JP2018509379A5 - - Google Patents
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- JP2018509379A5 JP2018509379A5 JP2017532702A JP2017532702A JP2018509379A5 JP 2018509379 A5 JP2018509379 A5 JP 2018509379A5 JP 2017532702 A JP2017532702 A JP 2017532702A JP 2017532702 A JP2017532702 A JP 2017532702A JP 2018509379 A5 JP2018509379 A5 JP 2018509379A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- alkyl
- cycloalkyl
- haloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 150000001875 compounds Chemical class 0.000 claims description 48
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 33
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 33
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 29
- 125000001424 substituent group Chemical group 0.000 claims description 27
- 229910052736 halogen Inorganic materials 0.000 claims description 26
- 150000002367 halogens Chemical class 0.000 claims description 26
- 125000000217 alkyl group Chemical group 0.000 claims description 20
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 15
- -1 and C 1 -C 4 alkyl Chemical group 0.000 claims description 11
- 239000000463 material Substances 0.000 claims description 8
- 238000000034 method Methods 0.000 claims description 8
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 8
- 229910052717 sulfur Inorganic materials 0.000 claims description 8
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 7
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 6
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 6
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 6
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 6
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 6
- 239000000203 mixture Substances 0.000 claims description 6
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 6
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 5
- 150000003839 salts Chemical class 0.000 claims description 5
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 3
- 150000001204 N-oxides Chemical class 0.000 claims description 3
- 125000001188 haloalkyl group Chemical group 0.000 claims description 3
- 229910052739 hydrogen Inorganic materials 0.000 claims description 3
- 239000001257 hydrogen Substances 0.000 claims description 3
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 3
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 3
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 3
- 229910052760 oxygen Inorganic materials 0.000 claims description 3
- 239000004480 active ingredient Substances 0.000 claims description 2
- 230000000361 pesticidal effect Effects 0.000 claims description 2
- 241001414900 Anopheles stephensi Species 0.000 description 3
- 125000000753 cycloalkyl group Chemical group 0.000 description 3
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 description 2
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 description 2
- 241001465754 Metazoa Species 0.000 description 2
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 2
- 230000006698 induction Effects 0.000 description 2
- 229920000742 Cotton Polymers 0.000 description 1
- 241000255925 Diptera Species 0.000 description 1
- CZMRCDWAGMRECN-UGDNZRGBSA-N Sucrose Chemical compound O[C@H]1[C@H](O)[C@@H](CO)O[C@@]1(CO)O[C@@H]1[C@H](O)[C@@H](O)[C@H](O)[C@@H](CO)O1 CZMRCDWAGMRECN-UGDNZRGBSA-N 0.000 description 1
- 229930006000 Sucrose Natural products 0.000 description 1
- 239000003905 agrochemical Substances 0.000 description 1
- 125000003545 alkoxy group Chemical group 0.000 description 1
- 238000002405 diagnostic procedure Methods 0.000 description 1
- 230000000694 effects Effects 0.000 description 1
- 201000004792 malaria Diseases 0.000 description 1
- 238000003359 percent control normalization Methods 0.000 description 1
- 239000013049 sediment Substances 0.000 description 1
- 239000000243 solution Substances 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 238000001356 surgical procedure Methods 0.000 description 1
- 239000012085 test solution Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14198495 | 2014-12-17 | ||
| EP14198495.5 | 2014-12-17 | ||
| PCT/EP2015/079188 WO2016096584A1 (en) | 2014-12-17 | 2015-12-10 | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018509379A JP2018509379A (ja) | 2018-04-05 |
| JP2018509379A5 true JP2018509379A5 (enExample) | 2020-03-05 |
| JP6675404B2 JP6675404B2 (ja) | 2020-04-01 |
Family
ID=52146179
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017532702A Active JP6675404B2 (ja) | 2014-12-17 | 2015-12-10 | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
Country Status (25)
| Country | Link |
|---|---|
| US (3) | US10323030B2 (enExample) |
| EP (1) | EP3233851B1 (enExample) |
| JP (1) | JP6675404B2 (enExample) |
| KR (1) | KR102540827B1 (enExample) |
| CN (2) | CN107001365B (enExample) |
| AU (1) | AU2015366548B2 (enExample) |
| BR (1) | BR112017012638B1 (enExample) |
| CA (1) | CA2969600C (enExample) |
| CL (1) | CL2017001533A1 (enExample) |
| CO (1) | CO2017005790A2 (enExample) |
| DK (1) | DK3233851T3 (enExample) |
| ES (1) | ES2813952T3 (enExample) |
| HR (1) | HRP20201355T1 (enExample) |
| HU (1) | HUE050562T2 (enExample) |
| LT (1) | LT3233851T (enExample) |
| MX (1) | MX394806B (enExample) |
| MY (1) | MY182124A (enExample) |
| PH (1) | PH12017501013A1 (enExample) |
| PL (1) | PL3233851T3 (enExample) |
| PT (1) | PT3233851T (enExample) |
| RS (1) | RS60709B1 (enExample) |
| RU (1) | RU2765282C2 (enExample) |
| SI (1) | SI3233851T1 (enExample) |
| UA (1) | UA122781C2 (enExample) |
| WO (1) | WO2016096584A1 (enExample) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107074846B (zh) * | 2014-08-12 | 2020-05-19 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| JP6633091B2 (ja) * | 2014-11-07 | 2020-01-22 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する殺有害生物的に活性な多環式誘導体 |
| US10071997B2 (en) * | 2014-12-01 | 2018-09-11 | Syngenta Participations Ag | Pesticidally active amide heterocyclic derivatives with sulphur containing substituents |
| CN107001365B (zh) * | 2014-12-17 | 2019-09-24 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| TWI696612B (zh) | 2015-01-29 | 2020-06-21 | 日商日本農藥股份有限公司 | 具有環烷基吡啶基的稠合雜環化合物或其鹽類及含有該化合物的農園藝用殺蟲劑以及其使用方法 |
| CA3031139A1 (en) * | 2016-07-19 | 2018-01-25 | Bayer Cropscience Aktiengesellschaft | Condensed bicyclic heterocycle derivatives as pest control agents |
| BR112019006985B1 (pt) | 2016-10-06 | 2023-02-07 | Bayer Cropscience Aktiengesellschaft | Derivados de heterocíclicos fundidos bicíclicos substituídos por 2- (het)arila, seu uso, formulação agroquímica, e método para controle de pragas animais |
| WO2018065288A1 (de) | 2016-10-07 | 2018-04-12 | Bayer Cropscience Aktiengesellschaft | 2-[2-phenyl-1-(sulfonylmethyl)vinyl]-imidazo[4,5-b]pyridin-derivate und verwandte verbindungen als schädlingsbekämpfungsmittel im pflanzenschutz |
| EP3554242A1 (en) * | 2016-12-15 | 2019-10-23 | Syngenta Participations AG | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| CA3047896C (en) | 2016-12-27 | 2021-11-09 | Nihon Nohyaku Co., Ltd. | 4h-pyrrolopyridine compound or salt thereof, agricultural and horticultural insecticide comprising the compound or the salt, and method for using the insecticide |
| AU2018207776B2 (en) | 2017-01-10 | 2021-06-17 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| MX2019008230A (es) | 2017-01-10 | 2019-10-24 | Bayer Ag | Derivados heterociclicos como agentes de control de plagas. |
| TWI793104B (zh) | 2017-02-21 | 2023-02-21 | 瑞士商先正達合夥公司 | 具有含硫取代基的殺有害生物活性雜環衍生物 |
| WO2018197315A1 (en) | 2017-04-25 | 2018-11-01 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| WO2018215304A1 (en) | 2017-05-22 | 2018-11-29 | Syngenta Participations Ag | Tetracyclic pyridazine sulphur containing compounds and their use as pesticides |
| WO2019059244A1 (ja) | 2017-09-21 | 2019-03-28 | 日本農薬株式会社 | シクロプロピルピリジル基を有するベンゾイミダゾール化合物又はその塩類、及びそれらの化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| CN112262140B (zh) | 2018-06-06 | 2024-05-28 | 先正达农作物保护股份公司 | 具有含亚砜亚胺取代基的杀有害生物活性杂环衍生物 |
| JP7353310B2 (ja) | 2018-06-26 | 2023-09-29 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| CN112384516A (zh) | 2018-07-10 | 2021-02-19 | 日本农药株式会社 | 具有任选被卤代的亚烷基二氧基的苯并咪唑化合物或其盐类、以及含有这些化合物的农业园艺用杀虫剂及其使用方法 |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| RS66446B1 (sr) * | 2018-10-29 | 2025-02-28 | Nippon Soda Co | (hetero)arilimidazol jedinjenja i sredstva za kontrolu štetnih organizama |
| WO2020175491A1 (ja) * | 2019-02-26 | 2020-09-03 | 日本曹達株式会社 | ピリジン ｎ－オキサイド化合物および有害生物防除剤 |
| BR112021010400A2 (pt) * | 2019-02-26 | 2021-08-24 | Bayer Aktiengesellschaft | Derivados heterocíclicos bicíclicos condensados como agentes de controle de praga |
| TW202120479A (zh) | 2019-11-27 | 2021-06-01 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-羧酸及羧酸酯之方法 |
| TW202134214A (zh) | 2020-03-04 | 2021-09-16 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-甲酸醯胺以及甲酸鹽之方法 |
| JP2023532548A (ja) | 2020-07-02 | 2023-07-28 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| WO2022043468A1 (en) | 2020-08-26 | 2022-03-03 | Syngenta Crop Protection Ag | Process for the preparation of 2,2-difluoro-1,3-benzodioxole derivatives with sulfur containing substituents |
| BR112023025278A2 (pt) | 2021-06-02 | 2024-02-27 | Syngenta Crop Protection Ag | Derivados heterocíclicos com substituintes contendo sulfoximina ativos em termos pesticidas |
| CN120882309A (zh) | 2023-03-14 | 2025-10-31 | 先正达农作物保护股份公司 | 对杀昆虫剂具有抗性的有害生物的控制 |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
| WO2026037853A1 (en) | 2024-08-14 | 2026-02-19 | Basf Se | Benzoxazole derivatives as pesticidal compounds |
| WO2026041702A1 (en) | 2024-08-21 | 2026-02-26 | Basf Se | Benzoxazole derivatives as pesticidal compounds |
| WO2026046760A1 (en) | 2024-08-29 | 2026-03-05 | Basf Se | Pesticidal mixtures comprising an ethylsulfone compound |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES8401486A1 (es) * | 1981-11-10 | 1983-12-01 | Wellcome Found | Un procedimiento para la preparacion de nuevos derivados de imidazo (4,5-c)piridina. |
| US4772600A (en) * | 1986-06-09 | 1988-09-20 | A. H. Robins Company, Inc. | Fused imidazoheterocyclic compounds and pharmaceutical compositions |
| NZ242756A (en) | 1991-06-03 | 1994-07-26 | Sumitomo Chemical Co | Benzimidazole derivatives having a fused ring which contains 1 or 2 o atoms and at least 1 -cf2- unit; use as fungicides; and precursors |
| US8273764B2 (en) * | 2009-04-28 | 2012-09-25 | Sumitomo Chemical Company, Limited | Fused heterocyclic compounds and use thereof |
| WO2012033548A2 (en) * | 2010-09-07 | 2012-03-15 | E. I. Du Pont De Nemours And Company | Herbicidal bis-nitrogen-containing oxo and sulfono heterocycles |
| TW201114762A (en) * | 2009-09-30 | 2011-05-01 | Sumitomo Chemical Co | Composition and method for controlling arthropod pests |
| PH12013501178A1 (en) * | 2010-12-24 | 2013-07-15 | Sumitomo Chemical Co | Fused heterocyclic compound and use for pest control thereof |
| TWI589570B (zh) * | 2011-08-04 | 2017-07-01 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| EP2857397B1 (en) * | 2012-05-30 | 2020-04-08 | Sumitomo Chemical Company Limited | Fused heterocyclic compound |
| WO2014119494A1 (ja) | 2013-01-31 | 2014-08-07 | 住友化学株式会社 | 有害生物防除組成物及び有害生物の防除方法 |
| UY35421A (es) * | 2013-03-15 | 2014-10-31 | Nihon Nohyaku Co Ltd | Compuesto heterocíclico condensado o su sal, insecticida agrícola u hortícola que comprende el comp uesto y método de uso del insecticida |
| PE20171645A1 (es) * | 2014-02-17 | 2017-11-13 | Bayer Cropscience Ag | Derivados de heterociclos biciclicos condensados sustituidos con 2-(het)arilo como agentes para combatir parasitos |
| JP2014208695A (ja) * | 2014-07-04 | 2014-11-06 | 住友化学株式会社 | 有害生物防除組成物およびその用途 |
| US10435401B2 (en) * | 2014-09-16 | 2019-10-08 | Syngenta Participations Ag | Pesticidally active tetracyclic derivatives with sulphur containing substituents |
| CN107001365B (zh) * | 2014-12-17 | 2019-09-24 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
-
2015
- 2015-12-10 CN CN201580068692.6A patent/CN107001365B/zh active Active
- 2015-12-10 KR KR1020177016823A patent/KR102540827B1/ko active Active
- 2015-12-10 SI SI201531332T patent/SI3233851T1/sl unknown
- 2015-12-10 US US15/536,820 patent/US10323030B2/en active Active
- 2015-12-10 HU HUE15807678A patent/HUE050562T2/hu unknown
- 2015-12-10 JP JP2017532702A patent/JP6675404B2/ja active Active
- 2015-12-10 ES ES15807678T patent/ES2813952T3/es active Active
- 2015-12-10 CN CN201910793016.5A patent/CN110526911B/zh active Active
- 2015-12-10 MX MX2017007900A patent/MX394806B/es unknown
- 2015-12-10 PL PL15807678T patent/PL3233851T3/pl unknown
- 2015-12-10 RS RS20201031A patent/RS60709B1/sr unknown
- 2015-12-10 AU AU2015366548A patent/AU2015366548B2/en active Active
- 2015-12-10 HR HRP20201355TT patent/HRP20201355T1/hr unknown
- 2015-12-10 LT LTEP15807678.6T patent/LT3233851T/lt unknown
- 2015-12-10 MY MYPI2017000809A patent/MY182124A/en unknown
- 2015-12-10 UA UAA201707453A patent/UA122781C2/uk unknown
- 2015-12-10 RU RU2017125267A patent/RU2765282C2/ru active
- 2015-12-10 BR BR112017012638-9A patent/BR112017012638B1/pt active IP Right Grant
- 2015-12-10 WO PCT/EP2015/079188 patent/WO2016096584A1/en not_active Ceased
- 2015-12-10 DK DK15807678.6T patent/DK3233851T3/da active
- 2015-12-10 PT PT158076786T patent/PT3233851T/pt unknown
- 2015-12-10 EP EP15807678.6A patent/EP3233851B1/en active Active
- 2015-12-10 CA CA2969600A patent/CA2969600C/en active Active
-
2017
- 2017-06-01 PH PH12017501013A patent/PH12017501013A1/en unknown
- 2017-06-12 CO CONC2017/0005790A patent/CO2017005790A2/es unknown
- 2017-06-14 CL CL2017001533A patent/CL2017001533A1/es unknown
-
2019
- 2019-06-17 US US16/443,596 patent/US11072608B2/en active Active
-
2021
- 2021-06-17 US US17/350,374 patent/US20210317119A1/en active Pending
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