JP2018509418A5 - - Google Patents
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- Publication number
- JP2018509418A5 JP2018509418A5 JP2017548037A JP2017548037A JP2018509418A5 JP 2018509418 A5 JP2018509418 A5 JP 2018509418A5 JP 2017548037 A JP2017548037 A JP 2017548037A JP 2017548037 A JP2017548037 A JP 2017548037A JP 2018509418 A5 JP2018509418 A5 JP 2018509418A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- haloalkyl
- halogen
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 229910052736 halogen Inorganic materials 0.000 claims description 62
- 150000002367 halogens Chemical group 0.000 claims description 62
- 125000000217 alkyl group Chemical group 0.000 claims description 60
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 50
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 50
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 46
- 125000001424 substituent group Chemical group 0.000 claims description 41
- -1 C 2 -C 6 haloalkynyl Chemical group 0.000 claims description 34
- 150000001875 compounds Chemical class 0.000 claims description 33
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 28
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 26
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 25
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 24
- 229910052739 hydrogen Inorganic materials 0.000 claims description 24
- 239000001257 hydrogen Substances 0.000 claims description 24
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 24
- 229910052757 nitrogen Inorganic materials 0.000 claims description 24
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 22
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 22
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 22
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 18
- 229910052760 oxygen Inorganic materials 0.000 claims description 18
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 18
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 16
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims description 16
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 16
- 239000001301 oxygen Chemical group 0.000 claims description 16
- 125000004122 cyclic group Chemical group 0.000 claims description 14
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims description 14
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 12
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 10
- CYRMSUTZVYGINF-UHFFFAOYSA-N trichlorofluoromethane Chemical group FC(Cl)(Cl)Cl CYRMSUTZVYGINF-UHFFFAOYSA-N 0.000 claims description 10
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 claims description 8
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 claims description 8
- 150000001412 amines Chemical group 0.000 claims description 8
- 125000001188 haloalkyl group Chemical group 0.000 claims description 8
- 229910052717 sulfur Inorganic materials 0.000 claims description 8
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims description 7
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims description 7
- 238000000034 method Methods 0.000 claims description 7
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 claims description 6
- 125000004740 (C1-C6) haloalkylsulfanyl group Chemical group 0.000 claims description 6
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 6
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- 125000003118 aryl group Chemical group 0.000 claims description 6
- 239000011593 sulfur Chemical group 0.000 claims description 6
- TVEXGJYMHHTVKP-UHFFFAOYSA-N 6-oxabicyclo[3.2.1]oct-3-en-7-one Chemical compound C1C2C(=O)OC1C=CC2 TVEXGJYMHHTVKP-UHFFFAOYSA-N 0.000 claims description 4
- 125000005842 heteroatom Chemical group 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 4
- 125000004434 sulfur atom Chemical group 0.000 claims description 4
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims description 4
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims description 3
- 229920006395 saturated elastomer Polymers 0.000 claims description 3
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000002837 carbocyclic group Chemical group 0.000 claims description 2
- 229910052799 carbon Inorganic materials 0.000 claims description 2
- 125000004432 carbon atom Chemical group C* 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 2
- 125000000623 heterocyclic group Chemical group 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 230000000361 pesticidal effect Effects 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- 125000004766 (C3-C6) cyclohaloalkyl group Chemical group 0.000 claims 2
- 125000003342 alkenyl group Chemical group 0.000 claims 2
- 125000000475 sulfinyl group Chemical group [*:2]S([*:1])=O 0.000 claims 2
- 239000002671 adjuvant Substances 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 description 29
- 125000004414 alkyl thio group Chemical group 0.000 description 14
- 125000000232 haloalkynyl group Chemical group 0.000 description 11
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 10
- 125000000753 cycloalkyl group Chemical group 0.000 description 9
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 5
- 125000004995 haloalkylthio group Chemical group 0.000 description 5
- 125000005347 halocycloalkyl group Chemical group 0.000 description 5
- 0 *C(N1*)=CC(N=C(*2)I)=C2C1=O Chemical compound *C(N1*)=CC(N=C(*2)I)=C2C1=O 0.000 description 2
- 241001465754 Metazoa Species 0.000 description 2
- 125000005161 aryl oxy carbonyl group Chemical group 0.000 description 2
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 description 2
- 241000256118 Aedes aegypti Species 0.000 description 1
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 description 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 description 1
- 125000005169 cycloalkylcarbonylamino group Chemical group 0.000 description 1
- 238000003745 diagnosis Methods 0.000 description 1
- 125000004438 haloalkoxy group Chemical group 0.000 description 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 1
- 238000003359 percent control normalization Methods 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15158762.3 | 2015-03-12 | ||
| EP15158762 | 2015-03-12 | ||
| EP15179249 | 2015-07-31 | ||
| EP15179249.6 | 2015-07-31 | ||
| PCT/EP2016/054757 WO2016142326A1 (en) | 2015-03-12 | 2016-03-07 | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018509418A JP2018509418A (ja) | 2018-04-05 |
| JP2018509418A5 true JP2018509418A5 (enExample) | 2019-04-18 |
| JP6774955B2 JP6774955B2 (ja) | 2020-10-28 |
Family
ID=55538187
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017548037A Active JP6774955B2 (ja) | 2015-03-12 | 2016-03-07 | 硫黄含有置換基を有する殺有害生物的に活性な四環式誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10323031B2 (enExample) |
| EP (1) | EP3268365B8 (enExample) |
| JP (1) | JP6774955B2 (enExample) |
| CN (2) | CN111646989A (enExample) |
| BR (1) | BR112017019372B1 (enExample) |
| ES (1) | ES2731078T3 (enExample) |
| WO (1) | WO2016142326A1 (enExample) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6779225B2 (ja) * | 2015-03-12 | 2020-11-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| JP2018524337A (ja) * | 2015-07-01 | 2018-08-30 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| CN107735396B (zh) * | 2015-07-01 | 2021-03-02 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性多环衍生物 |
| BR112018008440B1 (pt) * | 2015-10-26 | 2021-12-21 | Bayer Cropscience Aktiengesellschaft | Derivados de heterociclo bicíclico fusionado como pesticidas |
| WO2017155103A1 (ja) | 2016-03-10 | 2017-09-14 | 日産化学工業株式会社 | 縮合複素環化合物及び有害生物防除剤 |
| JP7077314B2 (ja) * | 2016-10-27 | 2022-05-30 | シンジェンタ パーティシペーションズ アーゲー | 硫黄およびヒドロキシルアミン置換基を有する有害生物防除的に活性な複素環式誘導体 |
| CN110248938A (zh) | 2016-11-23 | 2019-09-17 | 拜耳作物科学股份公司 | 用作农药的2-[3-(烷基磺酰基)-2h-吲唑-2-基]-3h-咪唑并[4,5-b]吡啶衍生物和类似化合物 |
| KR102515694B1 (ko) | 2017-01-10 | 2023-03-29 | 바이엘 악티엔게젤샤프트 | 해충 방제제로서의 헤테로사이클 유도체 |
| BR112019014270B1 (pt) | 2017-01-10 | 2023-12-26 | Bayer Cropscience Aktiengesellschaft | Derivados de heterociclo, seus usos, formulação agroquímica, e método para controlar pragas animais |
| CN110198942B (zh) * | 2017-01-24 | 2022-04-15 | 住友化学株式会社 | 稠合杂环化合物及含有其的组合物 |
| WO2018138050A1 (de) | 2017-01-26 | 2018-08-02 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| EP3672966B1 (de) | 2017-08-22 | 2022-09-21 | Bayer Aktiengesellschaft | Heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CN111433215B (zh) | 2017-10-04 | 2023-10-03 | 拜耳公司 | 用作害虫防治剂的杂环化合物的衍生物 |
| CN108048372B (zh) * | 2018-01-30 | 2021-07-02 | 西南大学 | 一种短小芽孢杆菌及其防治蚕核型多角体病毒感染的应用 |
| ES2906077T3 (es) | 2018-02-21 | 2022-04-13 | Bayer Ag | Derivados de heterociclos bicíclicos condensados como pesticidas |
| WO2019175046A1 (de) | 2018-03-12 | 2019-09-19 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| KR102808245B1 (ko) | 2018-06-06 | 2025-05-14 | 신젠타 크롭 프로텍션 아게 | 설폭시민 함유 치환체를 갖는 살충 활성 헤테로사이클릭 유도체 |
| JP7353310B2 (ja) | 2018-06-26 | 2023-09-29 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| WO2020173861A1 (de) | 2019-02-26 | 2020-09-03 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CN115702149B (zh) | 2020-04-30 | 2025-08-19 | 先正达农作物保护股份公司 | 具有含硫取代基的杀有害生物活性的杂环衍生物 |
| US20230247994A1 (en) | 2020-07-02 | 2023-08-10 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| WO2023017094A1 (en) | 2021-08-10 | 2023-02-16 | Syngenta Crop Protection Ag | 2,2-difluoro-5h-[1,3]dioxolo[4,5-f]isoindol-7-one derivatives as pesticides |
| EP4680028A1 (en) | 2023-03-14 | 2026-01-21 | Syngenta Crop Protection AG | Control of pests resistant to insecticides |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3445299A1 (de) * | 1984-12-12 | 1986-06-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue imidazoderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
| US8853238B2 (en) * | 2010-12-24 | 2014-10-07 | Sumitomo Chemical Company, Limited | Fused heterocyclic compound and use thereof for pest control |
| TWI545119B (zh) * | 2011-08-04 | 2016-08-11 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| HUE049733T2 (hu) * | 2013-07-02 | 2020-10-28 | Syngenta Participations Ag | Növényvédõszerként aktív biciklusos vagy triciklusos heterociklusok kéntartalmú szubsztituensekkel |
| WO2016023954A2 (en) * | 2014-08-12 | 2016-02-18 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| US10308650B2 (en) * | 2014-12-11 | 2019-06-04 | Syngenta Participations Ag | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
| BR112017014061B1 (pt) * | 2014-12-29 | 2021-07-20 | Syngenta Participations Ag | Composto da formula i, composição pesticida, método para controle de pragas e método para a proteção de material de propagação de plantas a partir do mesmo |
| JP6779225B2 (ja) * | 2015-03-12 | 2020-11-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| WO2017133994A1 (en) * | 2016-02-04 | 2017-08-10 | Syngenta Participations Ag | Pesticidally active derivatives with sulfur and cyclopropyl containing substituents |
-
2016
- 2016-03-07 CN CN202010494058.1A patent/CN111646989A/zh active Pending
- 2016-03-07 CN CN201680015190.1A patent/CN107428751B/zh active Active
- 2016-03-07 ES ES16710116T patent/ES2731078T3/es active Active
- 2016-03-07 JP JP2017548037A patent/JP6774955B2/ja active Active
- 2016-03-07 WO PCT/EP2016/054757 patent/WO2016142326A1/en not_active Ceased
- 2016-03-07 US US15/554,283 patent/US10323031B2/en active Active
- 2016-03-07 BR BR112017019372-8A patent/BR112017019372B1/pt not_active IP Right Cessation
- 2016-03-07 EP EP16710116.1A patent/EP3268365B8/en active Active