JP2019534706A5 - - Google Patents
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- Publication number
- JP2019534706A5 JP2019534706A5 JP2019520386A JP2019520386A JP2019534706A5 JP 2019534706 A5 JP2019534706 A5 JP 2019534706A5 JP 2019520386 A JP2019520386 A JP 2019520386A JP 2019520386 A JP2019520386 A JP 2019520386A JP 2019534706 A5 JP2019534706 A5 JP 2019534706A5
- Authority
- JP
- Japan
- Prior art keywords
- antibody
- drug conjugate
- seq
- heavy chain
- variable region
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021190070A JP7383682B2 (ja) | 2016-10-17 | 2021-11-24 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2023191037A JP2023184697A (ja) | 2016-10-17 | 2023-11-08 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2025146227A JP2025175010A (ja) | 2016-10-17 | 2025-09-03 | 抗edb抗体および抗体-薬物コンジュゲート |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662409081P | 2016-10-17 | 2016-10-17 | |
| US62/409,081 | 2016-10-17 | ||
| PCT/IB2017/056093 WO2018073680A1 (en) | 2016-10-17 | 2017-10-03 | Anti-edb antibodies and antibody-drug conjugates |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021190070A Division JP7383682B2 (ja) | 2016-10-17 | 2021-11-24 | 抗edb抗体および抗体-薬物コンジュゲート |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019534706A JP2019534706A (ja) | 2019-12-05 |
| JP2019534706A5 true JP2019534706A5 (enExample) | 2020-11-12 |
| JP7039577B2 JP7039577B2 (ja) | 2022-03-22 |
Family
ID=60117722
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019520386A Active JP7039577B2 (ja) | 2016-10-17 | 2017-10-03 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2021190070A Active JP7383682B2 (ja) | 2016-10-17 | 2021-11-24 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2023191037A Pending JP2023184697A (ja) | 2016-10-17 | 2023-11-08 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2025146227A Pending JP2025175010A (ja) | 2016-10-17 | 2025-09-03 | 抗edb抗体および抗体-薬物コンジュゲート |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021190070A Active JP7383682B2 (ja) | 2016-10-17 | 2021-11-24 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2023191037A Pending JP2023184697A (ja) | 2016-10-17 | 2023-11-08 | 抗edb抗体および抗体-薬物コンジュゲート |
| JP2025146227A Pending JP2025175010A (ja) | 2016-10-17 | 2025-09-03 | 抗edb抗体および抗体-薬物コンジュゲート |
Country Status (22)
| Country | Link |
|---|---|
| US (5) | US20190269791A1 (enExample) |
| EP (3) | EP3525828B1 (enExample) |
| JP (4) | JP7039577B2 (enExample) |
| KR (1) | KR102338660B1 (enExample) |
| CN (2) | CN116251196A (enExample) |
| AU (3) | AU2017344440B2 (enExample) |
| CA (1) | CA3040423A1 (enExample) |
| DK (1) | DK3525828T3 (enExample) |
| ES (1) | ES3007557T3 (enExample) |
| FI (1) | FI3525828T3 (enExample) |
| HR (1) | HRP20250056T1 (enExample) |
| HU (1) | HUE070615T2 (enExample) |
| IL (2) | IL310865A (enExample) |
| LT (1) | LT3525828T (enExample) |
| MX (2) | MX2019004434A (enExample) |
| PL (1) | PL3525828T3 (enExample) |
| PT (1) | PT3525828T (enExample) |
| RS (1) | RS66524B1 (enExample) |
| RU (1) | RU2758632C2 (enExample) |
| SG (1) | SG11201903400WA (enExample) |
| SI (1) | SI3525828T1 (enExample) |
| WO (1) | WO2018073680A1 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3824906A1 (en) | 2016-12-21 | 2021-05-26 | Amgen Inc. | Anti-tnf alpha antibody formulations |
| WO2020123425A2 (en) * | 2018-12-12 | 2020-06-18 | Bristol-Myers Squibb Company | Antibodies modified for transglutaminase conjugation, conjugates thereof, and methods and uses |
| KR102614063B1 (ko) | 2020-12-24 | 2023-12-19 | 대화제약 주식회사 | 엑스트라도메인 b 피브로넥틴에 특이적으로 결합하는 신규한 항체 |
| CN112816453B (zh) * | 2021-02-09 | 2022-07-08 | 黑龙江大学 | 蛋白在预测药物性能上的应用 |
| EP4340944A4 (en) * | 2021-05-20 | 2026-04-01 | Univ Case Western Reserve | Specific Peptide and Drug Conjugates of Fibronectin Isotypes for Cancer Therapy |
| EP4370541A1 (en) | 2021-07-14 | 2024-05-22 | 2seventy bio, Inc. | Engineered t cell receptors fused to binding domains from antibodies |
| AU2023248532A1 (en) | 2022-04-08 | 2024-11-21 | Regeneron Pharmaceuticals, Inc. | Multipartite receptor and signaling complexes |
| EP4716555A1 (en) * | 2023-07-10 | 2026-04-01 | Wuxi Xdc Singapore Private Limited | Antibody-drug conjugates and production thereof |
| WO2025149667A1 (en) | 2024-01-12 | 2025-07-17 | Pheon Therapeutics Ltd | Antibody drug conjugates and uses thereof |
| WO2025208105A1 (en) * | 2024-03-29 | 2025-10-02 | Pyxis Oncology, Inc. | Constructs, compositions, and methods for treating extra domain b splice variant of fibronectin-expressing diseases and disorders |
Family Cites Families (37)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5663149A (en) | 1994-12-13 | 1997-09-02 | Arizona Board Of Regents Acting On Behalf Of Arizona State University | Human cancer inhibitory pentapeptide heterocyclic and halophenyl amides |
| WO1997026885A1 (en) | 1996-01-23 | 1997-07-31 | The General Hospital Corporation Doing Business As Massachusetts General Hospital | Benzophenothiazine and benzoporphyrin dye combination photodynamic therapy of tumors |
| GB9610967D0 (en) | 1996-05-24 | 1996-07-31 | Cambridge Antibody Tech | Specific binding members,materials and methods |
| TWI259837B (en) | 1998-05-11 | 2006-08-11 | Eidgenossische Tech Hochscule | Specific binding molecules for scintigraphy, conjugates containing them and therapeutic method for treatment of angiogenesis |
| EP1259548A1 (en) | 2000-02-24 | 2002-11-27 | Eidgenössische Technische Hochschule Zürich | Antibody specific for the ed-b domain of fibronectin, conjugates comprising said antibody, and their use for the detection and treatment of angiogenesis |
| US8623373B2 (en) * | 2000-02-24 | 2014-01-07 | Philogen S.P.A. | Compositions and methods for treatment of angiogenesis in pathological lesions |
| AU2002348477A1 (en) | 2001-05-01 | 2002-12-23 | The General Hospital Corporation | Photoimmunotherapies for cancer using photosensitizer immunoconjugates and combination therapies |
| US6997863B2 (en) | 2001-07-25 | 2006-02-14 | Triton Biosystems, Inc. | Thermotherapy via targeted delivery of nanoscale magnetic particles |
| PL369371A1 (en) * | 2002-01-03 | 2005-04-18 | Schering Aktiengesellschaft | New methods for diagnosis and treatment of tumours |
| ES2337566T3 (es) | 2002-03-11 | 2010-04-27 | Philogen S.P.A. | Anticuerpos derivados de anti ed-b l19 y vasculatura tumoral objetivo. |
| KR20050026033A (ko) * | 2002-07-31 | 2005-03-14 | 쉐링 악티엔게젤샤프트 | 신규 효과기 접합체, 그의 제조 방법 및 그의 약학적 용도 |
| WO2006113546A2 (en) | 2005-04-15 | 2006-10-26 | Neogenix Oncology, Inc. | Recombinant monoclonal antibodies and corresponding antigens for colon and pancreatic cancers |
| MX2007013875A (es) * | 2005-05-11 | 2008-01-28 | Philogen Spa | Proteinas de fusion del anticuerpo l19 contra fibronectina ed-b e interlucina 12. |
| RU2467015C2 (ru) | 2005-10-05 | 2012-11-20 | Коммонвелт Сайентифик Энд Индастриал Рисерч Организейшн | Белки шелка |
| EP1842553A1 (en) | 2006-04-07 | 2007-10-10 | Bayer Schering Pharma Aktiengesellschaft | Combination of an anti-EDb fibronectin domain antibody/IL2 fusion protein and a further small molecule |
| JP2009535372A (ja) * | 2006-05-03 | 2009-10-01 | バイエル・シエーリング・ファーマ アクチエンゲゼルシャフト | 抗edbフィブロネクチンドメイン抗体l19−sip及び抗−egfr−抗体の組合せ |
| TWI412367B (zh) * | 2006-12-28 | 2013-10-21 | 梅達雷克斯有限責任公司 | 化學鏈接劑與可裂解基質以及其之綴合物 |
| CA2682851C (en) | 2007-04-02 | 2017-01-17 | Philogen S.P.A. | A novel antigen associated with the neovasculature of tumour metastases |
| EA017995B1 (ru) | 2007-07-25 | 2013-04-30 | Филоджен С.П.А. | Антиген, связанный с вариантами рака легкого и лимфомами |
| EP2085095B1 (en) | 2008-01-17 | 2012-03-07 | Philogen S.p.A. | Combination of an anti-EDb fibronectin antibody-IL-2 fusion protein, and a molecule binding to B cells, B cell progenitors and/or their cancerous counterpart |
| PL3912643T3 (pl) * | 2009-02-13 | 2023-01-23 | Immunomedics Inc. | Immunokoniugaty z połączeniem rozszczepialnym wewnątrzkomórkowo |
| US8679488B2 (en) | 2009-08-05 | 2014-03-25 | Philogen S.P.A. | Targeting of bone marrow neovasculature |
| RU2583876C2 (ru) | 2009-08-17 | 2016-05-10 | Роше Гликарт Аг | Иммуноконъюгаты направленного действия |
| BR112012014417B1 (pt) | 2009-12-14 | 2021-11-09 | Scil Proteins Gmbh | Proteínas ubiquitinas modificadas tendo uma atividade de ligação específica para o extradomínio b de fibronectina |
| EP3842074A1 (en) | 2010-09-29 | 2021-06-30 | Philogen S.p.A. | Protein-drug conjugates |
| CA2813411C (en) * | 2010-11-05 | 2016-08-02 | Rinat Neuroscience Corporation | Engineered polypeptide conjugates and methods for making thereof using transglutaminase |
| EA201892619A1 (ru) * | 2011-04-29 | 2019-04-30 | Роше Гликарт Аг | Иммуноконъюгаты, содержащие мутантные полипептиды интерлейкина-2 |
| EP2780039B9 (en) | 2011-11-17 | 2018-04-18 | Pfizer Inc | Cytotoxic peptides and antibody drug conjugates thereof |
| EP3539982B1 (en) | 2011-12-23 | 2025-02-19 | Pfizer Inc. | Engineered antibody constant regions for site-specific conjugation and methods and uses therefor |
| EA201591465A1 (ru) * | 2013-02-08 | 2015-12-30 | АйАрЭм ЭлЭлСи | Специфичные участки для модификации антител для получения иммуноконъюгатов |
| EP2988784A1 (en) * | 2013-04-25 | 2016-03-02 | Philogen S.p.A. | Antibody-drug conjugates |
| SG11201605437YA (en) * | 2014-01-27 | 2016-08-30 | Pfizer | Bifunctional cytotoxic agents |
| WO2015114166A2 (en) * | 2014-02-03 | 2015-08-06 | Philochem Ag | Targeted drug conjugates |
| KR20190072663A (ko) * | 2014-04-25 | 2019-06-25 | 리나트 뉴로사이언스 코프. | 약물이 고도로 로딩된 항체-약물 접합체 |
| TW201625689A (zh) | 2014-09-12 | 2016-07-16 | 建南德克公司 | 抗-b7-h4抗體及免疫結合物 |
| TWI812873B (zh) * | 2015-11-30 | 2023-08-21 | 美商輝瑞股份有限公司 | 用於部位專一性接合之抗體和抗體片段 |
| US10689458B2 (en) | 2015-11-30 | 2020-06-23 | Pfizer Inc. | Site specific HER2 antibody drug conjugates |
-
2017
- 2017-10-03 IL IL310865A patent/IL310865A/en unknown
- 2017-10-03 PL PL17784700.1T patent/PL3525828T3/pl unknown
- 2017-10-03 KR KR1020197013908A patent/KR102338660B1/ko active Active
- 2017-10-03 IL IL266112A patent/IL266112B2/en unknown
- 2017-10-03 CN CN202310030234.XA patent/CN116251196A/zh active Pending
- 2017-10-03 PT PT177847001T patent/PT3525828T/pt unknown
- 2017-10-03 FI FIEP17784700.1T patent/FI3525828T3/fi active
- 2017-10-03 CN CN201780078019.XA patent/CN110087691B/zh active Active
- 2017-10-03 SG SG11201903400WA patent/SG11201903400WA/en unknown
- 2017-10-03 EP EP17784700.1A patent/EP3525828B1/en active Active
- 2017-10-03 HU HUE17784700A patent/HUE070615T2/hu unknown
- 2017-10-03 WO PCT/IB2017/056093 patent/WO2018073680A1/en not_active Ceased
- 2017-10-03 ES ES17784700T patent/ES3007557T3/es active Active
- 2017-10-03 AU AU2017344440A patent/AU2017344440B2/en active Active
- 2017-10-03 HR HRP20250056TT patent/HRP20250056T1/hr unknown
- 2017-10-03 MX MX2019004434A patent/MX2019004434A/es unknown
- 2017-10-03 CA CA3040423A patent/CA3040423A1/en active Pending
- 2017-10-03 RS RS20250049A patent/RS66524B1/sr unknown
- 2017-10-03 SI SI201731585T patent/SI3525828T1/sl unknown
- 2017-10-03 RU RU2019111303A patent/RU2758632C2/ru active
- 2017-10-03 US US16/342,275 patent/US20190269791A1/en not_active Abandoned
- 2017-10-03 EP EP25168356.1A patent/EP4635516A3/en active Pending
- 2017-10-03 DK DK17784700.1T patent/DK3525828T3/da active
- 2017-10-03 LT LTEPPCT/IB2017/056093T patent/LT3525828T/lt unknown
- 2017-10-03 EP EP24223209.8A patent/EP4617283A2/en active Pending
- 2017-10-03 JP JP2019520386A patent/JP7039577B2/ja active Active
-
2019
- 2019-04-15 MX MX2024003463A patent/MX2024003463A/es unknown
-
2020
- 2020-10-26 AU AU2020260375A patent/AU2020260375B2/en active Active
-
2021
- 2021-11-24 JP JP2021190070A patent/JP7383682B2/ja active Active
-
2023
- 2023-02-09 US US18/166,774 patent/US11833216B2/en active Active
- 2023-10-23 US US18/492,055 patent/US12653901B2/en active Active
- 2023-10-23 US US18/492,348 patent/US12636377B2/en active Active
- 2023-11-08 JP JP2023191037A patent/JP2023184697A/ja active Pending
- 2023-12-04 US US18/528,539 patent/US20240261423A1/en active Pending
-
2024
- 2024-02-23 AU AU2024201216A patent/AU2024201216A1/en active Pending
-
2025
- 2025-09-03 JP JP2025146227A patent/JP2025175010A/ja active Pending
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