|
ZA859575B
(en)
|
1984-12-21 |
1986-08-27 |
Hoffmann La Roche |
Oxetanones
|
|
FR2692579B1
(fr)
|
1992-06-19 |
1995-06-02 |
Roussel Uclaf |
Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
|
|
FR2718450B1
(fr)
|
1994-04-08 |
1997-01-10 |
Roussel Uclaf |
Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
|
|
JP3652394B2
(ja)
|
1995-01-27 |
2005-05-25 |
高砂香料工業株式会社 |
N−置換−7−アミノ−5−ヒドロキシ−3−オキソヘプタン酸誘導体およびその製造法
|
|
HN1998000074A
(es)
|
1997-06-11 |
1999-01-08 |
Pfizer Prod Inc |
Derivados de macrolidos c-4 sustituidos
|
|
AU7986098A
(en)
|
1997-06-27 |
1999-01-19 |
Merck & Co., Inc. |
9a-aza-3-ketolides, compositions containing such compounds and methods of treatment
|
|
HN1998000159A
(es)
|
1997-10-29 |
1999-02-09 |
Monsanto Co |
Derivados de 9- amino - 3 ceto eritromicina
|
|
GB9814006D0
(en)
|
1998-06-29 |
1998-08-26 |
Biotica Tech Ltd |
Polyketides and their synthesis
|
|
FR2785612A1
(fr)
|
1998-11-10 |
2000-05-12 |
Hoechst Marion Roussel Inc |
Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
|
|
US6262030B1
(en)
*
|
1998-11-03 |
2001-07-17 |
Pfizer Inc. |
Erythromycin derivatives
|
|
US6590083B1
(en)
|
1999-04-16 |
2003-07-08 |
Ortho-Mcneil Pharmaceutical, Inc. |
Ketolide antibacterials
|
|
US6939861B2
(en)
|
1999-04-16 |
2005-09-06 |
Kosan Biosciences, Inc. |
Amido macrolides
|
|
CA2370743A1
(en)
|
1999-04-16 |
2000-10-26 |
Dennis Hlasta |
Ketolide antibacterials
|
|
HRP990116B1
(en)
|
1999-04-20 |
2007-10-31 |
GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. |
NOVEL 8a AND 9a- 15-MEMBERED LACTAMES
|
|
HUP0201516A3
(en)
|
1999-05-24 |
2003-03-28 |
Pfizer Prod Inc |
13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them
|
|
AU6316400A
(en)
|
1999-08-06 |
2001-03-05 |
Taisho Pharmaceutical Co., Ltd. |
Erythromycin a derivatives
|
|
DK1206476T3
(da)
|
1999-08-24 |
2006-05-15 |
Abbott Lab |
9a-azalider med antibakteriel virkning
|
|
BRPI0017013B1
(pt)
|
2000-01-27 |
2015-07-14 |
Zoetis P Llc |
Composição de antibiótico azalídeo e método para sua obtenção
|
|
JP4596591B2
(ja)
|
2000-03-09 |
2010-12-08 |
塩野義製薬株式会社 |
8a−オキサホモエリスロマイシン誘導体、製造方法、合成中間体および医薬組成物
|
|
US6440942B1
(en)
|
2000-12-22 |
2002-08-27 |
Enanta Pharmaceuticals, Inc. |
14-membered macrolides derived from leucomycins
|
|
AU2002346475A1
(en)
|
2001-12-05 |
2003-06-23 |
Ortho-Mcneil Pharmaceutical, Inc. |
6-o-acyl ketolide derivatives of erythromycine useful as antibacterials
|
|
US8063021B2
(en)
|
2002-01-17 |
2011-11-22 |
Kosan Biosciences Incorporated |
Ketolide anti-infective compounds
|
|
BR0316746A
(pt)
|
2002-11-29 |
2005-10-18 |
Mercian Corp |
Método de produção do composto macrolida 11107d, linhagem streptomyces sp.ab-1704 (ferm bp-8551), linhagem mortierella sp. f1529 (ferm bp-8547) ou linhagem f-1530 (ferm bp-8548), e linhagem ab-1896 (ferm bp-8550)
|
|
JPWO2004065346A1
(ja)
|
2003-01-21 |
2006-05-18 |
住友化学株式会社 |
(−)−テトラヒドロリプスタチンおよびその中間体の製造方法
|
|
EP1638549A4
(en)
*
|
2003-03-10 |
2011-06-15 |
Optimer Pharmaceuticals Inc |
NEW ANTIBACTERIAL AGENTS
|
|
CN1530079A
(zh)
|
2003-03-13 |
2004-09-22 |
钱本文 |
中空分叉髓内钉
|
|
HRP20030381B1
(en)
|
2003-05-14 |
2007-05-31 |
GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. |
3-DECLADINOZYL 9a-N-CARBAMOYL AND 9a-N-THIOCARBAMOYL DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICYNE A
|
|
WO2005030227A1
(en)
|
2003-09-23 |
2005-04-07 |
Enanta Pharmaceuticals, Inc. |
9a, 11-3C-BICYCLIC 9a-AZALIDE DERIVATIVES
|
|
US20080287376A1
(en)
|
2004-07-28 |
2008-11-20 |
Mohammad Salman |
Ketolide Derivatives as Antibacterial Agents
|
|
US7767797B1
(en)
|
2004-09-30 |
2010-08-03 |
Synovo Gmbh |
Macrocyclic compounds and methods of use thereof
|
|
US20090170790A1
(en)
|
2004-10-25 |
2009-07-02 |
Biswajit Das |
Ketolide derivatives as antibacterial agents
|
|
US20060096158A1
(en)
|
2004-11-08 |
2006-05-11 |
Robinson J M |
Lactones as new oxygenate fuel additives, fuels based thereon and methods for using same
|
|
CN101103039A
(zh)
|
2005-01-12 |
2008-01-09 |
阿尔法马股份公司 |
作为抗菌剂的红霉素衍生物
|
|
US20100035832A1
(en)
|
2005-01-12 |
2010-02-11 |
Alpharma Aps |
Macrolides
|
|
PT1851236E
(pt)
|
2005-01-13 |
2010-10-25 |
Glaxosmithkline Zagreb |
Macrólidos com actividade anti-inflamatória
|
|
WO2006120541A1
(en)
|
2005-05-10 |
2006-11-16 |
Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. |
Ether linked macrolides useful for the treatment of microbial infections
|
|
RU2008106915A
(ru)
|
2005-07-26 |
2009-09-10 |
Меркле Гмбх (De) |
Макролидные конъюгаты пирролиновых и индолизиновых соединений
|
|
WO2007034909A1
(ja)
|
2005-09-22 |
2007-03-29 |
Kaneka Corporation |
(3r,5r)-7-アミノ-3,5-ジヒドロキシヘプタン酸誘導体の製造法
|
|
JPWO2007043621A1
(ja)
|
2005-10-13 |
2009-04-16 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
プラジエノライドb及びプラジエノライドdの全合成方法
|
|
US8097708B2
(en)
|
2006-02-07 |
2012-01-17 |
Taisho Pharmaceutical Co., Ltd. |
10a-Azalide compound
|
|
AP2009004985A0
(en)
|
2007-03-13 |
2009-10-31 |
Pfizer Prod Inc |
Erythromycin-based macrolides
|
|
EP2214484A4
(en)
|
2007-10-25 |
2013-01-02 |
Cempra Pharmaceuticals Inc |
PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
|
|
US20090209547A1
(en)
|
2008-02-15 |
2009-08-20 |
In Jong Kim |
C-8 halogenated macrolides
|
|
KR100980379B1
(ko)
|
2008-04-02 |
2010-09-06 |
주식회사 파마코스텍 |
광학활성을 갖는 5-히드록시-3-옥소헵타노에이트 유도체의제조방법
|
|
WO2010015703A2
(en)
|
2008-08-07 |
2010-02-11 |
Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. |
Novel 6-o-substituted 15-membered 8a- and 9a-lactams
|
|
JP5711135B2
(ja)
|
2008-10-24 |
2015-04-30 |
センプラ ファーマシューティカルズ,インコーポレイテッド |
胃腸疾患を治療するための方法
|
|
ES2582794T3
(es)
|
2009-08-13 |
2016-09-15 |
Basilea Pharmaceutica Ag |
Nuevos macrólidos y su uso
|
|
ES2608285T3
(es)
|
2009-09-10 |
2017-04-07 |
Cempra Pharmaceuticals, Inc. |
Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC
|
|
ES2637072T3
(es)
|
2010-03-10 |
2017-10-10 |
Cempra Pharmaceuticals, Inc. |
Formulación parenteral de antibióticos macrólidos
|
|
MX361413B
(es)
|
2010-03-22 |
2018-12-05 |
Cempra Pharmaceuticals Inc Star |
Formas cristalinas de un macrólido y usos para las mismas.
|
|
WO2011131749A1
(en)
|
2010-04-23 |
2011-10-27 |
Glaxo Group Limited |
New 14 and 15 membered macrolides for the treatment of neutrophil dominated inflammatory diseases
|
|
CN102917708B
(zh)
|
2010-05-20 |
2015-11-25 |
森普拉制药公司 |
制备大环内酯和酮内酯及其中间体的方法
|
|
US8975232B2
(en)
|
2010-07-29 |
2015-03-10 |
President And Fellows Of Harvard College |
Macrocyclic kinase inhibitors and uses thereof
|
|
US8796474B1
(en)
|
2010-08-23 |
2014-08-05 |
Rutgers, The State University Of New Jersey |
Macrolide compounds and methods and intermediates useful for their preparation
|
|
EP2613630A4
(en)
|
2010-09-10 |
2014-01-15 |
Cempra Pharmaceuticals Inc |
HYDROGEN BOND FOR THE PREPARATION OF FLUOROCHETOLIDES FOR THE TREATMENT OF DISEASES
|
|
EP2625185A4
(en)
|
2010-10-10 |
2014-03-26 |
Synovo Gmbh |
INFLAMMATORY MAKROLIDE
|
|
WO2012127351A1
(en)
|
2011-03-22 |
2012-09-27 |
Wockhardt Limited |
Process for preparation of ketolide compounds
|
|
CN102690297A
(zh)
|
2011-03-22 |
2012-09-26 |
连云港海康生物科技有限公司 |
一种壳寡糖季铵盐及其合成方法
|
|
US9243038B2
(en)
|
2011-07-01 |
2016-01-26 |
President And Fellows Of Harvard College |
Macrocyclic insulin-degrading enzyme (IDE) inhibitors and uses thereof
|
|
NZ700182A
(en)
|
2012-03-27 |
2017-02-24 |
Cempra Pharmaceuticals Inc |
Parenteral formulations for administering macrolide antibiotics
|
|
AU2014239959A1
(en)
*
|
2013-03-14 |
2015-10-01 |
Cempra Pharmaceuticals, Inc. |
Methods for treating respiratory diseases and formulations therefor
|
|
CN105188712A
(zh)
|
2013-03-15 |
2015-12-23 |
森普拉制药公司 |
用于制备大环内酯抗菌剂的收敛方法
|
|
JP6437523B2
(ja)
|
2013-04-04 |
2018-12-12 |
プレジデント アンド フェローズ オブ ハーバード カレッジ |
マクロライドならびにそれらの調製および使用の方法
|
|
CN106998685A
(zh)
|
2014-10-08 |
2017-08-01 |
哈佛大学的校长及成员们 |
14‑元酮内酯及其制备和使用方法
|
|
WO2016154533A1
(en)
|
2015-03-25 |
2016-09-29 |
President And Fellows Of Harvard College |
Synthesis of desosamines
|
|
EP3273969A4
(en)
|
2015-03-25 |
2018-11-21 |
President and Fellows of Harvard College |
Macrolides with modified desosamine sugars and uses thereof
|