JP2018509418A5 - - Google Patents
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- Publication number
- JP2018509418A5 JP2018509418A5 JP2017548037A JP2017548037A JP2018509418A5 JP 2018509418 A5 JP2018509418 A5 JP 2018509418A5 JP 2017548037 A JP2017548037 A JP 2017548037A JP 2017548037 A JP2017548037 A JP 2017548037A JP 2018509418 A5 JP2018509418 A5 JP 2018509418A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- haloalkyl
- halogen
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 229910052736 halogen Inorganic materials 0.000 claims description 62
- 150000002367 halogens Chemical group 0.000 claims description 62
- 125000000217 alkyl group Chemical group 0.000 claims description 60
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 50
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 50
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 46
- 125000001424 substituent group Chemical group 0.000 claims description 41
- -1 C 2 -C 6 haloalkynyl Chemical group 0.000 claims description 34
- 150000001875 compounds Chemical class 0.000 claims description 33
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 28
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 26
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 25
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 24
- 229910052739 hydrogen Inorganic materials 0.000 claims description 24
- 239000001257 hydrogen Substances 0.000 claims description 24
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 24
- 229910052757 nitrogen Inorganic materials 0.000 claims description 24
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 22
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 22
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 22
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 18
- 229910052760 oxygen Inorganic materials 0.000 claims description 18
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 18
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 16
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims description 16
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 16
- 239000001301 oxygen Chemical group 0.000 claims description 16
- 125000004122 cyclic group Chemical group 0.000 claims description 14
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims description 14
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 12
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 10
- CYRMSUTZVYGINF-UHFFFAOYSA-N trichlorofluoromethane Chemical group FC(Cl)(Cl)Cl CYRMSUTZVYGINF-UHFFFAOYSA-N 0.000 claims description 10
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 claims description 8
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 claims description 8
- 150000001412 amines Chemical group 0.000 claims description 8
- 125000001188 haloalkyl group Chemical group 0.000 claims description 8
- 229910052717 sulfur Inorganic materials 0.000 claims description 8
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims description 7
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims description 7
- 238000000034 method Methods 0.000 claims description 7
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 claims description 6
- 125000004740 (C1-C6) haloalkylsulfanyl group Chemical group 0.000 claims description 6
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 6
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- 125000003118 aryl group Chemical group 0.000 claims description 6
- 239000011593 sulfur Chemical group 0.000 claims description 6
- TVEXGJYMHHTVKP-UHFFFAOYSA-N 6-oxabicyclo[3.2.1]oct-3-en-7-one Chemical compound C1C2C(=O)OC1C=CC2 TVEXGJYMHHTVKP-UHFFFAOYSA-N 0.000 claims description 4
- 125000005842 heteroatom Chemical group 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 4
- 125000004434 sulfur atom Chemical group 0.000 claims description 4
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims description 4
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims description 3
- 229920006395 saturated elastomer Polymers 0.000 claims description 3
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000002837 carbocyclic group Chemical group 0.000 claims description 2
- 229910052799 carbon Inorganic materials 0.000 claims description 2
- 125000004432 carbon atom Chemical group C* 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 2
- 125000000623 heterocyclic group Chemical group 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 230000000361 pesticidal effect Effects 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- 125000004766 (C3-C6) cyclohaloalkyl group Chemical group 0.000 claims 2
- 125000003342 alkenyl group Chemical group 0.000 claims 2
- 125000000475 sulfinyl group Chemical group [*:2]S([*:1])=O 0.000 claims 2
- 239000002671 adjuvant Substances 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 description 29
- 125000004414 alkyl thio group Chemical group 0.000 description 14
- 125000000232 haloalkynyl group Chemical group 0.000 description 11
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 10
- 125000000753 cycloalkyl group Chemical group 0.000 description 9
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 5
- 125000004995 haloalkylthio group Chemical group 0.000 description 5
- 125000005347 halocycloalkyl group Chemical group 0.000 description 5
- 0 *C(N1*)=CC(N=C(*2)I)=C2C1=O Chemical compound *C(N1*)=CC(N=C(*2)I)=C2C1=O 0.000 description 2
- 241001465754 Metazoa Species 0.000 description 2
- 125000005161 aryl oxy carbonyl group Chemical group 0.000 description 2
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 description 2
- 241000256118 Aedes aegypti Species 0.000 description 1
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 description 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 description 1
- 125000005169 cycloalkylcarbonylamino group Chemical group 0.000 description 1
- 238000003745 diagnosis Methods 0.000 description 1
- 125000004438 haloalkoxy group Chemical group 0.000 description 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 1
- 238000003359 percent control normalization Methods 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15158762.3 | 2015-03-12 | ||
| EP15158762 | 2015-03-12 | ||
| EP15179249 | 2015-07-31 | ||
| EP15179249.6 | 2015-07-31 | ||
| PCT/EP2016/054757 WO2016142326A1 (en) | 2015-03-12 | 2016-03-07 | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018509418A JP2018509418A (ja) | 2018-04-05 |
| JP2018509418A5 true JP2018509418A5 (enExample) | 2019-04-18 |
| JP6774955B2 JP6774955B2 (ja) | 2020-10-28 |
Family
ID=55538187
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017548037A Active JP6774955B2 (ja) | 2015-03-12 | 2016-03-07 | 硫黄含有置換基を有する殺有害生物的に活性な四環式誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10323031B2 (enExample) |
| EP (1) | EP3268365B8 (enExample) |
| JP (1) | JP6774955B2 (enExample) |
| CN (2) | CN111646989A (enExample) |
| BR (1) | BR112017019372B1 (enExample) |
| ES (1) | ES2731078T3 (enExample) |
| WO (1) | WO2016142326A1 (enExample) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6779225B2 (ja) * | 2015-03-12 | 2020-11-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| US10202380B2 (en) * | 2015-07-01 | 2019-02-12 | Syngenta Participations Ag | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
| CN107735396B (zh) * | 2015-07-01 | 2021-03-02 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性多环衍生物 |
| US10550116B2 (en) * | 2015-10-26 | 2020-02-04 | Bayer Cropscience Aktiengesellschaft | Fused bicyclic heterocycle derivatives as pesticides |
| EA036621B1 (ru) | 2016-03-10 | 2020-12-01 | Ниссан Кемикал Корпорейшн | Конденсированные гетероциклические соединения и пестициды |
| CN114456164B (zh) * | 2016-10-27 | 2024-03-12 | 先正达参股股份有限公司 | 具有硫和羟胺取代基的杀有害生物活性杂环衍生物 |
| KR20190084310A (ko) | 2016-11-23 | 2019-07-16 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 살충제로서의 2-[3-(알킬술포닐)-2H-인다졸-2-일]-3H-이미다조[4,5-b]피리딘 유도체 및 유사한 화합물 |
| AU2018208422B2 (en) | 2017-01-10 | 2021-11-11 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| UY37556A (es) | 2017-01-10 | 2018-07-31 | Bayer Ag | Derivados heterocíclicos como pesticidas |
| CN110198942B (zh) * | 2017-01-24 | 2022-04-15 | 住友化学株式会社 | 稠合杂环化合物及含有其的组合物 |
| WO2018138050A1 (de) | 2017-01-26 | 2018-08-02 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019038195A1 (de) | 2017-08-22 | 2019-02-28 | Bayer Aktiengesellschaft | Heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019068572A1 (de) | 2017-10-04 | 2019-04-11 | Bayer Aktiengesellschaft | Heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CN108048372B (zh) * | 2018-01-30 | 2021-07-02 | 西南大学 | 一种短小芽孢杆菌及其防治蚕核型多角体病毒感染的应用 |
| CN111741958A (zh) | 2018-02-21 | 2020-10-02 | 拜耳公司 | 作为害虫防治剂的稠合双环杂环衍生物 |
| EP3765466B1 (de) * | 2018-03-12 | 2022-05-25 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| CN112262140B (zh) | 2018-06-06 | 2024-05-28 | 先正达农作物保护股份公司 | 具有含亚砜亚胺取代基的杀有害生物活性杂环衍生物 |
| BR122023022434A2 (pt) | 2018-06-26 | 2024-02-20 | Bayer Aktiengesellschaft | Derivados de heterocicleno como agentes de controle de pragas |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| JP7535532B2 (ja) | 2019-02-26 | 2024-08-16 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としての縮合二環式複素環式誘導体 |
| WO2021219810A1 (en) | 2020-04-30 | 2021-11-04 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| US20230247994A1 (en) | 2020-07-02 | 2023-08-10 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| AR126700A1 (es) | 2021-08-10 | 2023-11-01 | Syngenta Crop Protection Ag | Derivados heterocíclicos activos como plaguicidas con sustituyentes que contienen azufre |
| EP4680028A1 (en) | 2023-03-14 | 2026-01-21 | Syngenta Crop Protection AG | Control of pests resistant to insecticides |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3445299A1 (de) * | 1984-12-12 | 1986-06-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue imidazoderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
| BR112013016022B1 (pt) * | 2010-12-24 | 2019-05-07 | Sumitomo Chemical Company, Limited | Composto heterocíclico fundido e uso do mesmo para controle de peste. |
| TWI545119B (zh) | 2011-08-04 | 2016-08-11 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| US10939682B2 (en) * | 2013-07-02 | 2021-03-09 | Syngenta Participations Ag | Pesticidally active bi- or tricyclic heterocycles with sulfur containing substituents |
| JP6689821B2 (ja) * | 2014-08-12 | 2020-04-28 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| ES2806598T3 (es) * | 2014-12-11 | 2021-02-18 | Syngenta Participations Ag | Derivados tetracíclicos activos como plaguicidas con sustituyentes que contienen azufre |
| CN107108612B (zh) * | 2014-12-29 | 2020-05-15 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性四环衍生物 |
| JP6779225B2 (ja) * | 2015-03-12 | 2020-11-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| WO2017133994A1 (en) * | 2016-02-04 | 2017-08-10 | Syngenta Participations Ag | Pesticidally active derivatives with sulfur and cyclopropyl containing substituents |
-
2016
- 2016-03-07 JP JP2017548037A patent/JP6774955B2/ja active Active
- 2016-03-07 ES ES16710116T patent/ES2731078T3/es active Active
- 2016-03-07 CN CN202010494058.1A patent/CN111646989A/zh active Pending
- 2016-03-07 EP EP16710116.1A patent/EP3268365B8/en active Active
- 2016-03-07 US US15/554,283 patent/US10323031B2/en active Active
- 2016-03-07 BR BR112017019372-8A patent/BR112017019372B1/pt not_active IP Right Cessation
- 2016-03-07 WO PCT/EP2016/054757 patent/WO2016142326A1/en not_active Ceased
- 2016-03-07 CN CN201680015190.1A patent/CN107428751B/zh not_active Expired - Fee Related