JP2017523167A5 - - Google Patents
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- Publication number
- JP2017523167A5 JP2017523167A5 JP2017501239A JP2017501239A JP2017523167A5 JP 2017523167 A5 JP2017523167 A5 JP 2017523167A5 JP 2017501239 A JP2017501239 A JP 2017501239A JP 2017501239 A JP2017501239 A JP 2017501239A JP 2017523167 A5 JP2017523167 A5 JP 2017523167A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- haloalkyl
- cyano
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 29
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 23
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 22
- 229910052736 halogen Inorganic materials 0.000 claims description 20
- 150000002367 halogens Chemical class 0.000 claims description 20
- 125000000217 alkyl group Chemical group 0.000 claims description 17
- 238000000034 method Methods 0.000 claims description 10
- 125000001424 substituent group Chemical group 0.000 claims description 10
- 239000000463 material Substances 0.000 claims description 8
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 7
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- -1 C 1 -C 4 alkoxy Chemical group 0.000 claims description 5
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 4
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 4
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 4
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 4
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 4
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000002883 imidazolyl group Chemical group 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000001715 oxadiazolyl group Chemical group 0.000 claims description 4
- 125000002971 oxazolyl group Chemical group 0.000 claims description 4
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 4
- 125000003226 pyrazolyl group Chemical group 0.000 claims description 4
- 125000004076 pyridyl group Chemical group 0.000 claims description 4
- 125000000714 pyrimidinyl group Chemical group 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- 125000000335 thiazolyl group Chemical group 0.000 claims description 4
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 2
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 2
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 2
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 claims description 2
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 claims description 2
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 claims description 2
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 2
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 125000004663 dialkyl amino group Chemical group 0.000 claims description 2
- 229910052739 hydrogen Inorganic materials 0.000 claims description 2
- 239000001257 hydrogen Substances 0.000 claims description 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 125000001181 organosilyl group Chemical group [SiH3]* 0.000 claims description 2
- 229910052760 oxygen Inorganic materials 0.000 claims description 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 2
- 229910052717 sulfur Inorganic materials 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims 1
- 125000001188 haloalkyl group Chemical group 0.000 claims 1
- 239000000575 pesticide Substances 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 description 6
- 241001465754 Metazoa Species 0.000 description 2
- 125000004414 alkyl thio group Chemical group 0.000 description 2
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 2
- 229910052799 carbon Inorganic materials 0.000 description 1
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 description 1
- 230000000361 pesticidal effect Effects 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14176055.3 | 2014-07-08 | ||
| EP14176055 | 2014-07-08 | ||
| EP15158668.2 | 2015-03-11 | ||
| EP15158668 | 2015-03-11 | ||
| PCT/EP2015/065095 WO2016005263A1 (en) | 2014-07-08 | 2015-07-02 | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017523167A JP2017523167A (ja) | 2017-08-17 |
| JP2017523167A5 true JP2017523167A5 (enExample) | 2018-08-09 |
| JP6663907B2 JP6663907B2 (ja) | 2020-03-13 |
Family
ID=53502677
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017501239A Expired - Fee Related JP6663907B2 (ja) | 2014-07-08 | 2015-07-02 | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US9775353B2 (enExample) |
| EP (1) | EP3166941B1 (enExample) |
| JP (1) | JP6663907B2 (enExample) |
| KR (1) | KR20170029554A (enExample) |
| CN (1) | CN106661021B (enExample) |
| BR (1) | BR112017000269B1 (enExample) |
| CA (1) | CA2954238A1 (enExample) |
| ES (1) | ES2663523T3 (enExample) |
| MX (1) | MX2017000305A (enExample) |
| RU (1) | RU2017103953A (enExample) |
| WO (1) | WO2016005263A1 (enExample) |
Families Citing this family (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| US10081641B2 (en) * | 2014-08-21 | 2018-09-25 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| CN106604922B (zh) * | 2014-08-25 | 2020-05-05 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| PL3257853T3 (pl) | 2015-02-12 | 2022-03-21 | Nissan Chemical Corporation | Skondensowany związek heterocykliczny i środek zwalczający szkodliwe organizmy |
| EP3331870B1 (de) | 2015-08-07 | 2021-06-16 | Bayer CropScience Aktiengesellschaft | 2-(het)aryl-substituierte kondensierte heterocyclen-derivate als schädlingsbekämpfungsmittel |
| ES2866911T3 (es) | 2015-09-28 | 2021-10-20 | Bayer Cropscience Ag | Derivados heterocíclicos condensados sustituidos por 2-(het)arilo como pesticidas |
| PH12018500877B1 (en) | 2015-10-26 | 2023-09-20 | Bayer Cropscience Ag | Condensed bicyclic heterocycle derivatives as pest control agents |
| JP2019502713A (ja) | 2016-01-11 | 2019-01-31 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| WO2017134066A1 (en) * | 2016-02-05 | 2017-08-10 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| NZ745681A (en) | 2016-03-07 | 2022-05-27 | Agrofresh Inc | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| CA3016398A1 (en) | 2016-03-10 | 2017-09-14 | Nissan Chemical Corporation | Condensed heterocyclic compounds and pesticides |
| US11149027B2 (en) | 2016-03-31 | 2021-10-19 | Sumitomo Chemical Company, Limited | Heterocyclic compound |
| BR112018070537B1 (pt) | 2016-04-06 | 2022-11-01 | Sumitomo Chemical Company, Limited | Composto heterocíclico, composição compreendendo o mesmo e seus usos |
| BR112019006985B1 (pt) | 2016-10-06 | 2023-02-07 | Bayer Cropscience Aktiengesellschaft | Derivados de heterocíclicos fundidos bicíclicos substituídos por 2- (het)arila, seu uso, formulação agroquímica, e método para controle de pragas animais |
| WO2018065288A1 (de) | 2016-10-07 | 2018-04-12 | Bayer Cropscience Aktiengesellschaft | 2-[2-phenyl-1-(sulfonylmethyl)vinyl]-imidazo[4,5-b]pyridin-derivate und verwandte verbindungen als schädlingsbekämpfungsmittel im pflanzenschutz |
| CN109890818B (zh) | 2016-10-27 | 2022-11-25 | 先正达参股股份有限公司 | 具有硫和羟胺取代基的杀有害生物活性杂环衍生物 |
| HUE058180T2 (hu) | 2016-12-01 | 2022-07-28 | Syngenta Participations Ag | Eljárás kéntartalmú szubsztituenseket tartalmazó peszticid hatású heterociklusos származékok köztitermékének elõállítására |
| MX2019008230A (es) | 2017-01-10 | 2019-10-24 | Bayer Ag | Derivados heterociclicos como agentes de control de plagas. |
| AU2018207776B2 (en) | 2017-01-10 | 2021-06-17 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| TWI793104B (zh) | 2017-02-21 | 2023-02-21 | 瑞士商先正達合夥公司 | 具有含硫取代基的殺有害生物活性雜環衍生物 |
| CN110461834B (zh) | 2017-03-23 | 2024-03-12 | 住友化学株式会社 | 稠合杂环化合物及含有其的组合物 |
| WO2018197315A1 (en) | 2017-04-25 | 2018-11-01 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| EP3619203A1 (en) | 2017-05-02 | 2020-03-11 | Syngenta Participations AG | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| WO2019008072A1 (en) | 2017-07-05 | 2019-01-10 | Syngenta Participations Ag | HETEROCYCLIC DERIVATIVES HAVING PESTICIDE ACTIVITY HAVING SUBSTITUENTS CONTAINING SULFUR |
| AU2018332263B2 (en) | 2017-09-18 | 2023-02-09 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| CN107821422A (zh) * | 2017-11-09 | 2018-03-23 | 山西大学 | 一种含有绿僵菌素和啶虫脒的杀虫组合物及其应用 |
| JP7337810B2 (ja) | 2018-01-15 | 2023-09-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| AR115495A1 (es) | 2018-06-06 | 2021-01-27 | Syngenta Crop Protection Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| JP7353310B2 (ja) | 2018-06-26 | 2023-09-29 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| BR112021012991A2 (pt) | 2018-12-31 | 2021-09-14 | Syngenta Crop Protection Ag | Derivados heterocíclicos pesticidamente ativos com substituintes contendo enxofre |
| US20230060425A1 (en) | 2019-02-26 | 2023-03-02 | Bayer Aktiengesellschaft | Fused bicyclic heterocycle derivatives as pesticides |
| BR112021010400A2 (pt) | 2019-02-26 | 2021-08-24 | Bayer Aktiengesellschaft | Derivados heterocíclicos bicíclicos condensados como agentes de controle de praga |
| TW202120479A (zh) * | 2019-11-27 | 2021-06-01 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-羧酸及羧酸酯之方法 |
| TW202134214A (zh) | 2020-03-04 | 2021-09-16 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-甲酸醯胺以及甲酸鹽之方法 |
| KR102335886B1 (ko) * | 2020-03-11 | 2021-12-07 | 서울대학교병원 | 엘리오카퍼스 페티오라투스를 포함하는 심혈관 대사 질환의 예방 또는 치료용 조성물 |
| KR20230007398A (ko) | 2020-04-21 | 2023-01-12 | 바이엘 악티엔게젤샤프트 | 해충 방제제로서 2-(헤트)아릴-치환된 축합 헤테로시클릭 유도체 |
| CN115702149B (zh) | 2020-04-30 | 2025-08-19 | 先正达农作物保护股份公司 | 具有含硫取代基的杀有害生物活性的杂环衍生物 |
| JP2023532548A (ja) | 2020-07-02 | 2023-07-28 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| CA3201212A1 (en) | 2020-12-14 | 2022-06-23 | Rizwan Shabbir SHAIKH | Sulfoximine pesticides |
| EP4337661A1 (de) | 2021-05-12 | 2024-03-20 | Bayer Aktiengesellschaft | 2-(het)aryl-substituierte kondensierte heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CN120882309A (zh) | 2023-03-14 | 2025-10-31 | 先正达农作物保护股份公司 | 对杀昆虫剂具有抗性的有害生物的控制 |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
| WO2026027562A1 (en) * | 2024-07-30 | 2026-02-05 | Syngenta Crop Protection Ag | Synthesis of 5-(1-cyanocyclopropyl)-3-ethylsulfanyl-pyridine-2-carbonitrile |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0262845A1 (en) * | 1986-09-27 | 1988-04-06 | FISONS plc | Heterocyclic substituted azole derivatives |
| PH12013501178A1 (en) * | 2010-12-24 | 2013-07-15 | Sumitomo Chemical Co | Fused heterocyclic compound and use for pest control thereof |
| TWI589570B (zh) * | 2011-08-04 | 2017-07-01 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| JP2014111558A (ja) * | 2013-05-15 | 2014-06-19 | Sumitomo Chemical Co Ltd | 有害生物防除組成物およびその用途 |
| CN106604922B (zh) * | 2014-08-25 | 2020-05-05 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| US10435401B2 (en) * | 2014-09-16 | 2019-10-08 | Syngenta Participations Ag | Pesticidally active tetracyclic derivatives with sulphur containing substituents |
-
2015
- 2015-07-02 KR KR1020177003154A patent/KR20170029554A/ko not_active Withdrawn
- 2015-07-02 BR BR112017000269-8A patent/BR112017000269B1/pt not_active IP Right Cessation
- 2015-07-02 EP EP15733741.1A patent/EP3166941B1/en active Active
- 2015-07-02 CN CN201580036892.3A patent/CN106661021B/zh not_active Expired - Fee Related
- 2015-07-02 MX MX2017000305A patent/MX2017000305A/es unknown
- 2015-07-02 ES ES15733741.1T patent/ES2663523T3/es active Active
- 2015-07-02 RU RU2017103953A patent/RU2017103953A/ru unknown
- 2015-07-02 CA CA2954238A patent/CA2954238A1/en not_active Abandoned
- 2015-07-02 JP JP2017501239A patent/JP6663907B2/ja not_active Expired - Fee Related
- 2015-07-02 US US15/323,983 patent/US9775353B2/en not_active Expired - Fee Related
- 2015-07-02 WO PCT/EP2015/065095 patent/WO2016005263A1/en not_active Ceased
-
2017
- 2017-08-24 US US15/685,416 patent/US10051864B2/en active Active
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