JP2016505019A5 - - Google Patents

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JP2016505019A5
JP2016505019A5 JP2015552887A JP2015552887A JP2016505019A5 JP 2016505019 A5 JP2016505019 A5 JP 2016505019A5 JP 2015552887 A JP2015552887 A JP 2015552887A JP 2015552887 A JP2015552887 A JP 2015552887A JP 2016505019 A5 JP2016505019 A5 JP 2016505019A5
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deuterium
compound according
disease
pharmaceutically acceptable
enriched compound
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JP2015552887A
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JP2016505019A (ja
JP6359563B2 (ja
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Priority claimed from PCT/US2014/011440 external-priority patent/WO2014110558A1/en
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JP2015552887A 2013-01-14 2014-01-14 ３−（５置換−４−オキソキナゾリン−３（４ｈ）−イル）−３−ジュウテロピペリジン−２，６−ジオン誘導体 Active JP6359563B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361752055P 2013-01-14 2013-01-14
US61/752,055 2013-01-14
US201361786024P 2013-03-14 2013-03-14
US61/786,024 2013-03-14
PCT/US2014/011440 WO2014110558A1 (en) 2013-01-14 2014-01-14 3-(5-substituted-4-oxoquinazolin-3(4h)-yl)-3-deutero-piperidine-2,6-dione derivatives

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JP2018116936A Division JP6749364B2 (ja) 2013-01-14 2018-06-20 ３−（５置換−４−オキソキナゾリン−３（４ｈ）−イル）−３−ジュウテロピペリジン−２，６−ジオン誘導体

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JP2016505019A JP2016505019A (ja) 2016-02-18
JP2016505019A5 true JP2016505019A5 (enExample) 2017-02-16
JP6359563B2 JP6359563B2 (ja) 2018-07-18

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JP2015552887A Active JP6359563B2 (ja) 2013-01-14 2014-01-14 ３−（５置換−４−オキソキナゾリン−３（４ｈ）−イル）−３−ジュウテロピペリジン−２，６−ジオン誘導体
JP2018116936A Active JP6749364B2 (ja) 2013-01-14 2018-06-20 ３−（５置換−４−オキソキナゾリン−３（４ｈ）−イル）−３−ジュウテロピペリジン−２，６−ジオン誘導体

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JP2018116936A Active JP6749364B2 (ja) 2013-01-14 2018-06-20 ３−（５置換−４−オキソキナゾリン−３（４ｈ）−イル）−３−ジュウテロピペリジン−２，６−ジオン誘導体

Country Status (6)

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US (5) US9540340B2 (enExample)
EP (1) EP2943201B2 (enExample)
JP (2) JP6359563B2 (enExample)
AU (1) AU2014205043B2 (enExample)
CA (1) CA2935495C (enExample)
WO (1) WO2014110558A1 (enExample)

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CN116670118B (zh) 2020-11-13 2026-02-06 伊尼制药公司 二氯苯酚hsd17b13抑制剂及其用途
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WO2014039421A1 (en) 2012-09-04 2014-03-13 Celgene Corporation Isotopologues of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4h)-yl) piperidine-2-6-dione and methods of preparation thereof
CN104797256A (zh) 2012-09-10 2015-07-22 细胞基因公司 用于治疗局部晚期乳腺癌的方法
AU2014205043B2 (en) * 2013-01-14 2018-10-04 Deuterx, Llc 3-(5-substituted-4-oxoquinazolin-3(4h)-yl)-3-deutero-piperidine-2,6-dione derivatives
US9695145B2 (en) 2013-01-22 2017-07-04 Celgene Corporation Processes for the preparation of isotopologues of 3-(4-((4- morpholinomethyl)benzyl)oxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione and pharmaceutically acceptable salts thereof
AU2014236597A1 (en) 2013-03-14 2015-09-24 Deuterx, Llc 3-(substituted-4-oxo-quinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives

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