JP2016527184A - Slc2a輸送体阻害剤 - Google Patents
Slc2a輸送体阻害剤 Download PDFInfo
- Publication number
- JP2016527184A JP2016527184A JP2016514421A JP2016514421A JP2016527184A JP 2016527184 A JP2016527184 A JP 2016527184A JP 2016514421 A JP2016514421 A JP 2016514421A JP 2016514421 A JP2016514421 A JP 2016514421A JP 2016527184 A JP2016527184 A JP 2016527184A
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
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- Diabetes (AREA)
- Neurology (AREA)
- Hematology (AREA)
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- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Tropical Medicine & Parasitology (AREA)
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- Rheumatology (AREA)
- Heart & Thoracic Surgery (AREA)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB201309405A GB201309405D0 (en) | 2013-05-24 | 2013-05-24 | Pharmaceutical compound |
| GB1309405.7 | 2013-05-24 | ||
| GB201402341A GB201402341D0 (en) | 2014-02-11 | 2014-02-11 | Pharmaceutical compound |
| GB1402341.0 | 2014-02-11 | ||
| PCT/EP2014/060586 WO2014187922A1 (en) | 2013-05-24 | 2014-05-22 | Slc2a transporter inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016527184A true JP2016527184A (ja) | 2016-09-08 |
| JP2016527184A5 JP2016527184A5 (enExample) | 2017-06-29 |
Family
ID=50771498
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016514421A Pending JP2016527184A (ja) | 2013-05-24 | 2014-05-22 | Slc2a輸送体阻害剤 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20160120863A1 (enExample) |
| EP (1) | EP3004088A1 (enExample) |
| JP (1) | JP2016527184A (enExample) |
| SG (1) | SG11201509650YA (enExample) |
| WO (1) | WO2014187922A1 (enExample) |
Cited By (1)
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| JP2022108114A (ja) * | 2021-01-12 | 2022-07-25 | 株式会社スタイルアンドバリュージャパン | オートファジー誘導剤 |
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| US10759794B2 (en) * | 2015-12-10 | 2020-09-01 | Bayer Pharma Aktiengesellschaft | 2-phenyl-3-(piperazinomethyl)imidazo[1,2-A]pyridine derivatives as blockers of task-1 and task-2 channels, for the treatment of sleep-related breathing disorders |
| JOP20190005A1 (ar) | 2016-07-20 | 2019-01-20 | Bayer Ag | مركبات ديازاهيترو ثنائية الحلقة مستبدلة واستخداماتها |
| WO2018227427A1 (en) * | 2017-06-14 | 2018-12-20 | Bayer Aktiengesellschaft | Substituted bridged diazepane derivatives and use thereof |
| JOP20190284A1 (ar) * | 2017-06-14 | 2019-12-11 | Bayer Pharma AG | مركبات إيميدازوبيريميدين مستبدلة بديازا ثنائي الحلقة واستخدامها للمعالجة من اضطرابات التنفس |
| RS65335B1 (sr) | 2018-10-05 | 2024-04-30 | Annapurna Bio Inc | Jedinjenja i kompozicije za lečenje stanja povezanih sa aktivnošću receptora apj |
| US20240034729A9 (en) * | 2018-12-29 | 2024-02-01 | Wuhan Ll Science And Technology Development Co., Ltd. | Heterocyclic compound, intermediate, preparation method therefor and application thereof |
| US20240252454A1 (en) | 2021-05-03 | 2024-08-01 | Lead Discovery Center Gmbh | Composition comprising an inhibitor of mitochondrial transcription |
| CN114457045B (zh) * | 2022-02-25 | 2023-07-14 | 中国人民解放军军事科学院军事医学研究院 | 抑制Slc2a1的RNAi腺相关病毒及其制备和应用 |
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- 2014-05-22 US US14/893,513 patent/US20160120863A1/en not_active Abandoned
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2022108114A (ja) * | 2021-01-12 | 2022-07-25 | 株式会社スタイルアンドバリュージャパン | オートファジー誘導剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2014187922A1 (en) | 2014-11-27 |
| EP3004088A1 (en) | 2016-04-13 |
| US20160120863A1 (en) | 2016-05-05 |
| SG11201509650YA (en) | 2015-12-30 |
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