JP2017533215A5 - - Google Patents
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- Publication number
- JP2017533215A5 JP2017533215A5 JP2017523293A JP2017523293A JP2017533215A5 JP 2017533215 A5 JP2017533215 A5 JP 2017533215A5 JP 2017523293 A JP2017523293 A JP 2017523293A JP 2017523293 A JP2017523293 A JP 2017523293A JP 2017533215 A5 JP2017533215 A5 JP 2017533215A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- pyrido
- pyrimidin
- amino
- chloro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462069915P | 2014-10-29 | 2014-10-29 | |
| US62/069,915 | 2014-10-29 | ||
| PCT/KR2015/011386 WO2016068580A2 (en) | 2014-10-29 | 2015-10-27 | Novel pyridopyrimidinone compounds for modulating the catalytic activity of histone lysine demethylases (kdms) |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017533215A JP2017533215A (ja) | 2017-11-09 |
| JP2017533215A5 true JP2017533215A5 (https=) | 2018-11-01 |
| JP6505222B2 JP6505222B2 (ja) | 2019-04-24 |
Family
ID=55851908
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017523293A Expired - Fee Related JP6505222B2 (ja) | 2014-10-29 | 2015-10-27 | ヒストンリジン脱メチル化触媒活性を調節するための新規ピリドピリミジノン化合物 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US9834550B2 (https=) |
| EP (1) | EP3212647B1 (https=) |
| JP (1) | JP6505222B2 (https=) |
| KR (1) | KR101978899B1 (https=) |
| CN (1) | CN107001358A (https=) |
| AU (1) | AU2015340215B2 (https=) |
| BR (1) | BR112017008312A2 (https=) |
| CA (1) | CA2962917C (https=) |
| MX (1) | MX2017005346A (https=) |
| NZ (1) | NZ730475A (https=) |
| RU (1) | RU2684396C2 (https=) |
| SG (1) | SG11201702075QA (https=) |
| WO (1) | WO2016068580A2 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3359154B1 (en) * | 2015-10-08 | 2021-05-26 | Suzhou Yunxuan Yiyao Keji Youxian Gongsi | Wnt signaling pathway inhibitors and therapeutic applications thereof |
| JP7114076B2 (ja) | 2015-12-22 | 2022-08-08 | シャイ・セラピューティクス・エルエルシー | がん及び炎症性疾患の処置のための化合物 |
| JP7514005B2 (ja) | 2017-06-21 | 2024-07-10 | シャイ・セラピューティクス・エルエルシー | がん、炎症性疾患、ラソパシー、及び線維性疾患の治療のためのｒａｓスーパーファミリーと相互作用する化合物 |
| CN112119065B (zh) * | 2018-07-13 | 2024-01-23 | 四川科伦博泰生物医药股份有限公司 | 苯并二氮杂环类化合物、其制备方法及用途 |
| JP7407461B2 (ja) | 2018-12-19 | 2024-01-04 | シャイ・セラピューティクス・エルエルシー | がん、炎症性疾患、ｒａｓ病、及び線維性疾患の処置のためのｒａｓスーパーファミリーと相互作用する化合物 |
| US20230110603A1 (en) | 2020-01-31 | 2023-04-13 | Kumiai Chemical Industry Co., Ltd. | 3-alkoxybenzamide derivative, and pest control agent |
| WO2021198191A1 (en) | 2020-03-30 | 2021-10-07 | Enyo Pharma | Quinazolinone derivatives and uses thereof for treating a cancer |
| US20230150978A1 (en) * | 2020-03-30 | 2023-05-18 | Enyo Pharma | Quinazolinone derivatives and uses thereof for treating a cancer |
| GB202114315D0 (en) * | 2021-10-06 | 2021-11-17 | Duke Street Bio Ltd | Pharmaceutical compound |
| US20240217968A1 (en) * | 2021-03-31 | 2024-07-04 | Duke Street Bio Limited | Pharmaceutical compound |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5939421A (en) * | 1997-07-01 | 1999-08-17 | Signal Pharmaceuticals, Inc. | Quinazoline analogs and related compounds and methods for treating inflammatory conditions |
| GB9909135D0 (en) * | 1999-04-22 | 1999-06-16 | Univ Wales Medicine | Cystic fibrosis medicaments |
| MXPA04004955A (es) * | 2001-11-26 | 2004-08-11 | Dsm Ip Assets Bv | Procedimiento para la recuperacion de caprolactama. |
| FR2846657B1 (fr) | 2002-11-05 | 2004-12-24 | Servier Lab | Nouveaux composes pyridopyrimidinone, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| US7232824B2 (en) * | 2003-09-30 | 2007-06-19 | Scios, Inc. | Quinazoline derivatives as medicaments |
| NZ546477A (en) * | 2006-04-07 | 2009-04-30 | Auckland Uniservices Ltd | 4-Alkylamino-2-(heterocyclic)quinazolines and their use in cancer therapy |
| WO2013012915A1 (en) * | 2011-07-19 | 2013-01-24 | Infinity Pharmaceuticals Inc. | Heterocyclic compounds and uses thereof |
| US9914730B2 (en) * | 2012-09-28 | 2018-03-13 | Cancer Research Technology Limited | Azaquinazoline inhibitors of Atypical protein Kinase C |
| RS55764B1 (sr) | 2012-10-02 | 2017-07-31 | Gilead Sciences | Inhibitori histonskih demetilaza |
| US20150272939A1 (en) | 2012-10-02 | 2015-10-01 | Yale University | Identification of Small Molecule Inhibitors of Jumonji AT-Rich Interactive Domain 1A (JARID1A) and 1B (JARID1B) Histone Demethylase |
| WO2014087165A1 (en) * | 2012-12-06 | 2014-06-12 | University Of Bath | Tankyrase inhibitors |
| CA2901022C (en) | 2013-02-27 | 2021-05-04 | Epitherapeutics Aps | Substituted pyridine compounds as inhibitors of histone demethylases |
| JP6320506B2 (ja) | 2013-03-12 | 2018-05-09 | セルジーン クオンティセル リサーチ，インク． | ヒストンデメチラーゼ阻害剤 |
| WO2014139326A1 (en) | 2013-03-13 | 2014-09-18 | Genentech, Inc. | Pyrazolo compounds and uses thereof |
| HRP20171609T1 (hr) | 2013-03-15 | 2017-12-15 | Quanticel Pharmaceuticals Inc | Inhibitori histon demetilaze |
| MX2016002794A (es) | 2013-09-05 | 2016-09-13 | Genentech Inc | Compuestos antiproliferativos. |
| CN103694255A (zh) * | 2014-01-09 | 2014-04-02 | 华中师范大学 | 吡啶并噁嗪酮和吡啶并嘧啶酮类化合物及其制备方法与应用 |
| TWI675836B (zh) * | 2014-03-25 | 2019-11-01 | 美商伊格尼塔公司 | 非典型蛋白質激酶ｃ之氮雜喹唑啉抑制劑 |
-
2015
- 2015-10-27 NZ NZ730475A patent/NZ730475A/en unknown
- 2015-10-27 CA CA2962917A patent/CA2962917C/en active Active
- 2015-10-27 BR BR112017008312A patent/BR112017008312A2/pt not_active Application Discontinuation
- 2015-10-27 EP EP15853996.5A patent/EP3212647B1/en not_active Not-in-force
- 2015-10-27 AU AU2015340215A patent/AU2015340215B2/en active Active
- 2015-10-27 MX MX2017005346A patent/MX2017005346A/es unknown
- 2015-10-27 US US14/923,525 patent/US9834550B2/en active Active
- 2015-10-27 RU RU2017113007A patent/RU2684396C2/ru active
- 2015-10-27 WO PCT/KR2015/011386 patent/WO2016068580A2/en not_active Ceased
- 2015-10-27 JP JP2017523293A patent/JP6505222B2/ja not_active Expired - Fee Related
- 2015-10-27 SG SG11201702075QA patent/SG11201702075QA/en unknown
- 2015-10-27 KR KR1020177014472A patent/KR101978899B1/ko not_active Expired - Fee Related
- 2015-10-27 CN CN201580061545.6A patent/CN107001358A/zh active Pending
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