JP2020138980A5 - - Google Patents
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- Publication number
- JP2020138980A5 JP2020138980A5 JP2020100953A JP2020100953A JP2020138980A5 JP 2020138980 A5 JP2020138980 A5 JP 2020138980A5 JP 2020100953 A JP2020100953 A JP 2020100953A JP 2020100953 A JP2020100953 A JP 2020100953A JP 2020138980 A5 JP2020138980 A5 JP 2020138980A5
- Authority
- JP
- Japan
- Prior art keywords
- therapeutic agent
- agent according
- dry eye
- eye therapeutic
- diquafosol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 208000003556 Dry Eye Syndromes Diseases 0.000 claims 19
- 206010013774 Dry eye Diseases 0.000 claims 19
- 239000003814 drug Substances 0.000 claims 18
- 229940124597 therapeutic agent Drugs 0.000 claims 18
- NMLMACJWHPHKGR-NCOIDOBVSA-N P(1),P(4)-bis(uridin-5'-yl) tetraphosphate Chemical compound N1([C@@H]2O[C@@H]([C@H]([C@H]2O)O)COP(O)(=O)OP(O)(=O)OP(O)(=O)OP(O)(=O)OC[C@@H]2[C@H]([C@H]([C@@H](O2)N2C(NC(=O)C=C2)=O)O)O)C=CC(=O)NC1=O NMLMACJWHPHKGR-NCOIDOBVSA-N 0.000 claims 7
- 229950003529 diquafosol Drugs 0.000 claims 7
- 235000013855 polyvinylpyrrolidone Nutrition 0.000 claims 6
- 229920000036 polyvinylpyrrolidone Polymers 0.000 claims 6
- 239000001267 polyvinylpyrrolidone Substances 0.000 claims 6
- 150000003839 salts Chemical class 0.000 claims 6
- 239000003889 eye drop Substances 0.000 claims 4
- 239000006196 drop Substances 0.000 claims 3
- 229940012356 eye drops Drugs 0.000 claims 3
- 238000004090 dissolution Methods 0.000 claims 1
- 239000000725 suspension Substances 0.000 claims 1
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022116528A JP7472202B2 (ja) | 2018-02-28 | 2022-07-21 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
| JP2024019332A JP2024045506A (ja) | 2018-02-28 | 2024-02-13 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2018035578 | 2018-02-28 | ||
| JP2018035578 | 2018-02-28 | ||
| JP2020503563A JP6716800B2 (ja) | 2018-02-28 | 2019-02-27 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020503563A Division JP6716800B2 (ja) | 2018-02-28 | 2019-02-27 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022116528A Division JP7472202B2 (ja) | 2018-02-28 | 2022-07-21 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020138980A JP2020138980A (ja) | 2020-09-03 |
| JP2020138980A5 true JP2020138980A5 (enExample) | 2022-03-04 |
| JP7297718B2 JP7297718B2 (ja) | 2023-06-26 |
Family
ID=67806273
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020503563A Active JP6716800B2 (ja) | 2018-02-28 | 2019-02-27 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
| JP2020100953A Active JP7297718B2 (ja) | 2018-02-28 | 2020-06-10 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
| JP2022116528A Active JP7472202B2 (ja) | 2018-02-28 | 2022-07-21 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
| JP2024019332A Pending JP2024045506A (ja) | 2018-02-28 | 2024-02-13 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020503563A Active JP6716800B2 (ja) | 2018-02-28 | 2019-02-27 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022116528A Active JP7472202B2 (ja) | 2018-02-28 | 2022-07-21 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
| JP2024019332A Pending JP2024045506A (ja) | 2018-02-28 | 2024-02-13 | ジクアホソルおよびカチオン性ポリマーを含有する眼科用組成物 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20210000844A1 (enExample) |
| EP (1) | EP3760207A4 (enExample) |
| JP (4) | JP6716800B2 (enExample) |
| KR (3) | KR102472773B1 (enExample) |
| CN (2) | CN117137866A (enExample) |
| BR (1) | BR112020017661A2 (enExample) |
| CA (1) | CA3091700A1 (enExample) |
| EA (1) | EA202092030A1 (enExample) |
| MX (2) | MX2020008925A (enExample) |
| PH (1) | PH12020551313B1 (enExample) |
| SG (1) | SG11202007977RA (enExample) |
| TW (3) | TWI833406B (enExample) |
| UA (1) | UA129517C2 (enExample) |
| WO (1) | WO2019168023A1 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI833406B (zh) * | 2018-02-28 | 2024-02-21 | 日商參天製藥股份有限公司 | 含有迪夸弗索(Diquafosol)及陽離子性聚合物之眼科用組合物 |
| TWI833913B (zh) * | 2019-02-27 | 2024-03-01 | 日商參天製藥股份有限公司 | 含有迪夸弗索(diquafosol)或其鹽、乙烯系高分子及纖維素系高分子之眼科用組合物 |
| KR20240049646A (ko) * | 2019-08-27 | 2024-04-16 | 산텐 세이야꾸 가부시키가이샤 | 디쿠아포솔 또는 그 염 및 폴리비닐피롤리돈을 함유하는 수성 안과용 조성물 |
| KR102365008B1 (ko) * | 2020-06-23 | 2022-02-23 | 주식회사태준제약 | 디쿠아포솔을 포함하는 점안 조성물 |
| JP7230169B2 (ja) * | 2020-12-25 | 2023-02-28 | 参天製薬株式会社 | ジクアホソルまたはその塩、銀塩およびイオン性等張化剤を含有する水性点眼液 |
| CN113712910A (zh) * | 2021-08-05 | 2021-11-30 | 广州市桐晖药业有限公司 | 一种滴眼液及其制备方法 |
| KR102794468B1 (ko) | 2022-04-04 | 2025-04-14 | 서울대학교산학협력단 | 감미 억제용 조성물 및 식품의 감미 억제 방법 |
| KR20250038935A (ko) * | 2023-09-13 | 2025-03-20 | 루다큐어 주식회사 | 8-옥소-2'-데옥시구아노신 또는 이의 약학적으로 허용가능한 염을 포함하는 수용액 형태의 점안제 |
| KR20250160050A (ko) | 2024-05-03 | 2025-11-11 | 삼천당제약주식회사 | 물리화학적 특성이 개선된 안구건조증 예방 또는 치료용 약학 조성물 |
| CN119970633A (zh) * | 2025-03-26 | 2025-05-13 | 苏州乐珠制药有限公司 | 一种地夸磷索钠滴眼液及其制备方法 |
Family Cites Families (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH01294620A (ja) | 1988-05-19 | 1989-11-28 | Kissei Pharmaceut Co Ltd | 水溶液製剤およびその製造方法 |
| US5358706A (en) * | 1992-09-30 | 1994-10-25 | Union Carbide Chemicals & Plastics Technology Corporation | Muco-adhesive polymers |
| US5422116A (en) * | 1994-02-18 | 1995-06-06 | Ciba-Geigy Corporation | Liquid ophthalmic sustained release delivery system |
| JP3155689B2 (ja) * | 1995-08-10 | 2001-04-16 | 昭和薬品化工株式会社 | 消炎点眼剤 |
| US5900407A (en) * | 1997-02-06 | 1999-05-04 | Inspire Pharmaceuticals, Inc. | Method of treating dry eye disease with uridine triphosphates and related compounds |
| KR20010013797A (ko) | 1997-07-25 | 2001-02-26 | 인스파이어 파마슈티컬스 인코퍼레이티드 | 디(우리딘 5'-테트라포스페이트) 염 및 그의 제조방법과용도 |
| JP2001294620A (ja) | 2000-04-11 | 2001-10-23 | Showa Denko Kk | プラスチックレンズ材料、該材料の製造方法、プラスチックレンズ用組成物、該組成物を硬化してなるプラスチックレンズ、及び該プラスチックレンズの製造方法 |
| AU6064301A (en) * | 2000-05-30 | 2001-12-11 | Santen Pharmaceutical Co Ltd | Ectocornea extension promoters |
| KR101389300B1 (ko) * | 2005-02-14 | 2014-04-25 | 존슨 앤드 존슨 비젼 케어, 인코포레이티드 | 안과용 렌즈의 제조방법, 안과용 장치 및 콘택트 렌즈 |
| JP4515960B2 (ja) | 2005-05-19 | 2010-08-04 | 株式会社資生堂 | 整髪料洗浄剤及びその使用方法 |
| KR100870104B1 (ko) * | 2005-11-28 | 2008-11-26 | 주식회사 머젠스 | 안구건조증 치료 및 예방용 조성물 |
| KR20150115959A (ko) * | 2007-10-12 | 2015-10-14 | 레솔빅스 파마슈티칼즈, 인코퍼레이티드 | 안과 질환의 치료를 위한 옥실리핀 화합물 |
| BRPI0909797A2 (pt) * | 2008-03-07 | 2017-08-22 | Sun Pharma Advanced Res Co Ltd | Composição oftálmica |
| JP2012149057A (ja) * | 2010-12-28 | 2012-08-09 | Santen Pharmaceut Co Ltd | ジクアホソル含有点眼液およびその製造方法、不溶性析出物発生の抑制方法 |
| SG10201607872PA (en) * | 2012-03-26 | 2016-11-29 | Santen Pharmaceutical Co Ltd | Ophthalmic solution comprising diquafosol |
| ES2747808T3 (es) * | 2014-05-07 | 2020-03-11 | Croma Pharma Ges M B H | Solución oftálmica acuosa y método para tratar el síndrome del ojo seco |
| WO2015190483A1 (ja) * | 2014-06-10 | 2015-12-17 | ロート製薬株式会社 | 眼科用水性組成物 |
| SG11201705138QA (en) * | 2014-12-25 | 2017-07-28 | Santen Pharmaceutical Co Ltd | Aqueous ophthalmic solution |
| KR101587385B1 (ko) | 2015-07-29 | 2016-01-21 | 국제약품공업주식회사 | 사이클로스포린 함유 무자극성의 안약조성물 및 편리한 제조방법 |
| WO2017033967A1 (ja) * | 2015-08-24 | 2017-03-02 | 参天製薬株式会社 | 眼科用フィルム製剤 |
| LT3266446T (lt) * | 2016-07-07 | 2019-01-25 | Laboratorios Salvat, S.A. | Oftalmologinė kompozicija, apimanti ricinos aliejų ir vidutinio grandinės ilgio trigliceridą |
| CN106772747B (zh) * | 2016-12-26 | 2022-10-18 | 深圳市光科全息技术有限公司 | 一种光学膜及其制作方法 |
| MY196565A (en) * | 2017-04-25 | 2023-04-19 | Wakamoto Pharma Co Ltd | Thermogelling Artificial Tears |
| JP6582029B2 (ja) * | 2017-10-03 | 2019-09-25 | 株式会社メニコン | 眼科用組成液及びその使用方法 |
| TWI833406B (zh) * | 2018-02-28 | 2024-02-21 | 日商參天製藥股份有限公司 | 含有迪夸弗索(Diquafosol)及陽離子性聚合物之眼科用組合物 |
| CN108853016A (zh) * | 2018-09-26 | 2018-11-23 | 广州大光制药有限公司 | 一种地夸磷索钠滴眼液及其制备方法 |
| TWI833913B (zh) * | 2019-02-27 | 2024-03-01 | 日商參天製藥股份有限公司 | 含有迪夸弗索(diquafosol)或其鹽、乙烯系高分子及纖維素系高分子之眼科用組合物 |
| KR20240049646A (ko) * | 2019-08-27 | 2024-04-16 | 산텐 세이야꾸 가부시키가이샤 | 디쿠아포솔 또는 그 염 및 폴리비닐피롤리돈을 함유하는 수성 안과용 조성물 |
-
2019
- 2019-02-27 TW TW111140996A patent/TWI833406B/zh active
- 2019-02-27 US US16/976,504 patent/US20210000844A1/en not_active Abandoned
- 2019-02-27 KR KR1020207027473A patent/KR102472773B1/ko active Active
- 2019-02-27 BR BR112020017661-3A patent/BR112020017661A2/pt unknown
- 2019-02-27 KR KR1020227041383A patent/KR102796051B1/ko active Active
- 2019-02-27 WO PCT/JP2019/007542 patent/WO2019168023A1/ja not_active Ceased
- 2019-02-27 SG SG11202007977RA patent/SG11202007977RA/en unknown
- 2019-02-27 UA UAA202006163A patent/UA129517C2/uk unknown
- 2019-02-27 JP JP2020503563A patent/JP6716800B2/ja active Active
- 2019-02-27 KR KR1020257011738A patent/KR20250053220A/ko active Pending
- 2019-02-27 CN CN202311151214.4A patent/CN117137866A/zh active Pending
- 2019-02-27 EP EP19759990.5A patent/EP3760207A4/en active Pending
- 2019-02-27 CN CN201980015357.8A patent/CN111757742B/zh active Active
- 2019-02-27 CA CA3091700A patent/CA3091700A1/en active Pending
- 2019-02-27 TW TW108106730A patent/TWI781296B/zh active
- 2019-02-27 EA EA202092030A patent/EA202092030A1/ru unknown
- 2019-02-27 MX MX2020008925A patent/MX2020008925A/es unknown
- 2019-02-27 PH PH1/2020/551313A patent/PH12020551313B1/en unknown
- 2019-02-27 TW TW113102160A patent/TWI898399B/zh active
-
2020
- 2020-06-10 JP JP2020100953A patent/JP7297718B2/ja active Active
- 2020-08-26 MX MX2022014791A patent/MX2022014791A/es unknown
-
2022
- 2022-07-21 JP JP2022116528A patent/JP7472202B2/ja active Active
-
2024
- 2024-02-13 JP JP2024019332A patent/JP2024045506A/ja active Pending
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