JP2019180396A - 半固形状組成物 - Google Patents
半固形状組成物 Download PDFInfo
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Landscapes
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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Abstract
Description
(1)冷感刺激剤、増粘多糖類及びカフェインを含有し、粘度が1.4〜27Pa・sであることを特徴とする半固形状組成物、
(2)冷感刺激剤が、コハク酸モノメンチル及びエチル−3−p−メンタン−3−カルボキサミドアセテートから選ばれる少なくとも1種である(1)に記載の半固形状組成物、
(3)冷感刺激剤が0.00001〜0.04%W/Wであることを特徴とする(1)又は(2)に記載の半固形状組成物、
(4)増粘多糖類がキサンタンガム、ローカストビーンガム、タラガム、グアーガム、寒天及びカラギーナンからなる群より選ばれる少なくとも1種である(1)に記載の半固形状組成物、
(5)眠気防止用又は集中力維持用の(1)〜(4)に記載の半固形状組成物、
である。
下記表4〜9に記載の処方および次の方法に従い経口組成物を調製した。水にカフェイン、クエン酸、安息香酸ナトリウム、コハク酸モノメンチルまたはエチル−3−p−メンタン−3−カルボキサミドアセテート(表中ではWS−5と表記)、および増粘多糖類を添加、攪拌した後、90℃20分以上の殺菌をかけパウチ容器に充填し、半固形状組成物を得た(実施例1〜15)。コハク酸モノメンチルまたはエチル−3−p−メンタン−3−カルボキサミドアセテートは水に溶解しづらいため、予め2W/V%となるよう95%エタノールに溶解したものを使用した。また、増粘剤を添加しない飲料を対照とした(比較例1〜13)。
はりつき感については、吐き出し直後の口中のはりつき感を表1の通り6段階絶対評価し、パネルの平均値を算出し、さらに、表2の判定基準に従い評価結果を表した。はりつき感とは、口中に含んだ組成物が口腔内で滞留し、口腔粘膜に接したまま剥がれないような感覚である。
冷涼感については、吐き出し後から、冷涼感が完全に消失するまでの時間を記録し、対照サンプルとの持続時間の差の平均値を求めた。さらに、表3に従って評価結果を表した。
事前にパネル間で同じ評価手順でできるよう確認し、はりつき感と冷涼感の持続についても基準のすり合わせを行った。冷涼感については、消失時間の記録漏れを防ぐため、1分ごとに冷涼感を記録したのち、完全に消失するまでの時間を記録した。また、評価は複数日に渡って行われたため、対照サンプルは同じ処方でも複数回評価を行った。
結果を表4〜9に示した。なお、はりつき感(評点)、冷涼感の持続時間(秒)の結果は、パネル3名の平均値を、それぞれ表2、表3に従って示した。
Claims (5)
- 冷感刺激剤、増粘多糖類及びカフェインを含有し、粘度が1.4〜27Pa・sであることを特徴とする半固形状組成物。
- 冷感刺激剤が、コハク酸モノメンチル及びエチル−3−p−メンタン−3−カルボキサミドアセテートから選ばれる少なくとも1種である請求項1に記載の半固形状組成物。
- 冷感刺激剤が0.00001〜0.04%W/Wであることを特徴とする請求項1又は2に記載の半固形状組成物。
- 増粘多糖類がキサンタンガム、ローカストビーンガム、タラガム、グアーガム、寒天及びカラギーナンからなる群より選ばれる少なくとも1種である請求項1に記載の半固形状組成物。
- 眠気防止用又は集中力維持用の請求項1〜4に記載の半固形状組成物。
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