JP2018530566A5 - - Google Patents

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Publication number
JP2018530566A5
JP2018530566A5 JP2018517867A JP2018517867A JP2018530566A5 JP 2018530566 A5 JP2018530566 A5 JP 2018530566A5 JP 2018517867 A JP2018517867 A JP 2018517867A JP 2018517867 A JP2018517867 A JP 2018517867A JP 2018530566 A5 JP2018530566 A5 JP 2018530566A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
linagliptin
tablets
polymorphic form
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2018517867A
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English (en)
Japanese (ja)
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JP2018530566A (ja
JP6839708B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2016/073952 external-priority patent/WO2017060398A1/en
Publication of JP2018530566A publication Critical patent/JP2018530566A/ja
Publication of JP2018530566A5 publication Critical patent/JP2018530566A5/ja
Application granted granted Critical
Publication of JP6839708B2 publication Critical patent/JP6839708B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2018517867A 2015-10-09 2016-10-07 8−[(3r)−3−アミノ−1−ピペリジニル]−7−(2−ブチン−1−イル)−3,7−ジヒドロ−3−メチル−1−[4−メチル−2−キナゾリニル)メチル]−1h−プリン−2,6−ジオンまたは薬学上許容できるその塩を含有する医薬組成物 Expired - Fee Related JP6839708B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15189208.0 2015-10-09
EP15189208 2015-10-09
PCT/EP2016/073952 WO2017060398A1 (en) 2015-10-09 2016-10-07 Pharmaceutical composition containing 8-[(3r)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[4-methyl-2-quinazolinyl)methyl]-1h-purine-2,6-dione or a pharmaceutically acceptable salt thereof

Publications (3)

Publication Number Publication Date
JP2018530566A JP2018530566A (ja) 2018-10-18
JP2018530566A5 true JP2018530566A5 (enExample) 2019-11-07
JP6839708B2 JP6839708B2 (ja) 2021-03-10

Family

ID=54293102

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018517867A Expired - Fee Related JP6839708B2 (ja) 2015-10-09 2016-10-07 8−[(3r)−3−アミノ−1−ピペリジニル]−7−(2−ブチン−1−イル)−3,7−ジヒドロ−3−メチル−1−[4−メチル−2−キナゾリニル)メチル]−1h−プリン−2,6−ジオンまたは薬学上許容できるその塩を含有する医薬組成物

Country Status (8)

Country Link
US (1) US10668073B2 (enExample)
EP (1) EP3359136A1 (enExample)
JP (1) JP6839708B2 (enExample)
CN (1) CN108174596A (enExample)
AU (1) AU2016335082A1 (enExample)
CA (1) CA2998982A1 (enExample)
EA (1) EA037498B1 (enExample)
WO (1) WO2017060398A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020009675A2 (en) 2018-06-01 2020-01-09 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Solid oral pharmaceutical compositions of linagliptin
CN110496129B (zh) * 2018-11-23 2021-06-04 北京中医药大学 利拉利汀的抗肿瘤活性及其新用途
JP7245694B2 (ja) * 2019-03-26 2023-03-24 エルメッド株式会社 リナグリプチン含有医薬組成物及びその製造方法、並びにリナグリプチン含有医薬組成物の品質の向上方法
WO2022102457A1 (ja) * 2020-11-10 2022-05-19 沢井製薬株式会社 リナグリプチン含有口腔内崩壊錠

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101150449B1 (ko) 2002-08-21 2012-06-01 베링거 잉겔하임 파르마 게엠베하 운트 코 카게 8-[3-아미노-피페리딘-1-일]-크산틴, 이의 제조방법 및 이를 포함하는 약제학적 조성물
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
EA030606B1 (ru) 2006-05-04 2018-08-31 Бёрингер Ингельхайм Интернациональ Гмбх Способы приготовления лекарственного средства, содержащего полиморфы
CN102256976A (zh) 2008-12-23 2011-11-23 贝林格尔.英格海姆国际有限公司 有机化合物的盐形式
US20120258170A1 (en) * 2009-05-20 2012-10-11 Nutracryst Therapeutics Private Limited Pharmaceutical co-crystals of quercetin
WO2012152837A1 (en) 2011-05-10 2012-11-15 Sandoz Ag Polymorph of linagliptin benzoate
CN103006663A (zh) * 2011-09-23 2013-04-03 重庆药友制药有限责任公司 一种瑞舒伐他汀钙的药物组合物
CN102631331A (zh) * 2012-04-26 2012-08-15 北京哈三联科技股份有限公司 奥氮平口腔崩解片制剂及其制备方法
EP3311803A1 (en) 2012-08-13 2018-04-25 Sandoz AG Stable pharmaceutical composition containing 8-[(3r)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-1h-purine-2,6-dione or a pharmaceutically acceptable salt thereof
WO2014193528A1 (en) 2013-04-29 2014-12-04 Anovel Pharmaceuticals, Llc Amorphous dosage forms and methods
WO2014184378A1 (en) * 2013-05-16 2014-11-20 Sandoz Ag Tablet with increased drug load of odanacatib
EP2848242A1 (en) 2013-09-12 2015-03-18 Sanovel Ilac Sanayi ve Ticaret A.S. Orally disintegrating formulations of Linagliptin

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