JP2009517353A5 - - Google Patents
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- Publication number
- JP2009517353A5 JP2009517353A5 JP2008541641A JP2008541641A JP2009517353A5 JP 2009517353 A5 JP2009517353 A5 JP 2009517353A5 JP 2008541641 A JP2008541641 A JP 2008541641A JP 2008541641 A JP2008541641 A JP 2008541641A JP 2009517353 A5 JP2009517353 A5 JP 2009517353A5
- Authority
- JP
- Japan
- Prior art keywords
- crystalline form
- compound
- acid addition
- addition salt
- methanesulfonic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- KTUFNOKKBVMGRW-UHFFFAOYSA-N Cc(ccc(NC(c1ccc(CN2CCN(C)CC2)cc1)=O)c1)c1Nc1nc(-c2cnccc2)ccn1 Chemical compound Cc(ccc(NC(c1ccc(CN2CCN(C)CC2)cc1)=O)c1)c1Nc1nc(-c2cnccc2)ccn1 KTUFNOKKBVMGRW-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (11)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0524061A GB0524061D0 (en) | 2005-11-25 | 2005-11-25 | Organic compounds |
| GB0524062A GB0524062D0 (en) | 2005-11-25 | 2005-11-25 | Organic compounds |
| GB0524061.9 | 2005-11-25 | ||
| GB0524062.7 | 2005-11-25 | ||
| US74001805P | 2005-11-28 | 2005-11-28 | |
| US74001605P | 2005-11-28 | 2005-11-28 | |
| US74001705P | 2005-11-28 | 2005-11-28 | |
| US60/740,017 | 2005-11-28 | ||
| US60/740,016 | 2005-11-28 | ||
| US60/740,018 | 2005-11-28 | ||
| PCT/EP2006/011240 WO2007059963A1 (en) | 2005-11-25 | 2006-11-23 | F,g,h,i and k crystal forms of imatinib mesylate |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014005741A Division JP2014074067A (ja) | 2005-11-25 | 2014-01-16 | メシル酸イマチニブのｆ、ｇ、ｈ、ｉおよびｋ結晶形 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009517353A JP2009517353A (ja) | 2009-04-30 |
| JP2009517353A5 true JP2009517353A5 (https=) | 2010-01-14 |
| JP5844508B2 JP5844508B2 (ja) | 2016-01-20 |
Family
ID=37847165
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008541641A Expired - Fee Related JP5844508B2 (ja) | 2005-11-25 | 2006-11-23 | メシル酸イマチニブのｆ結晶形 |
| JP2014005741A Pending JP2014074067A (ja) | 2005-11-25 | 2014-01-16 | メシル酸イマチニブのｆ、ｇ、ｈ、ｉおよびｋ結晶形 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014005741A Pending JP2014074067A (ja) | 2005-11-25 | 2014-01-16 | メシル酸イマチニブのｆ、ｇ、ｈ、ｉおよびｋ結晶形 |
Country Status (13)
| Country | Link |
|---|---|
| US (6) | US7893076B2 (https=) |
| EP (3) | EP1960380A1 (https=) |
| JP (2) | JP5844508B2 (https=) |
| KR (4) | KR20130141712A (https=) |
| CN (1) | CN102351842B (https=) |
| AU (2) | AU2006316823A1 (https=) |
| BR (1) | BRPI0618993A2 (https=) |
| CA (3) | CA2824301C (https=) |
| EC (1) | ECSP088473A (https=) |
| MY (1) | MY146403A (https=) |
| NO (1) | NO20082684L (https=) |
| UY (1) | UY29964A1 (https=) |
| WO (1) | WO2007059963A1 (https=) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR047530A1 (es) * | 2004-02-04 | 2006-01-25 | Novartis Ag | Formas de sal de 4-(4-metilpiperazin-1-ilmetil)-n-(4-metil-3-(4-piridin-3-il)pirimidin-2-ilamino)fenil)-benzamida |
| AU2006316823A1 (en) * | 2005-11-25 | 2007-05-31 | Novartis Ag | F,G,H,I and K crystal forms of imatinib mesylate |
| BRPI0817946A2 (pt) * | 2007-09-25 | 2015-05-05 | Teva Pharma | Composições de imatinibe estável |
| RU2365587C1 (ru) * | 2008-02-22 | 2009-08-27 | Закрытое Акционерное Общество "Фарм-Синтез" | Рентгеноаморфная безводная модификация 4-[(4-метил-1-пиперазинил)метил]-n-[4-метил-3-[[4-(3-пиридинил)-2-пиримидинил]-амино]-фенил]бензамида метансульфоната и способ ее получения |
| CZ2009570A3 (cs) | 2009-08-26 | 2011-03-09 | Zentiva, K. S. | Príprava, stabilizace a využití polymorfu imatinib mesylátu pro vývoj lékových forem |
| PL389357A1 (pl) | 2009-10-22 | 2011-04-26 | Tomasz Koźluk | Sole imatinibu z pochodnymi kwasów winowych i sposób ich wytwarzania |
| AU2011213936A1 (en) | 2010-02-15 | 2012-09-06 | Sharma Ashwani | Process for the preparation of alpha form of imatinib mesylate |
| PL390611A1 (pl) | 2010-03-04 | 2011-09-12 | Tomasz Koźluk | Sposób otrzymywania polimorficznej formy alfa i nowa forma polimorficzna mesylanu imatinibu |
| WO2012090221A1 (en) | 2010-12-29 | 2012-07-05 | Cadila Healthcare Limited | Novel salts of imatinib |
| EP2604596A1 (en) * | 2011-12-16 | 2013-06-19 | Deva Holding Anonim Sirketi | Polymorphs of imatinib |
| EP2864313A1 (en) | 2012-06-22 | 2015-04-29 | Basf Se | Multicomponent crystals comprising imatinib mesilate and selected co-crystal formers |
| KR101242955B1 (ko) * | 2012-06-25 | 2013-03-12 | 제일약품주식회사 | 이마티닙 메실레이트 결정형 α의 제조 방법 |
| ES2683361T3 (es) | 2013-05-14 | 2018-09-26 | Hetero Research Foundation | Composiciones de Imatinib |
| WO2015081175A1 (en) * | 2013-11-26 | 2015-06-04 | Children's Medical Center Corporation | Expandable stent valve |
| PL3539138T3 (pl) | 2016-11-11 | 2021-12-13 | Curium Us Llc | Sposoby generowania germanu-68 ze zmniejszoną ilością części lotnych |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW225528B (https=) | 1992-04-03 | 1994-06-21 | Ciba Geigy Ag | |
| CO4940418A1 (es) | 1997-07-18 | 2000-07-24 | Novartis Ag | Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso |
| US20060073185A1 (en) | 2002-12-13 | 2006-04-06 | Bausch & Lomb Incorporated | Method and composition for contact lenses |
| TR200504337T1 (tr) * | 2003-06-02 | 2006-12-21 | Hetero Drugs Limited | Imatinib mezilat'ın yeni polimorfları |
| AR047530A1 (es) | 2004-02-04 | 2006-01-25 | Novartis Ag | Formas de sal de 4-(4-metilpiperazin-1-ilmetil)-n-(4-metil-3-(4-piridin-3-il)pirimidin-2-ilamino)fenil)-benzamida |
| US8048883B2 (en) * | 2004-02-11 | 2011-11-01 | Natco Pharma Limited | Polymorphic form of imatinib mesylate and a process for its preparation |
| UA84462C2 (ru) * | 2004-04-02 | 2008-10-27 | Институт Фармацевтични | Полиморфные модификации кислотно-аддитивных солей иматиниба с метансульфоновой кислотой |
| AP2715A (en) | 2004-06-04 | 2013-07-31 | Bioniche Life Sciences Inc | Use of imatinib to treat liver disorders and viralinfections |
| WO2006024863A1 (en) * | 2004-09-02 | 2006-03-09 | Cipla Limited | Stable crystal form of imatinib mesylate and process for the preparation thereof |
| WO2006048890A1 (en) * | 2004-11-04 | 2006-05-11 | Sun Pharmaceutical Industries Limited | Imatinib mesylate crystal form and process for preparation thereof |
| WO2006054314A1 (en) | 2004-11-17 | 2006-05-26 | Natco Pharma Limited | Polymorphic forms of imatinib mesylate |
| US9804295B2 (en) | 2005-05-05 | 2017-10-31 | Novartis Ag | Ophthalmic devices for sustained delivery of active compounds |
| GB0511066D0 (en) | 2005-05-31 | 2005-07-06 | Novartis Ag | Organic compounds |
| EP1922314A1 (en) * | 2005-08-26 | 2008-05-21 | Novartis AG | Delta and epsilon crystal forms of imatinib mesylate |
| AU2006316823A1 (en) * | 2005-11-25 | 2007-05-31 | Novartis Ag | F,G,H,I and K crystal forms of imatinib mesylate |
-
2006
- 2006-11-23 AU AU2006316823A patent/AU2006316823A1/en not_active Abandoned
- 2006-11-23 KR KR1020137031543A patent/KR20130141712A/ko not_active Ceased
- 2006-11-23 EP EP06818763A patent/EP1960380A1/en not_active Withdrawn
- 2006-11-23 WO PCT/EP2006/011240 patent/WO2007059963A1/en not_active Ceased
- 2006-11-23 KR KR1020137031544A patent/KR20130140909A/ko not_active Ceased
- 2006-11-23 US US12/094,629 patent/US7893076B2/en not_active Expired - Fee Related
- 2006-11-23 KR KR1020087012363A patent/KR20080078804A/ko not_active Ceased
- 2006-11-23 JP JP2008541641A patent/JP5844508B2/ja not_active Expired - Fee Related
- 2006-11-23 CN CN201110232553.6A patent/CN102351842B/zh not_active Expired - Fee Related
- 2006-11-23 CA CA2824301A patent/CA2824301C/en not_active Expired - Fee Related
- 2006-11-23 EP EP12177119A patent/EP2546248A1/en not_active Withdrawn
- 2006-11-23 KR KR1020137031545A patent/KR20130137721A/ko not_active Ceased
- 2006-11-23 EP EP12177131.5A patent/EP2578580A1/en not_active Withdrawn
- 2006-11-23 BR BRPI0618993-8A patent/BRPI0618993A2/pt not_active IP Right Cessation
- 2006-11-23 UY UY29964A patent/UY29964A1/es not_active Application Discontinuation
- 2006-11-23 CA CA2824307A patent/CA2824307C/en not_active Expired - Fee Related
- 2006-11-23 CA CA2628330A patent/CA2628330C/en not_active Expired - Fee Related
- 2006-11-23 MY MYPI20081624A patent/MY146403A/en unknown
-
2008
- 2008-05-20 EC EC2008008473A patent/ECSP088473A/es unknown
- 2008-06-16 NO NO20082684A patent/NO20082684L/no not_active Application Discontinuation
-
2011
- 2011-01-14 US US13/006,505 patent/US8198289B2/en not_active Expired - Fee Related
- 2011-03-22 AU AU2011201286A patent/AU2011201286A1/en not_active Ceased
- 2011-07-15 US US13/183,600 patent/US8846706B2/en not_active Expired - Fee Related
- 2011-07-15 US US13/183,572 patent/US8592440B2/en not_active Expired - Fee Related
- 2011-07-15 US US13/183,557 patent/US8507515B2/en not_active Expired - Fee Related
-
2012
- 2012-05-15 US US13/472,000 patent/US8633213B2/en not_active Expired - Fee Related
-
2014
- 2014-01-16 JP JP2014005741A patent/JP2014074067A/ja active Pending
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