JP2018502912A5 - - Google Patents
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- Publication number
- JP2018502912A5 JP2018502912A5 JP2017552222A JP2017552222A JP2018502912A5 JP 2018502912 A5 JP2018502912 A5 JP 2018502912A5 JP 2017552222 A JP2017552222 A JP 2017552222A JP 2017552222 A JP2017552222 A JP 2017552222A JP 2018502912 A5 JP2018502912 A5 JP 2018502912A5
- Authority
- JP
- Japan
- Prior art keywords
- cycloalkyl
- alkyl
- haloalkyl
- formula
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 40
- 150000001875 compounds Chemical class 0.000 claims description 37
- 229910052736 halogen Inorganic materials 0.000 claims description 36
- 150000002367 halogens Chemical class 0.000 claims description 36
- 125000000217 alkyl group Chemical group 0.000 claims description 35
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 30
- -1 C 2 -C 6 haloalkynyl Chemical group 0.000 claims description 28
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 27
- 229910052739 hydrogen Inorganic materials 0.000 claims description 26
- 239000001257 hydrogen Substances 0.000 claims description 26
- 125000001424 substituent group Chemical group 0.000 claims description 26
- 229910052757 nitrogen Inorganic materials 0.000 claims description 21
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 20
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 20
- 150000002431 hydrogen Chemical class 0.000 claims description 20
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 18
- 229910052760 oxygen Inorganic materials 0.000 claims description 18
- 239000001301 oxygen Substances 0.000 claims description 18
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 12
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 12
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 11
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 10
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims description 10
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 10
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims description 10
- 125000003545 alkoxy group Chemical group 0.000 claims description 9
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 8
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 8
- 238000000034 method Methods 0.000 claims description 7
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 6
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims description 6
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- 239000000463 material Substances 0.000 claims description 6
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical group [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 5
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 claims description 4
- 125000004432 carbon atom Chemical group C* 0.000 claims description 4
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 4
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims description 3
- 125000001188 haloalkyl group Chemical group 0.000 claims description 3
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 claims description 2
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 claims description 2
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims description 2
- 125000004740 (C1-C6) haloalkylsulfanyl group Chemical group 0.000 claims description 2
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 claims description 2
- 125000006771 (C1-C6) haloalkylthio group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000000304 alkynyl group Chemical group 0.000 claims description 2
- 125000003118 aryl group Chemical group 0.000 claims description 2
- 125000002837 carbocyclic group Chemical group 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 125000000623 heterocyclic group Chemical group 0.000 claims description 2
- 125000002883 imidazolyl group Chemical group 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 229910052717 sulfur Inorganic materials 0.000 claims description 2
- 239000011593 sulfur Substances 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 claims 1
- 239000002671 adjuvant Substances 0.000 claims 1
- 230000000361 pesticidal effect Effects 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 description 8
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 8
- 125000005347 halocycloalkyl group Chemical group 0.000 description 7
- 125000000232 haloalkynyl group Chemical group 0.000 description 5
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 4
- 125000004414 alkyl thio group Chemical group 0.000 description 4
- 125000004995 haloalkylthio group Chemical group 0.000 description 3
- 0 *c1cc2nc(I)c[n]2cc1 Chemical compound *c1cc2nc(I)c[n]2cc1 0.000 description 2
- 241001465754 Metazoa Species 0.000 description 2
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 description 2
- 239000012752 auxiliary agent Substances 0.000 description 1
- 125000005169 cycloalkylcarbonylamino group Chemical group 0.000 description 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 1
- 239000000575 pesticide Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14200413.4 | 2014-12-29 | ||
| EP14200413 | 2014-12-29 | ||
| PCT/EP2015/079877 WO2016107742A1 (en) | 2014-12-29 | 2015-12-15 | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018502912A JP2018502912A (ja) | 2018-02-01 |
| JP2018502912A5 true JP2018502912A5 (enExample) | 2019-01-31 |
| JP6736578B2 JP6736578B2 (ja) | 2020-08-05 |
Family
ID=52146355
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017552222A Active JP6736578B2 (ja) | 2014-12-29 | 2015-12-15 | 硫黄含有置換基を有する殺有害生物的に活性な四環式誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10196398B2 (enExample) |
| EP (1) | EP3240788B1 (enExample) |
| JP (1) | JP6736578B2 (enExample) |
| CN (1) | CN107108612B (enExample) |
| BR (1) | BR112017014061B1 (enExample) |
| ES (1) | ES2703172T3 (enExample) |
| WO (1) | WO2016107742A1 (enExample) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107428751B (zh) * | 2015-03-12 | 2020-06-30 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性四环衍生物 |
| WO2017026384A1 (ja) * | 2015-08-07 | 2017-02-16 | 日本農薬株式会社 | インダゾール化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| JP6916175B2 (ja) * | 2015-10-26 | 2021-08-11 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 有害生物防除剤としての縮合二環式ヘテロ環誘導体 |
| BR112018008765B1 (pt) | 2015-11-05 | 2022-05-24 | Sumitomo Chemical Company, Limited | Composto heterocíclico condensado, composição e método para o controle de um artrópode nocivo |
| WO2017093180A1 (de) | 2015-12-01 | 2017-06-08 | Bayer Cropscience Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CA3016398A1 (en) | 2016-03-10 | 2017-09-14 | Nissan Chemical Corporation | Condensed heterocyclic compounds and pesticides |
| WO2017174414A1 (de) | 2016-04-05 | 2017-10-12 | Bayer Cropscience Aktiengesellschaft | Naphthalin-derivate als schädlingsbekämpfungsmittel |
| ES2877571T3 (es) * | 2016-07-19 | 2021-11-17 | Bayer Cropscience Ag | Derivados de heterociclos bicíclicos condensados como pesticidas |
| US10660334B2 (en) | 2016-08-15 | 2020-05-26 | Bayer Cropscience Aktiengesellschaft | Fused bicyclic heterocycle derivatives as pesticides |
| JP2019206478A (ja) * | 2016-08-31 | 2019-12-05 | 日本農薬株式会社 | ３ｈ‐ピロロピリジン化合物及びｎ‐オキサイド、又はそれらの塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| CA3036776A1 (en) * | 2016-09-16 | 2018-03-22 | Sumitomo Chemical Company, Limited | Heterocyclic compound, and harmful-arthropod-controlling agent containing same |
| CN118702706A (zh) | 2016-09-19 | 2024-09-27 | 拜耳作物科学股份公司 | 吡唑并[1,5-a]吡啶衍生物及其作为农药的用途 |
| WO2018065288A1 (de) | 2016-10-07 | 2018-04-12 | Bayer Cropscience Aktiengesellschaft | 2-[2-phenyl-1-(sulfonylmethyl)vinyl]-imidazo[4,5-b]pyridin-derivate und verwandte verbindungen als schädlingsbekämpfungsmittel im pflanzenschutz |
| ES2837396T3 (es) | 2016-11-23 | 2021-06-30 | Bayer Cropscience Ag | Derivados de 2-[3-(alquilsulfonil)-2H-indazol-2-il]-3H-imidazo[4,5-b]piridina y compuestos similares como pesticidas |
| MX2019008230A (es) | 2017-01-10 | 2019-10-24 | Bayer Ag | Derivados heterociclicos como agentes de control de plagas. |
| JP7101177B2 (ja) | 2017-01-10 | 2022-07-14 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| US11064699B2 (en) | 2017-04-27 | 2021-07-20 | Nihon Nohyaku Co., Ltd. | Condensed heterocyclic compound or salt thereof, agricultural and horticultural insecticide comprising the compound or the salt, and method for using the insecticide |
| ES2914616T3 (es) | 2017-05-08 | 2022-06-14 | Syngenta Participations Ag | Derivados de imidazopirimidina con sustituyentes fenilo y piridilo que contienen azufre |
| BR112020003481B1 (pt) | 2017-08-22 | 2023-12-05 | Bayer Aktiengesellschaft | Derivados de heterocicleno, seus usos, formulação agroquímica, e métodos para controlar pragas animais e para proteger sementes ou uma planta germinativa de pragas |
| EP3305786A3 (de) | 2018-01-22 | 2018-07-25 | Bayer CropScience Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019162174A1 (de) | 2018-02-21 | 2019-08-29 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| CN112368280B (zh) | 2018-06-26 | 2023-01-20 | 拜耳公司 | 作为害虫防治剂的杂环衍生物 |
| TWI820231B (zh) * | 2018-10-11 | 2023-11-01 | 德商拜耳廠股份有限公司 | 用於製備經取代咪唑衍生物之方法 |
| WO2020141135A1 (en) | 2018-12-31 | 2020-07-09 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| KR20210133984A (ko) | 2019-02-26 | 2021-11-08 | 바이엘 악티엔게젤샤프트 | 해충 방제제로서의 축합된 비시클릭 헤테로시클릭 유도체 |
| JP7667745B2 (ja) * | 2020-01-09 | 2025-04-23 | 住友化学株式会社 | 複素環化合物及びそれを含有する有害節足動物防除組成物 |
| KR20230006482A (ko) | 2020-04-06 | 2023-01-10 | 바스프 에스이 | 살충제로서의 이미다조-피리미돈 화합물 |
| US20230247994A1 (en) | 2020-07-02 | 2023-08-10 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| EP4259627B1 (en) | 2020-12-14 | 2025-08-20 | Basf Se | Sulfoximine pesticides |
| CN120882309A (zh) | 2023-03-14 | 2025-10-31 | 先正达农作物保护股份公司 | 对杀昆虫剂具有抗性的有害生物的控制 |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
| WO2025229111A1 (en) | 2024-05-01 | 2025-11-06 | Basf Se | Pyrimidinone derivatives as pesticidal compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3445299A1 (de) * | 1984-12-12 | 1986-06-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue imidazoderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
| JPH07121937B2 (ja) * | 1987-03-18 | 1995-12-25 | 大塚製薬株式会社 | カルボスチリル誘導体 |
| TW201234965A (en) * | 2010-12-24 | 2012-09-01 | Sumitomo Chemical Co | Fused heterocyclic compound and use for pest control thereof |
| TWI589570B (zh) * | 2011-08-04 | 2017-07-01 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| BR112014029578B1 (pt) * | 2012-06-18 | 2019-10-22 | Sumitomo Chemical Co | composto heterocíclico fundido, composição e método de controle de peste |
-
2015
- 2015-12-15 EP EP15808685.0A patent/EP3240788B1/en active Active
- 2015-12-15 ES ES15808685T patent/ES2703172T3/es active Active
- 2015-12-15 BR BR112017014061-6A patent/BR112017014061B1/pt active IP Right Grant
- 2015-12-15 WO PCT/EP2015/079877 patent/WO2016107742A1/en not_active Ceased
- 2015-12-15 CN CN201580071577.4A patent/CN107108612B/zh active Active
- 2015-12-15 US US15/540,057 patent/US10196398B2/en active Active
- 2015-12-15 JP JP2017552222A patent/JP6736578B2/ja active Active
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