JP2016527184A5 - - Google Patents
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- Publication number
- JP2016527184A5 JP2016527184A5 JP2016514421A JP2016514421A JP2016527184A5 JP 2016527184 A5 JP2016527184 A5 JP 2016527184A5 JP 2016514421 A JP2016514421 A JP 2016514421A JP 2016514421 A JP2016514421 A JP 2016514421A JP 2016527184 A5 JP2016527184 A5 JP 2016527184A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- branched
- nme
- och
- straight
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB201309405A GB201309405D0 (en) | 2013-05-24 | 2013-05-24 | Pharmaceutical compound |
| GB1309405.7 | 2013-05-24 | ||
| GB201402341A GB201402341D0 (en) | 2014-02-11 | 2014-02-11 | Pharmaceutical compound |
| GB1402341.0 | 2014-02-11 | ||
| PCT/EP2014/060586 WO2014187922A1 (en) | 2013-05-24 | 2014-05-22 | Slc2a transporter inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016527184A JP2016527184A (ja) | 2016-09-08 |
| JP2016527184A5 true JP2016527184A5 (enExample) | 2017-06-29 |
Family
ID=50771498
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016514421A Pending JP2016527184A (ja) | 2013-05-24 | 2014-05-22 | Slc2a輸送体阻害剤 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20160120863A1 (enExample) |
| EP (1) | EP3004088A1 (enExample) |
| JP (1) | JP2016527184A (enExample) |
| SG (1) | SG11201509650YA (enExample) |
| WO (1) | WO2014187922A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2999852A1 (en) * | 2015-09-29 | 2017-04-06 | Oncotherapy Science, Inc. | Bicyclic compound and use thereof for inhibiting suv39h2 |
| WO2017097671A1 (de) | 2015-12-10 | 2017-06-15 | Bayer Pharma Aktiengesellschaft | Substituierte perhydropyrrolo[3,4-c]pyrrol-derivate und ihre verwendung |
| CU20180056A7 (es) * | 2015-12-10 | 2018-10-04 | Bayer Pharma AG | Derivados de 2-fenil-3-(piperazinometil)imidazo(1,2-a)piridina como bloqueadores de los canales task-1 y task-2 para el tratamiento de trastornos respiratorios |
| JOP20190005A1 (ar) | 2016-07-20 | 2019-01-20 | Bayer Ag | مركبات ديازاهيترو ثنائية الحلقة مستبدلة واستخداماتها |
| WO2018227427A1 (en) * | 2017-06-14 | 2018-12-20 | Bayer Aktiengesellschaft | Substituted bridged diazepane derivatives and use thereof |
| JOP20190284A1 (ar) * | 2017-06-14 | 2019-12-11 | Bayer Pharma AG | مركبات إيميدازوبيريميدين مستبدلة بديازا ثنائي الحلقة واستخدامها للمعالجة من اضطرابات التنفس |
| LT3860998T (lt) | 2018-10-05 | 2024-06-25 | Annapurna Bio Inc. | Junginiai ir kompozicijos, skirti gydyti būkles, susijusias su apj receptoriaus aktyvumu |
| KR102797127B1 (ko) * | 2018-12-29 | 2025-04-21 | 우한 크리에이터나 사이언스 앤드 테크놀로지 컴퍼니, 리미티드 | 헤테로고리계 화합물, 중간체, 이의 제조 방법 및 용도 |
| JP2022108114A (ja) * | 2021-01-12 | 2022-07-25 | 株式会社スタイルアンドバリュージャパン | オートファジー誘導剤 |
| CA3216716A1 (en) | 2021-05-03 | 2022-11-10 | Tim BERGBREDE | Composition comprising an inhibitor of mitochondrial transcription |
| CN114457045B (zh) * | 2022-02-25 | 2023-07-14 | 中国人民解放军军事科学院军事医学研究院 | 抑制Slc2a1的RNAi腺相关病毒及其制备和应用 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3318880A (en) * | 1963-04-30 | 1967-05-09 | Selvi & C Lab Bioterapico | Novel[1, 2-alpha]imidazopyridines and a process for the manufacture thereof |
| FR1536351A (fr) * | 1967-07-03 | 1968-08-27 | Pyridylimidazopyridines | |
| GB8305245D0 (en) * | 1983-02-25 | 1983-03-30 | Fujisawa Pharmaceutical Co | Imidazo-heterocyclic compounds |
| FR2568880B1 (fr) | 1984-08-07 | 1986-12-12 | Synthelabo | Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
| JP2775282B2 (ja) * | 1989-03-14 | 1998-07-16 | 日清製粉株式会社 | 紅麹の製造法 |
| JP2003095942A (ja) * | 2001-09-21 | 2003-04-03 | Ito En Ltd | 脂肪細胞におけるグルコース取込阻害剤及びglut4トランスロケーション抑制剤、筋肉細胞におけるグルコース取込活性化剤並びに脂肪軽減飲食物 |
| FR2857966A1 (fr) * | 2003-07-24 | 2005-01-28 | Aventis Pharma Sa | Produits aryl-heteroaromatiques, compositions les contenant et utilisation |
| JP5242885B2 (ja) * | 2004-05-20 | 2013-07-24 | 株式会社 伊藤園 | 筋肉内ampk活性化剤 |
| AR056187A1 (es) * | 2005-03-21 | 2007-09-26 | S Bio Pte Ltd | Derivados de imidazo[1,2-a)piridina: preparacion, composiciones farmaceuticas y uso para preparar medicamentos |
| US7345178B2 (en) * | 2005-08-04 | 2008-03-18 | Sirtris Pharmaceuticals, Inc. | Sirtuin modulating compounds |
| US7855201B2 (en) * | 2005-12-06 | 2010-12-21 | Merck Sharp & Dohme. Corp. | Morpholine carboxamide prokineticin receptor antagonists |
| CA2672960A1 (en) * | 2006-12-20 | 2008-07-10 | Schering Corporation | Novel jnk inhibitors |
| EP1974729A1 (en) * | 2007-03-28 | 2008-10-01 | Santhera Pharmaceuticals (Schweiz) AG | Substituted imidazopyridine derivates as melanocortin- 4 receptor antagonists |
| AU2009249186B2 (en) | 2008-05-19 | 2014-05-22 | Sunovion Pharmaceuticals Inc. | Imidazo [1, 2-a] pyridine compounds as GABA-A receptor modulators |
| JP2014509616A (ja) * | 2011-03-31 | 2014-04-21 | エーエムベーエルエーエム テクノロジー トランスファー ゲーエムベーハー | 治療用イミダゾ[1,2−a]ピリジン化合物 |
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2014
- 2014-05-22 WO PCT/EP2014/060586 patent/WO2014187922A1/en not_active Ceased
- 2014-05-22 US US14/893,513 patent/US20160120863A1/en not_active Abandoned
- 2014-05-22 JP JP2016514421A patent/JP2016527184A/ja active Pending
- 2014-05-22 SG SG11201509650YA patent/SG11201509650YA/en unknown
- 2014-05-22 EP EP14725702.6A patent/EP3004088A1/en not_active Withdrawn