JP2020502115A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2020502115A5 JP2020502115A5 JP2019531707A JP2019531707A JP2020502115A5 JP 2020502115 A5 JP2020502115 A5 JP 2020502115A5 JP 2019531707 A JP2019531707 A JP 2019531707A JP 2019531707 A JP2019531707 A JP 2019531707A JP 2020502115 A5 JP2020502115 A5 JP 2020502115A5
- Authority
- JP
- Japan
- Prior art keywords
- haloalkyl
- alkyl
- formula
- cyano
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 18
- -1 cyano, formyl Chemical group 0.000 claims description 16
- 125000000217 alkyl group Chemical group 0.000 claims description 15
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 12
- 229910052736 halogen Inorganic materials 0.000 claims description 12
- 150000002367 halogens Chemical class 0.000 claims description 12
- 125000001424 substituent group Chemical group 0.000 claims description 10
- 241000607479 Yersinia pestis Species 0.000 claims description 8
- 229910052739 hydrogen Inorganic materials 0.000 claims description 8
- 239000001257 hydrogen Substances 0.000 claims description 8
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 8
- 238000000034 method Methods 0.000 claims description 8
- 239000000203 mixture Substances 0.000 claims description 8
- 125000003545 alkoxy group Chemical group 0.000 claims description 6
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims description 6
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 claims description 6
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims description 6
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 6
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 claims description 6
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 6
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 4
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 4
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 4
- ORTFAQDWJHRMNX-UHFFFAOYSA-N hydroxidooxidocarbon(.) Chemical group O[C]=O ORTFAQDWJHRMNX-UHFFFAOYSA-N 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 4
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 4
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims description 2
- 238000009472 formulation Methods 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 125000004458 methylaminocarbonyl group Chemical group [H]N(C(*)=O)C([H])([H])[H] 0.000 claims description 2
- 229910052760 oxygen Inorganic materials 0.000 claims description 2
- 229910052717 sulfur Inorganic materials 0.000 claims description 2
- 125000003830 C1- C4 alkylcarbonylamino group Chemical group 0.000 claims 1
- 125000001188 haloalkyl group Chemical group 0.000 description 8
- 125000000753 cycloalkyl group Chemical group 0.000 description 6
- 125000004439 haloalkylsulfanyl group Chemical group 0.000 description 5
- IAZDPXIOMUYVGZ-UHFFFAOYSA-N Dimethylsulphoxide Chemical compound CS(C)=O IAZDPXIOMUYVGZ-UHFFFAOYSA-N 0.000 description 3
- 241001465754 Metazoa Species 0.000 description 3
- 125000004453 alkoxycarbonyl group Chemical group 0.000 description 3
- 125000004438 haloalkoxy group Chemical group 0.000 description 3
- 241000339374 Thrips tabaci Species 0.000 description 2
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 description 2
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 2
- 125000000304 alkynyl group Chemical group 0.000 description 2
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 description 2
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 2
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 description 1
- 229920001817 Agar Polymers 0.000 description 1
- 241000196324 Embryophyta Species 0.000 description 1
- 244000020551 Helianthus annuus Species 0.000 description 1
- 235000003222 Helianthus annuus Nutrition 0.000 description 1
- 241001414989 Thysanoptera Species 0.000 description 1
- 239000008272 agar Substances 0.000 description 1
- 238000002405 diagnostic procedure Methods 0.000 description 1
- 238000001035 drying Methods 0.000 description 1
- 125000000262 haloalkenyl group Chemical group 0.000 description 1
- 208000029380 parasitic ectoparasitic infectious disease Diseases 0.000 description 1
- 239000011550 stock solution Substances 0.000 description 1
- 238000001356 surgical procedure Methods 0.000 description 1
- 239000012085 test solution Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201611042841 | 2016-12-15 | ||
| IN201611042841 | 2016-12-15 | ||
| PCT/EP2017/081968 WO2018108726A1 (en) | 2016-12-15 | 2017-12-08 | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020502115A JP2020502115A (ja) | 2020-01-23 |
| JP2020502115A5 true JP2020502115A5 (enExample) | 2021-01-21 |
| JP7113014B2 JP7113014B2 (ja) | 2022-08-04 |
Family
ID=60702699
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019531707A Active JP7113014B2 (ja) | 2016-12-15 | 2017-12-08 | 硫黄含有置換基を有する有害生物防除に活性な複素環式誘導体 |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US20190308982A1 (enExample) |
| EP (1) | EP3554242A1 (enExample) |
| JP (1) | JP7113014B2 (enExample) |
| CN (1) | CN110022682B (enExample) |
| BR (1) | BR112019012127A2 (enExample) |
| WO (1) | WO2018108726A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI793104B (zh) * | 2017-02-21 | 2023-02-21 | 瑞士商先正達合夥公司 | 具有含硫取代基的殺有害生物活性雜環衍生物 |
| US12134616B2 (en) | 2018-10-23 | 2024-11-05 | Basf Se | Tricyclic pesticidal compounds |
| WO2020161209A1 (en) * | 2019-02-06 | 2020-08-13 | Syngenta Crop Protection Ag | Herbicidal fused pyridazine compounds |
| WO2020161208A1 (en) * | 2019-02-06 | 2020-08-13 | Syngenta Crop Protection Ag | Herbicidal fused pyridazine compounds |
| US12503461B2 (en) | 2019-09-20 | 2025-12-23 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur and sulfoximine containing substituents |
| WO2022013417A1 (en) | 2020-07-17 | 2022-01-20 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| WO2022017975A1 (en) | 2020-07-18 | 2022-01-27 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| JP2023538755A (ja) | 2020-08-26 | 2023-09-11 | シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト | 硫黄含有置換基を有する２，２－ジフルオロ－１，３－ベンゾジオキソール誘導体の調製のための方法 |
| PY2175588A (es) | 2020-09-02 | 2022-06-14 | Syngenta Crop Protection Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| TWI911299B (zh) * | 2020-10-09 | 2026-01-11 | 瑞士商先正達農作物保護公司 | 用於製備5-(1-氰基環丙基)-吡啶-2-甲酸、酯、醯胺和腈之方法 |
| EP4303214A4 (en) * | 2021-03-01 | 2025-02-19 | Nihon Nohyaku Co., Ltd. | CONDENSED HETEROCYCLIC COMPOUND HAVING A SULFONAMIDE GROUP OR SALT THEREOF, AGRICULTURAL/HORTICULTURAL PESTICIDE AND EXTERNAL OR INTERNAL ANIMAL PARASITE CONTAINING SAID COMPOUND OR SALT THEREOF, AND METHOD OF USING THE SAME |
| JP2024520657A (ja) | 2021-06-02 | 2024-05-24 | シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト | スルホキシイミン含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| WO2024071440A1 (ja) * | 2023-02-20 | 2024-04-04 | 住友化学株式会社 | シクロプロパンカルボン酸エステル化合物及びその用途 |
| WO2024189139A1 (en) | 2023-03-14 | 2024-09-19 | Syngenta Crop Protection Ag | Control of pests resistant to insecticides |
Family Cites Families (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR8600161A (pt) | 1985-01-18 | 1986-09-23 | Plant Genetic Systems Nv | Gene quimerico,vetores de plasmidio hibrido,intermediario,processo para controlar insetos em agricultura ou horticultura,composicao inseticida,processo para transformar celulas de plantas para expressar uma toxina de polipeptideo produzida por bacillus thuringiensis,planta,semente de planta,cultura de celulas e plasmidio |
| CA1340685C (en) | 1988-07-29 | 1999-07-27 | Frederick Meins | Dna sequences encoding polypeptides having beta-1,3-glucanase activity |
| US5169629A (en) | 1988-11-01 | 1992-12-08 | Mycogen Corporation | Process of controlling lepidopteran pests, using bacillus thuringiensis isolate denoted b.t ps81gg |
| CA2005658A1 (en) | 1988-12-19 | 1990-06-19 | Eliahu Zlotkin | Insecticidal toxins, genes encoding these toxins, antibodies binding to them and transgenic plant cells and plants expressing these toxins |
| ES2199931T3 (es) | 1989-03-24 | 2004-03-01 | Syngenta Participations Ag | Plantas transgenicas resistentes a enfermedades. |
| GB8910624D0 (en) | 1989-05-09 | 1989-06-21 | Ici Plc | Bacterial strains |
| CA2015951A1 (en) | 1989-05-18 | 1990-11-18 | Mycogen Corporation | Novel bacillus thuringiensis isolates active against lepidopteran pests, and genes encoding novel lepidopteran-active toxins |
| EP0427529B1 (en) | 1989-11-07 | 1995-04-19 | Pioneer Hi-Bred International, Inc. | Larvicidal lectins and plant insect resistance based thereon |
| US5639949A (en) | 1990-08-20 | 1997-06-17 | Ciba-Geigy Corporation | Genes for the synthesis of antipathogenic substances |
| UA48104C2 (uk) | 1991-10-04 | 2002-08-15 | Новартіс Аг | Фрагмент днк, який містить послідовність,що кодує інсектицидний протеїн, оптимізовану для кукурудзи,фрагмент днк, який забезпечує направлену бажану для серцевини стебла експресію зв'язаного з нею структурного гена в рослині, фрагмент днк, який забезпечує специфічну для пилку експресію зв`язаного з нею структурного гена в рослині, рекомбінантна молекула днк, спосіб одержання оптимізованої для кукурудзи кодуючої послідовності інсектицидного протеїну, спосіб захисту рослин кукурудзи щонайменше від однієї комахи-шкідника |
| US5530195A (en) | 1994-06-10 | 1996-06-25 | Ciba-Geigy Corporation | Bacillus thuringiensis gene encoding a toxin active against insects |
| US5631072A (en) | 1995-03-10 | 1997-05-20 | Avondale Incorporated | Method and means for increasing efficacy and wash durability of insecticide treated fabric |
| EP1114030B1 (en) | 1998-09-15 | 2005-06-01 | Syngenta Participations AG | Pyridine ketones useful as herbicides |
| KR100581163B1 (ko) | 2000-08-25 | 2006-05-22 | 신젠타 파티서페이션즈 아게 | 하이브리드 바실러스 튜린지엔시스 독소, 이를 암호화하는 핵산 및 이를 사용한 해충의 방제방법 |
| AU2002345250A1 (en) | 2001-06-22 | 2003-01-08 | Syngenta Participations Ag | Plant disease resistance genes |
| US7230167B2 (en) | 2001-08-31 | 2007-06-12 | Syngenta Participations Ag | Modified Cry3A toxins and nucleic acid sequences coding therefor |
| EP1439752B1 (en) | 2001-10-25 | 2005-08-24 | Siamdutch Mosquito Netting Company Limited | Treatment of fabric materials with an insecticide |
| AU2002361696A1 (en) | 2001-12-17 | 2003-06-30 | Syngenta Participations Ag | Novel corn event |
| US20050132500A1 (en) | 2003-12-22 | 2005-06-23 | Basf Aktiengesellschaft | Composition for impregnation of fibers, fabrics and nettings imparting a protective activity against pests |
| DK2256112T3 (en) | 2004-02-18 | 2016-03-21 | Ishihara Sangyo Kaisha | Anthranilamides, process for their production and insecticides containing the same |
| DE102004023894A1 (de) | 2004-05-12 | 2005-12-08 | Basf Ag | Verfahren zur Behandlung von flexiblen Substraten |
| JP2008505167A (ja) | 2004-07-05 | 2008-02-21 | アステックス、セラピューティックス、リミテッド | 医薬組成物 |
| DE102005007160A1 (de) | 2005-02-16 | 2006-08-24 | Basf Ag | Pyrazolcarbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| DE102005020889A1 (de) | 2005-05-04 | 2006-11-09 | Fritz Blanke Gmbh & Co.Kg | Verfahren zur antimikrobiellen Ausrüstung von textilen Flächengebilden |
| KR20080018934A (ko) | 2005-06-03 | 2008-02-28 | 바스프 악티엔게젤샤프트 | 해충에 대한 보호 활성을 제공하는 섬유, 직물 및 네팅함침용 조성물 |
| BRPI0617076B1 (pt) | 2005-09-02 | 2021-07-06 | Nissan Chemical Corporation | Composto benzamida substituída por isoxazolina da fórmula (1) ou sal do mesmo; composto benzamida substituido por 4-hidroxiiminametila da fórmula (2) ou sal do mesmo; pesticida; agente agroquímico; parasiticida interno ou externo para mamíferos ou aves; inseticida ou acaricida |
| ATE489372T1 (de) | 2005-10-25 | 2010-12-15 | Syngenta Participations Ag | Als mikrobiozide geeignete heterocyclische amidderivate |
| WO2007090739A1 (de) | 2006-02-03 | 2007-08-16 | Basf Se | Verfahren zum behandeln von substraten |
| WO2008128968A1 (en) | 2007-04-19 | 2008-10-30 | Novartis Ag | Nicotinic acid derivatives as modulators of metabotropic glutamate receptor-5 |
| EP2158354B1 (en) | 2007-06-12 | 2012-04-04 | Basf Se | Aqueous formulation and process for the impregnation of non-living-materials imparting a protective activity against pests |
| JP5369854B2 (ja) | 2008-04-21 | 2013-12-18 | 住友化学株式会社 | 有害節足動物防除組成物および縮合複素環化合物 |
| EP2216324B1 (en) | 2008-11-25 | 2013-03-13 | Qin, ZhaoHai | Condensed amino nitroguanidine compounds, synthesis and use as botanical insecticides thereof |
| CN102414195B (zh) | 2009-04-28 | 2014-11-12 | 住友化学株式会社 | 稠合的杂环化合物及其用途 |
| TW201234965A (en) | 2010-12-24 | 2012-09-01 | Sumitomo Chemical Co | Fused heterocyclic compound and use for pest control thereof |
| TWI528899B (zh) | 2010-12-29 | 2016-04-11 | 杜邦股份有限公司 | 中離子性殺蟲劑 |
| TWI545119B (zh) | 2011-08-04 | 2016-08-11 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| UY35421A (es) * | 2013-03-15 | 2014-10-31 | Nihon Nohyaku Co Ltd | Compuesto heterocíclico condensado o su sal, insecticida agrícola u hortícola que comprende el comp uesto y método de uso del insecticida |
| WO2015000715A1 (en) * | 2013-07-02 | 2015-01-08 | Syngenta Participations Ag | Pesticidally active bi- or tricyclic heterocycles with sulfur containing substituents |
| WO2016039441A1 (ja) | 2014-09-12 | 2016-03-17 | 日本農薬株式会社 | イミダゾピリダジン化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| CN106795167B (zh) | 2014-10-16 | 2021-02-09 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性的四环杂环衍生物 |
| BR112017012232B1 (pt) * | 2014-12-11 | 2021-08-17 | Syngenta Participations Ag | Derivados tetraciclicos ativos em termos pesticidas com substituintes contendo enxofre |
| RS60709B1 (sr) | 2014-12-17 | 2020-09-30 | Syngenta Participations Ag | Pesticidno aktivni heterociklični derivati sa supstituentima koji sadrže sumpor |
| JP2018052816A (ja) * | 2014-12-26 | 2018-04-05 | 日本農薬株式会社 | シクロアルキル基を有する縮合複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| ES2924890T3 (es) | 2015-01-19 | 2022-10-11 | Syngenta Participations Ag | Derivados policíclicos activos como plaguicidas con sustituyentes que contienen azufre |
| TWI696612B (zh) * | 2015-01-29 | 2020-06-21 | 日商日本農藥股份有限公司 | 具有環烷基吡啶基的稠合雜環化合物或其鹽類及含有該化合物的農園藝用殺蟲劑以及其使用方法 |
| BR112017019371A2 (pt) * | 2015-03-12 | 2018-07-03 | Syngenta Participations Ag | derivados tetracíclicos ativos em termos pesticidas com substituintes contendo enxofre |
| BR112018010347A2 (pt) | 2015-11-23 | 2018-12-04 | Syngenta Participations Ag | derivados heterocíclicos ativos em termos pesticidas com substituintes contendo enxofre e ciclopropila |
-
2017
- 2017-12-08 JP JP2019531707A patent/JP7113014B2/ja active Active
- 2017-12-08 WO PCT/EP2017/081968 patent/WO2018108726A1/en not_active Ceased
- 2017-12-08 EP EP17816655.9A patent/EP3554242A1/en active Pending
- 2017-12-08 US US16/470,165 patent/US20190308982A1/en not_active Abandoned
- 2017-12-08 BR BR112019012127-7A patent/BR112019012127A2/pt not_active Application Discontinuation
- 2017-12-08 CN CN201780074392.8A patent/CN110022682B/zh active Active
-
2021
- 2021-09-07 US US17/468,051 patent/US12421237B2/en active Active