JP2020502115A5 - - Google Patents
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- Publication number
- JP2020502115A5 JP2020502115A5 JP2019531707A JP2019531707A JP2020502115A5 JP 2020502115 A5 JP2020502115 A5 JP 2020502115A5 JP 2019531707 A JP2019531707 A JP 2019531707A JP 2019531707 A JP2019531707 A JP 2019531707A JP 2020502115 A5 JP2020502115 A5 JP 2020502115A5
- Authority
- JP
- Japan
- Prior art keywords
- haloalkyl
- alkyl
- formula
- cyano
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 150000001875 compounds Chemical class 0.000 claims description 18
- -1 cyano, formyl Chemical group 0.000 claims description 16
- 125000000217 alkyl group Chemical group 0.000 claims description 15
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 12
- 229910052736 halogen Inorganic materials 0.000 claims description 12
- 150000002367 halogens Chemical class 0.000 claims description 12
- 125000001424 substituent group Chemical group 0.000 claims description 10
- 241000607479 Yersinia pestis Species 0.000 claims description 8
- 229910052739 hydrogen Inorganic materials 0.000 claims description 8
- 239000001257 hydrogen Substances 0.000 claims description 8
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 8
- 238000000034 method Methods 0.000 claims description 8
- 239000000203 mixture Substances 0.000 claims description 8
- 125000003545 alkoxy group Chemical group 0.000 claims description 6
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims description 6
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 claims description 6
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims description 6
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 6
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 claims description 6
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 6
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 4
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 4
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 4
- ORTFAQDWJHRMNX-UHFFFAOYSA-N hydroxidooxidocarbon(.) Chemical group O[C]=O ORTFAQDWJHRMNX-UHFFFAOYSA-N 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 4
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 4
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims description 2
- 238000009472 formulation Methods 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 125000004458 methylaminocarbonyl group Chemical group [H]N(C(*)=O)C([H])([H])[H] 0.000 claims description 2
- 229910052760 oxygen Inorganic materials 0.000 claims description 2
- 229910052717 sulfur Inorganic materials 0.000 claims description 2
- 125000003830 C1- C4 alkylcarbonylamino group Chemical group 0.000 claims 1
- 125000001188 haloalkyl group Chemical group 0.000 description 8
- 125000000753 cycloalkyl group Chemical group 0.000 description 6
- 125000004439 haloalkylsulfanyl group Chemical group 0.000 description 5
- IAZDPXIOMUYVGZ-UHFFFAOYSA-N Dimethylsulphoxide Chemical compound CS(C)=O IAZDPXIOMUYVGZ-UHFFFAOYSA-N 0.000 description 3
- 241001465754 Metazoa Species 0.000 description 3
- 125000004453 alkoxycarbonyl group Chemical group 0.000 description 3
- 125000004438 haloalkoxy group Chemical group 0.000 description 3
- 241000339374 Thrips tabaci Species 0.000 description 2
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 description 2
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 2
- 125000000304 alkynyl group Chemical group 0.000 description 2
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 description 2
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 2
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 description 1
- 229920001817 Agar Polymers 0.000 description 1
- 241000196324 Embryophyta Species 0.000 description 1
- 244000020551 Helianthus annuus Species 0.000 description 1
- 235000003222 Helianthus annuus Nutrition 0.000 description 1
- 241001414989 Thysanoptera Species 0.000 description 1
- 239000008272 agar Substances 0.000 description 1
- 238000002405 diagnostic procedure Methods 0.000 description 1
- 238000001035 drying Methods 0.000 description 1
- 125000000262 haloalkenyl group Chemical group 0.000 description 1
- 208000029380 parasitic ectoparasitic infectious disease Diseases 0.000 description 1
- 239000011550 stock solution Substances 0.000 description 1
- 238000001356 surgical procedure Methods 0.000 description 1
- 239000012085 test solution Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201611042841 | 2016-12-15 | ||
| IN201611042841 | 2016-12-15 | ||
| PCT/EP2017/081968 WO2018108726A1 (en) | 2016-12-15 | 2017-12-08 | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020502115A JP2020502115A (ja) | 2020-01-23 |
| JP2020502115A5 true JP2020502115A5 (enExample) | 2021-01-21 |
| JP7113014B2 JP7113014B2 (ja) | 2022-08-04 |
Family
ID=60702699
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019531707A Active JP7113014B2 (ja) | 2016-12-15 | 2017-12-08 | 硫黄含有置換基を有する有害生物防除に活性な複素環式誘導体 |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US20190308982A1 (enExample) |
| EP (1) | EP3554242A1 (enExample) |
| JP (1) | JP7113014B2 (enExample) |
| CN (1) | CN110022682B (enExample) |
| BR (1) | BR112019012127A2 (enExample) |
| WO (1) | WO2018108726A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI793104B (zh) * | 2017-02-21 | 2023-02-21 | 瑞士商先正達合夥公司 | 具有含硫取代基的殺有害生物活性雜環衍生物 |
| JP7443357B2 (ja) | 2018-10-23 | 2024-03-05 | ビーエーエスエフ ソシエタス・ヨーロピア | 三環式の殺有害生物化合物 |
| WO2020161208A1 (en) * | 2019-02-06 | 2020-08-13 | Syngenta Crop Protection Ag | Herbicidal fused pyridazine compounds |
| WO2020161209A1 (en) * | 2019-02-06 | 2020-08-13 | Syngenta Crop Protection Ag | Herbicidal fused pyridazine compounds |
| JP7581336B2 (ja) | 2019-09-20 | 2024-11-12 | シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト | 硫黄及びスルホキシミン含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| WO2022013417A1 (en) | 2020-07-17 | 2022-01-20 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| WO2022017975A1 (en) | 2020-07-18 | 2022-01-27 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| EP4204422A1 (en) * | 2020-08-26 | 2023-07-05 | Syngenta Crop Protection AG | Process for the preparation of 2,2-difluoro-1,3-benzodioxole derivatives with sulfur containing substituents |
| PY2175588A (es) | 2020-09-02 | 2022-06-14 | Syngenta Crop Protection Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| TWI911299B (zh) | 2020-10-09 | 2026-01-11 | 瑞士商先正達農作物保護公司 | 用於製備5-(1-氰基環丙基)-吡啶-2-甲酸、酯、醯胺和腈之方法 |
| JP7644217B2 (ja) * | 2021-03-01 | 2025-03-11 | 日本農薬株式会社 | スルホンアミド基を有する縮合複素環化合物又はその塩類及び該化合物若しくはその塩類を含有する農園芸用殺虫剤又は動物用の外部若しくは内部寄生虫防除剤並びにそれらの使用方法 |
| JP2024520657A (ja) | 2021-06-02 | 2024-05-24 | シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト | スルホキシイミン含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| CN118339140B (zh) * | 2023-02-20 | 2024-09-27 | 住友化学株式会社 | 环丙烷羧酸酯化合物及其用途 |
| EP4680028A1 (en) | 2023-03-14 | 2026-01-21 | Syngenta Crop Protection AG | Control of pests resistant to insecticides |
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| CA1340685C (en) | 1988-07-29 | 1999-07-27 | Frederick Meins | Dna sequences encoding polypeptides having beta-1,3-glucanase activity |
| US5169629A (en) | 1988-11-01 | 1992-12-08 | Mycogen Corporation | Process of controlling lepidopteran pests, using bacillus thuringiensis isolate denoted b.t ps81gg |
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| DK0392225T3 (da) | 1989-03-24 | 2003-09-22 | Syngenta Participations Ag | Sygdomsresistente transgene planter |
| GB8910624D0 (en) | 1989-05-09 | 1989-06-21 | Ici Plc | Bacterial strains |
| CA2015951A1 (en) | 1989-05-18 | 1990-11-18 | Mycogen Corporation | Novel bacillus thuringiensis isolates active against lepidopteran pests, and genes encoding novel lepidopteran-active toxins |
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| US20110306639A1 (en) | 2008-11-25 | 2011-12-15 | Qin Zhaohai | Hydrocarbylidene nitrohydrozinecarboximidamides and a method for making the same, as well as their uses as an insecticide |
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| US10939682B2 (en) | 2013-07-02 | 2021-03-09 | Syngenta Participations Ag | Pesticidally active bi- or tricyclic heterocycles with sulfur containing substituents |
| TW201625522A (zh) | 2014-09-12 | 2016-07-16 | Nihon Nohyaku Co Ltd | 咪唑嗒化合物或其鹽類及含有該化合物之農園藝用殺蟲劑及其使用方法 |
| WO2016059145A1 (en) | 2014-10-16 | 2016-04-21 | Syngenta Participations Ag | Pesticidally active tetracyclic heterocyclic derivatives with sulphur containing substituents |
| ES2806598T3 (es) * | 2014-12-11 | 2021-02-18 | Syngenta Participations Ag | Derivados tetracíclicos activos como plaguicidas con sustituyentes que contienen azufre |
| UA122781C2 (uk) | 2014-12-17 | 2021-01-06 | Сінгента Партісіпейшнс Аг | Пестицидно активні гетероциклічні похідні з сірковмісними замісниками |
| JP2018052816A (ja) | 2014-12-26 | 2018-04-05 | 日本農薬株式会社 | シクロアルキル基を有する縮合複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| BR112017015514B1 (pt) * | 2015-01-19 | 2022-08-30 | Syngenta Participations Ag | Derivados policíclicos ativos com substituintes contendo enxofre ativo em termos pesticidas, composição pesticida e métodos para controle de pragas e proteção de sementes do ataque por pragas |
| TWI696612B (zh) * | 2015-01-29 | 2020-06-21 | 日商日本農藥股份有限公司 | 具有環烷基吡啶基的稠合雜環化合物或其鹽類及含有該化合物的農園藝用殺蟲劑以及其使用方法 |
| JP6779225B2 (ja) * | 2015-03-12 | 2020-11-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| US10738045B2 (en) | 2015-11-23 | 2020-08-11 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur and cyclopropyl containing substituents |
-
2017
- 2017-12-08 BR BR112019012127-7A patent/BR112019012127A2/pt not_active Application Discontinuation
- 2017-12-08 EP EP17816655.9A patent/EP3554242A1/en active Pending
- 2017-12-08 US US16/470,165 patent/US20190308982A1/en not_active Abandoned
- 2017-12-08 JP JP2019531707A patent/JP7113014B2/ja active Active
- 2017-12-08 CN CN201780074392.8A patent/CN110022682B/zh active Active
- 2017-12-08 WO PCT/EP2017/081968 patent/WO2018108726A1/en not_active Ceased
-
2021
- 2021-09-07 US US17/468,051 patent/US12421237B2/en active Active