JP2019509286A5 - - Google Patents

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Publication number
JP2019509286A5
JP2019509286A5 JP2018546864A JP2018546864A JP2019509286A5 JP 2019509286 A5 JP2019509286 A5 JP 2019509286A5 JP 2018546864 A JP2018546864 A JP 2018546864A JP 2018546864 A JP2018546864 A JP 2018546864A JP 2019509286 A5 JP2019509286 A5 JP 2019509286A5
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JP
Japan
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composition
crystalline form
form according
chloro
biphenyl
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Application number
JP2018546864A
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English (en)
Japanese (ja)
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JP2019509286A (ja
JP7306828B2 (ja
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Priority claimed from PCT/US2017/021172 external-priority patent/WO2017156009A1/en
Publication of JP2019509286A publication Critical patent/JP2019509286A/ja
Publication of JP2019509286A5 publication Critical patent/JP2019509286A5/ja
Priority to JP2021177448A priority Critical patent/JP2022017433A/ja
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Publication of JP7306828B2 publication Critical patent/JP7306828B2/ja
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JP2018546864A 2016-03-08 2017-03-07 結晶性（２ｓ，４ｒ）－５－（５’－クロロ－２’－フルオロ－［１，１’－ビフェニル］－４－イル）－２－（エトキシメチル）－４－（３－ヒドロキシイソオキサゾール－５－カルボキサミド）－２－メチルペンタン酸およびその使用 Active JP7306828B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021177448A JP2022017433A (ja) 2016-03-08 2021-10-29 結晶性（２ｓ，４ｒ）－５－（５’－クロロ－２’－フルオロ－［１，１’－ビフェニル］－４－イル）－２－（エトキシメチル）－４－（３－ヒドロキシイソオキサゾール－５－カルボキサミド）－２－メチルペンタン酸およびその使用

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662305393P 2016-03-08 2016-03-08
US62/305,393 2016-03-08
US201662346336P 2016-06-06 2016-06-06
US62/346,336 2016-06-06
PCT/US2017/021172 WO2017156009A1 (en) 2016-03-08 2017-03-07 Crystalline(2s,4r)-5-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2-methylpentanoic acid and uses thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021177448A Division JP2022017433A (ja) 2016-03-08 2021-10-29 結晶性（２ｓ，４ｒ）－５－（５’－クロロ－２’－フルオロ－［１，１’－ビフェニル］－４－イル）－２－（エトキシメチル）－４－（３－ヒドロキシイソオキサゾール－５－カルボキサミド）－２－メチルペンタン酸およびその使用

Publications (3)

Publication Number Publication Date
JP2019509286A JP2019509286A (ja) 2019-04-04
JP2019509286A5 true JP2019509286A5 (enExample) 2020-04-02
JP7306828B2 JP7306828B2 (ja) 2023-07-11

Family

ID=58387911

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018546864A Active JP7306828B2 (ja) 2016-03-08 2017-03-07 結晶性（２ｓ，４ｒ）－５－（５’－クロロ－２’－フルオロ－［１，１’－ビフェニル］－４－イル）－２－（エトキシメチル）－４－（３－ヒドロキシイソオキサゾール－５－カルボキサミド）－２－メチルペンタン酸およびその使用
JP2021177448A Pending JP2022017433A (ja) 2016-03-08 2021-10-29 結晶性（２ｓ，４ｒ）－５－（５’－クロロ－２’－フルオロ－［１，１’－ビフェニル］－４－イル）－２－（エトキシメチル）－４－（３－ヒドロキシイソオキサゾール－５－カルボキサミド）－２－メチルペンタン酸およびその使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021177448A Pending JP2022017433A (ja) 2016-03-08 2021-10-29 結晶性（２ｓ，４ｒ）－５－（５’－クロロ－２’－フルオロ－［１，１’－ビフェニル］－４－イル）－２－（エトキシメチル）－４－（３－ヒドロキシイソオキサゾール－５－カルボキサミド）－２－メチルペンタン酸およびその使用

Country Status (30)

Country Link
US (6) US10100021B2 (enExample)
EP (1) EP3408260B1 (enExample)
JP (2) JP7306828B2 (enExample)
KR (2) KR20220035991A (enExample)
CN (1) CN108779084A (enExample)
AU (1) AU2017229466C1 (enExample)
CA (1) CA3015505C (enExample)
CL (1) CL2018002539A1 (enExample)
CO (1) CO2018010568A2 (enExample)
CY (1) CY1124397T1 (enExample)
DK (1) DK3408260T3 (enExample)
ES (1) ES2880123T3 (enExample)
HR (1) HRP20211169T1 (enExample)
HU (1) HUE055546T2 (enExample)
IL (1) IL261244B (enExample)
LT (1) LT3408260T (enExample)
MX (1) MX377177B (enExample)
MY (1) MY198185A (enExample)
PH (1) PH12018501876A1 (enExample)
PL (1) PL3408260T3 (enExample)
PT (1) PT3408260T (enExample)
RS (1) RS62172B1 (enExample)
RU (1) RU2756223C2 (enExample)
SA (1) SA518392325B1 (enExample)
SG (1) SG11201807591VA (enExample)
SI (1) SI3408260T1 (enExample)
SM (1) SMT202100434T1 (enExample)
TW (1) TWI731943B (enExample)
WO (1) WO2017156009A1 (enExample)
ZA (1) ZA201805840B (enExample)

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PT3408260T (pt) 2016-03-08 2021-07-23 Theravance Biopharma R&D Ip Llc Ácido (2s,4r)-5-(5¿-cloro-2¿-fluoro-[1,1¿-bifenil]-4-il)-2- (etoximetil)-4-(3-hidroxi-isoxazole-5-carboxamido)-2- metilpentanoico cristalino e suas utilizações
KR102752382B1 (ko) * 2019-09-20 2025-01-09 심천 사루브리스 퍼머수티칼스 컴퍼니 리미티드 안지오텐신 ii 수용체 길항제 대사물질 및 nep 억제제의 복합체의 심부전 치료에서의 용도
KR102485499B1 (ko) * 2022-07-15 2023-01-09 오가노이드사이언스 주식회사 신장 질환의 치료 또는 예방용 조성물

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