JP2020059759A5 - - Google Patents

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Publication number
JP2020059759A5
JP2020059759A5 JP2020000332A JP2020000332A JP2020059759A5 JP 2020059759 A5 JP2020059759 A5 JP 2020059759A5 JP 2020000332 A JP2020000332 A JP 2020000332A JP 2020000332 A JP2020000332 A JP 2020000332A JP 2020059759 A5 JP2020059759 A5 JP 2020059759A5
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JP
Japan
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crystal
morpholinophenylamino
cyanomethyl
pyrimidin
benzamide
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JP2020000332A
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English (en)
Japanese (ja)
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JP6840909B2 (ja
JP2020059759A (ja
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Publication of JP2020059759A5 publication Critical patent/JP2020059759A5/ja
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JP2020000332A 2014-06-12 2020-01-06 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩 Active JP6840909B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462011315P 2014-06-12 2014-06-12
US62/011,315 2014-06-12

Related Parent Applications (1)

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JP2018164680A Division JP6883560B2 (ja) 2014-06-12 2018-09-03 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩

Publications (3)

Publication Number Publication Date
JP2020059759A JP2020059759A (ja) 2020-04-16
JP2020059759A5 true JP2020059759A5 (https=) 2020-12-24
JP6840909B2 JP6840909B2 (ja) 2021-03-10

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ID=53674249

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2016572271A Active JP6600649B2 (ja) 2014-06-12 2015-06-11 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩
JP2018164680A Active JP6883560B2 (ja) 2014-06-12 2018-09-03 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩
JP2020000332A Active JP6840909B2 (ja) 2014-06-12 2020-01-06 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩
JP2021079700A Active JP7198867B2 (ja) 2014-06-12 2021-05-10 N-(シアノメチル)-4-(2-(4-モルホリノフェニルアミノ)ピリミジン-4-イル)ベンズアミド塩酸塩
JP2022202374A Active JP7550205B2 (ja) 2014-06-12 2022-12-19 N-(シアノメチル)-4-(2-(4-モルホリノフェニルアミノ)ピリミジン-4-イル)ベンズアミド塩酸塩

Family Applications Before (2)

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JP2016572271A Active JP6600649B2 (ja) 2014-06-12 2015-06-11 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩
JP2018164680A Active JP6883560B2 (ja) 2014-06-12 2018-09-03 N−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド塩酸塩

Family Applications After (2)

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JP2021079700A Active JP7198867B2 (ja) 2014-06-12 2021-05-10 N-(シアノメチル)-4-(2-(4-モルホリノフェニルアミノ)ピリミジン-4-イル)ベンズアミド塩酸塩
JP2022202374A Active JP7550205B2 (ja) 2014-06-12 2022-12-19 N-(シアノメチル)-4-(2-(4-モルホリノフェニルアミノ)ピリミジン-4-イル)ベンズアミド塩酸塩

Country Status (36)

Country Link
US (5) US9469613B2 (https=)
EP (3) EP3154950B1 (https=)
JP (5) JP6600649B2 (https=)
KR (1) KR101928225B1 (https=)
CN (2) CN106458929A (https=)
AP (1) AP2016009551A0 (https=)
AR (1) AR100818A1 (https=)
AU (1) AU2015274554B9 (https=)
BR (1) BR112016028749A2 (https=)
CA (1) CA2951883C (https=)
CR (1) CR20160575A (https=)
CU (1) CU20160183A7 (https=)
CY (2) CY1123604T1 (https=)
DK (1) DK3154950T3 (https=)
EA (1) EA032639B1 (https=)
EC (1) ECSP16093323A (https=)
ES (1) ES2822773T3 (https=)
FI (1) FIC20240025I1 (https=)
FR (1) FR24C1030I2 (https=)
HR (1) HRP20201492T1 (https=)
HU (2) HUE051360T2 (https=)
IL (3) IL249038B (https=)
LT (2) LT3154950T (https=)
MA (1) MA40067A (https=)
MX (3) MX374541B (https=)
NL (1) NL301282I2 (https=)
NZ (1) NZ725966A (https=)
PH (1) PH12016502461A1 (https=)
PL (1) PL3154950T3 (https=)
PT (1) PT3154950T (https=)
RS (1) RS61065B1 (https=)
SG (2) SG11201610079VA (https=)
SI (1) SI3154950T1 (https=)
TW (3) TWI729644B (https=)
UY (1) UY36166A (https=)
WO (1) WO2015191846A1 (https=)

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TWI729644B (zh) * 2014-06-12 2021-06-01 美商西爾拉癌症醫學公司 N-(氰基甲基)-4-(2-(4-𠰌啉基苯基胺基)嘧啶-4-基)苯甲醯胺
CN106316963B (zh) * 2015-06-26 2021-06-08 苏州泽璟生物制药股份有限公司 吗啡啉苯基氨基嘧啶化合物或其盐的多晶型物
CN106316964B (zh) * 2015-06-26 2019-06-25 苏州泽璟生物制药股份有限公司 苯基氨基嘧啶化合物或其盐的多晶型物
TWI794171B (zh) 2016-05-11 2023-03-01 美商滬亞生物國際有限公司 Hdac抑制劑與pd-l1抑制劑之組合治療
TWI808055B (zh) 2016-05-11 2023-07-11 美商滬亞生物國際有限公司 Hdac 抑制劑與 pd-1 抑制劑之組合治療
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CN117794545A (zh) 2021-07-30 2024-03-29 葛兰素史密斯克莱有限责任公司 骨髓纤维化的治疗中的生物标志物和患者选择
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WO2023023473A1 (en) 2021-08-16 2023-02-23 Sierra Oncology, Inc. Methods of using momelotinib to treat chronic kidney disease
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