JP2016527184A5 - - Google Patents

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Publication number
JP2016527184A5
JP2016527184A5 JP2016514421A JP2016514421A JP2016527184A5 JP 2016527184 A5 JP2016527184 A5 JP 2016527184A5 JP 2016514421 A JP2016514421 A JP 2016514421A JP 2016514421 A JP2016514421 A JP 2016514421A JP 2016527184 A5 JP2016527184 A5 JP 2016527184A5
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JP
Japan
Prior art keywords
group
branched
nme
och
straight
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2016514421A
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English (en)
Japanese (ja)
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JP2016527184A (ja
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Publication date
Priority claimed from GB201309405A external-priority patent/GB201309405D0/en
Priority claimed from GB201402341A external-priority patent/GB201402341D0/en
Application filed filed Critical
Priority claimed from PCT/EP2014/060586 external-priority patent/WO2014187922A1/en
Publication of JP2016527184A publication Critical patent/JP2016527184A/ja
Publication of JP2016527184A5 publication Critical patent/JP2016527184A5/ja
Pending legal-status Critical Current

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JP2016514421A 2013-05-24 2014-05-22 Slc2a輸送体阻害剤 Pending JP2016527184A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB201309405A GB201309405D0 (en) 2013-05-24 2013-05-24 Pharmaceutical compound
GB1309405.7 2013-05-24
GB201402341A GB201402341D0 (en) 2014-02-11 2014-02-11 Pharmaceutical compound
GB1402341.0 2014-02-11
PCT/EP2014/060586 WO2014187922A1 (en) 2013-05-24 2014-05-22 Slc2a transporter inhibitors

Publications (2)

Publication Number Publication Date
JP2016527184A JP2016527184A (ja) 2016-09-08
JP2016527184A5 true JP2016527184A5 (enExample) 2017-06-29

Family

ID=50771498

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016514421A Pending JP2016527184A (ja) 2013-05-24 2014-05-22 Slc2a輸送体阻害剤

Country Status (5)

Country Link
US (1) US20160120863A1 (enExample)
EP (1) EP3004088A1 (enExample)
JP (1) JP2016527184A (enExample)
SG (1) SG11201509650YA (enExample)
WO (1) WO2014187922A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2999852A1 (en) * 2015-09-29 2017-04-06 Oncotherapy Science, Inc. Bicyclic compound and use thereof for inhibiting suv39h2
WO2017097671A1 (de) 2015-12-10 2017-06-15 Bayer Pharma Aktiengesellschaft Substituierte perhydropyrrolo[3,4-c]pyrrol-derivate und ihre verwendung
CU20180056A7 (es) * 2015-12-10 2018-10-04 Bayer Pharma AG Derivados de 2-fenil-3-(piperazinometil)imidazo(1,2-a)piridina como bloqueadores de los canales task-1 y task-2 para el tratamiento de trastornos respiratorios
JOP20190005A1 (ar) 2016-07-20 2019-01-20 Bayer Ag مركبات ديازاهيترو ثنائية الحلقة مستبدلة واستخداماتها
WO2018227427A1 (en) * 2017-06-14 2018-12-20 Bayer Aktiengesellschaft Substituted bridged diazepane derivatives and use thereof
JOP20190284A1 (ar) * 2017-06-14 2019-12-11 Bayer Pharma AG مركبات إيميدازوبيريميدين مستبدلة بديازا ثنائي الحلقة واستخدامها للمعالجة من اضطرابات التنفس
LT3860998T (lt) 2018-10-05 2024-06-25 Annapurna Bio Inc. Junginiai ir kompozicijos, skirti gydyti būkles, susijusias su apj receptoriaus aktyvumu
KR102797127B1 (ko) * 2018-12-29 2025-04-21 우한 크리에이터나 사이언스 앤드 테크놀로지 컴퍼니, 리미티드 헤테로고리계 화합물, 중간체, 이의 제조 방법 및 용도
JP2022108114A (ja) * 2021-01-12 2022-07-25 株式会社スタイルアンドバリュージャパン オートファジー誘導剤
CA3216716A1 (en) 2021-05-03 2022-11-10 Tim BERGBREDE Composition comprising an inhibitor of mitochondrial transcription
CN114457045B (zh) * 2022-02-25 2023-07-14 中国人民解放军军事科学院军事医学研究院 抑制Slc2a1的RNAi腺相关病毒及其制备和应用

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3318880A (en) * 1963-04-30 1967-05-09 Selvi & C Lab Bioterapico Novel[1, 2-alpha]imidazopyridines and a process for the manufacture thereof
FR1536351A (fr) * 1967-07-03 1968-08-27 Pyridylimidazopyridines
GB8305245D0 (en) * 1983-02-25 1983-03-30 Fujisawa Pharmaceutical Co Imidazo-heterocyclic compounds
FR2568880B1 (fr) 1984-08-07 1986-12-12 Synthelabo Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
JP2775282B2 (ja) * 1989-03-14 1998-07-16 日清製粉株式会社 紅麹の製造法
JP2003095942A (ja) * 2001-09-21 2003-04-03 Ito En Ltd 脂肪細胞におけるグルコース取込阻害剤及びglut4トランスロケーション抑制剤、筋肉細胞におけるグルコース取込活性化剤並びに脂肪軽減飲食物
FR2857966A1 (fr) * 2003-07-24 2005-01-28 Aventis Pharma Sa Produits aryl-heteroaromatiques, compositions les contenant et utilisation
JP5242885B2 (ja) * 2004-05-20 2013-07-24 株式会社 伊藤園 筋肉内ampk活性化剤
AR056187A1 (es) * 2005-03-21 2007-09-26 S Bio Pte Ltd Derivados de imidazo[1,2-a)piridina: preparacion, composiciones farmaceuticas y uso para preparar medicamentos
US7345178B2 (en) * 2005-08-04 2008-03-18 Sirtris Pharmaceuticals, Inc. Sirtuin modulating compounds
US7855201B2 (en) * 2005-12-06 2010-12-21 Merck Sharp & Dohme. Corp. Morpholine carboxamide prokineticin receptor antagonists
CA2672960A1 (en) * 2006-12-20 2008-07-10 Schering Corporation Novel jnk inhibitors
EP1974729A1 (en) * 2007-03-28 2008-10-01 Santhera Pharmaceuticals (Schweiz) AG Substituted imidazopyridine derivates as melanocortin- 4 receptor antagonists
AU2009249186B2 (en) 2008-05-19 2014-05-22 Sunovion Pharmaceuticals Inc. Imidazo [1, 2-a] pyridine compounds as GABA-A receptor modulators
JP2014509616A (ja) * 2011-03-31 2014-04-21 エーエムベーエルエーエム テクノロジー トランスファー ゲーエムベーハー 治療用イミダゾ[1,2−a]ピリジン化合物

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