP2021512889A5 true JP2021512889A5 (https=) | 2022-02-21 |
| JP7365347B2 JP7365347B2 (ja) | 2023-10-19 |
Family
ID=67548490
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020542437A Active JP7365347B2 (ja) | 2018-02-12 | 2019-02-11 | ソマトスタチンモジュレーターおよびその使用 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US11608335B2 (https=) |
| EP (1) | EP3752498B1 (https=) |
| JP (1) | JP7365347B2 (https=) |
| MA (1) | MA51840A (https=) |
| WO (1) | WO2019157458A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3596062A4 (en) | 2017-03-16 | 2020-08-26 | Crinetics Pharmaceuticals, Inc. | SOMATOSTATIN MODULATORS AND THEIR USES |
| MA51840A (fr) | 2018-02-12 | 2021-05-19 | Crinetics Pharmaceuticals Inc | Modulateurs de somatostatine et leurs utilisations |
| SMT202500155T1 (it) | 2018-09-18 | 2025-05-12 | Crinetics Pharmaceuticals Inc | Modulatori della somatostatina e loro usi |
| TWI841768B (zh) | 2019-08-14 | 2024-05-11 | 美商克林提克斯醫藥股份有限公司 | 非肽生長抑制素(somatostatin)5型受體激動劑及其用途 |
| JP2024506716A (ja) * | 2021-02-17 | 2024-02-14 | クリネティックス ファーマシューティカルズ，インク． | 高インスリン血症の処置のためのソマトスタチン受容体５型アゴニスト |
| JP2024506715A (ja) | 2021-02-17 | 2024-02-14 | クリネティックス ファーマシューティカルズ，インク． | ソマトスタチンモジュレーターの結晶形態 |
| IL320483A (en) * | 2022-10-28 | 2025-06-01 | Basecamp Bio Inc | Somatostatin receptor 2 agonists and uses thereof |
| TW202440164A (zh) | 2022-12-13 | 2024-10-16 | 美商克林提克斯醫藥股份有限公司 | 生長抑素亞型-2受體（sst2r）靶向治療劑及其用途 |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6127343A (en) | 1996-05-14 | 2000-10-03 | Novo Nordisk A/S | Somatostatin agonists and antagonists |
| US6025372A (en) | 1997-04-04 | 2000-02-15 | Merck & Co., Inc. | Somatostatin agonists |
| FR2802206B1 (fr) | 1999-12-14 | 2005-04-22 | Sod Conseils Rech Applic | Derives de 4-aminopiperidine et leur utilisation en tant que medicament |
| US20060281764A1 (en) * | 2005-06-10 | 2006-12-14 | Gaul Michael D | Aminopyrimidines as kinase modulators |
| AU2007309708A1 (en) * | 2006-03-13 | 2008-05-02 | Merck Sharp & Dohme Corp. | Somatostatin agonists |
| WO2008019967A2 (en) | 2006-08-15 | 2008-02-21 | F. Hoffmann-La Roche Ag | Phenyl, pyridine and quinoline derivatives |
| WO2009051705A1 (en) | 2007-10-18 | 2009-04-23 | Merck & Co., Inc. | Substituted 1,2,4-oxadiazoles and analogs thereof as cb2 receptor modulators, useful in the treatment of pain, respiratory and non-respiratory diseases |
| JP2011526294A (ja) | 2008-06-25 | 2011-10-06 | エンビボ ファーマシューティカルズ インコーポレイテッド | ホスホジエステラーゼ１０阻害剤としての二置換フェニル化合物 |
| GB0818241D0 (en) | 2008-10-06 | 2008-11-12 | Cancer Res Technology | Compounds and their use |
| JP2013503846A (ja) | 2009-09-01 | 2013-02-04 | ファイザー・インク | ベンズイミダゾール誘導体 |
| AU2011256444B2 (en) | 2010-05-18 | 2014-07-10 | Merck Sharp & Dohme Corp. | Spiro isoxazoline compounds as SSTR5 antagonists |
| GB201008290D0 (en) | 2010-05-18 | 2010-06-30 | Syngenta Ltd | Chemical compounds |
| WO2014007228A1 (ja) * | 2012-07-03 | 2014-01-09 | 小野薬品工業株式会社 | ソマトスタチン受容体作動活性を有する化合物およびその医薬用途 |
| US9643951B2 (en) | 2013-09-30 | 2017-05-09 | Ono Pharmaceutical Co., Ltd. | Compound having somatostatin receptor agonistic activity and pharmaceutical use thereof |
| ES2675504T3 (es) | 2013-10-02 | 2018-07-11 | Kuraray Co., Ltd. | Composición de resina, lámina de múltiples capas, material de envasado y recipiente |
| IL264178B2 (en) * | 2016-07-14 | 2024-05-01 | Crinetics Pharmaceuticals Inc | Somatostatin modulators and uses thereof |
| AU2018219644A1 (en) | 2017-02-08 | 2019-08-29 | Ono Pharmaceutical Co., Ltd. | Compound having somatostatin receptor agonistic activity and pharmaceutical use thereof |
| EP3596062A4 (en) | 2017-03-16 | 2020-08-26 | Crinetics Pharmaceuticals, Inc. | SOMATOSTATIN MODULATORS AND THEIR USES |
| EP3658560A4 (en) | 2017-07-25 | 2021-01-06 | Crinetics Pharmaceuticals, Inc. | SOMATOSTAT IN MODULATORS AND USES THEREOF |
| MA51840A (fr) | 2018-02-12 | 2021-05-19 | Crinetics Pharmaceuticals Inc | Modulateurs de somatostatine et leurs utilisations |
| SMT202500155T1 (it) | 2018-09-18 | 2025-05-12 | Crinetics Pharmaceuticals Inc | Modulatori della somatostatina e loro usi |
| TWI841768B (zh) | 2019-08-14 | 2024-05-11 | 美商克林提克斯醫藥股份有限公司 | 非肽生長抑制素(somatostatin)5型受體激動劑及其用途 |
-
2019
- 2019-02-11 MA MA051840A patent/MA51840A/fr unknown
- 2019-02-11 JP JP2020542437A patent/JP7365347B2/ja active Active
- 2019-02-11 US US16/968,533 patent/US11608335B2/en active Active
- 2019-02-11 WO PCT/US2019/017529 patent/WO2019157458A1/en not_active Ceased
- 2019-02-11 EP EP19751144.7A patent/EP3752498B1/en active Active
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