JP2016503058A5 - - Google Patents

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Publication number
JP2016503058A5
JP2016503058A5 JP2015549612A JP2015549612A JP2016503058A5 JP 2016503058 A5 JP2016503058 A5 JP 2016503058A5 JP 2015549612 A JP2015549612 A JP 2015549612A JP 2015549612 A JP2015549612 A JP 2015549612A JP 2016503058 A5 JP2016503058 A5 JP 2016503058A5
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JP
Japan
Prior art keywords
composition
formula
compound
thiosulfate
amount
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2015549612A
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English (en)
Japanese (ja)
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JP6373867B2 (ja
JP2016503058A (ja
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Priority claimed from PCT/US2013/076041 external-priority patent/WO2014100135A1/en
Publication of JP2016503058A publication Critical patent/JP2016503058A/ja
Publication of JP2016503058A5 publication Critical patent/JP2016503058A5/ja
Application granted granted Critical
Publication of JP6373867B2 publication Critical patent/JP6373867B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015549612A 2012-12-19 2013-12-18 Lfa−1阻害剤製剤 Active JP6373867B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261739609P 2012-12-19 2012-12-19
US61/739,609 2012-12-19
US201361758147P 2013-01-29 2013-01-29
US61/758,147 2013-01-29
PCT/US2013/076041 WO2014100135A1 (en) 2012-12-19 2013-12-18 Lfa-1 inhibitor formulations

Publications (3)

Publication Number Publication Date
JP2016503058A JP2016503058A (ja) 2016-02-01
JP2016503058A5 true JP2016503058A5 (enExample) 2016-07-28
JP6373867B2 JP6373867B2 (ja) 2018-08-15

Family

ID=50979140

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015549612A Active JP6373867B2 (ja) 2012-12-19 2013-12-18 Lfa−1阻害剤製剤

Country Status (20)

Country Link
US (2) US11058677B2 (enExample)
EP (2) EP2934510B1 (enExample)
JP (1) JP6373867B2 (enExample)
KR (1) KR101891144B1 (enExample)
CN (1) CN104955453B (enExample)
AU (1) AU2013361579B2 (enExample)
BR (1) BR112015014367B1 (enExample)
CA (1) CA2894170C (enExample)
DK (1) DK2934510T3 (enExample)
EA (2) EA201791321A1 (enExample)
ES (1) ES2846724T3 (enExample)
HU (1) HUE052299T2 (enExample)
IL (1) IL239490B (enExample)
MX (2) MX391620B (enExample)
NZ (1) NZ708821A (enExample)
PL (1) PL2934510T3 (enExample)
PT (1) PT2934510T (enExample)
SI (1) SI2934510T1 (enExample)
WO (1) WO2014100135A1 (enExample)
ZA (2) ZA201504404B (enExample)

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CN106995439B (zh) * 2016-01-26 2019-09-20 镇江圣安医药有限公司 氘取代3-(甲磺酰基)-l-苯丙氨酸衍生物及其药物组合物、药物制剂和用途
WO2019171260A1 (en) * 2018-03-09 2019-09-12 Mankind Pharma Ltd. Pharmaceutical composition of lifitegrast
KR20220003555A (ko) * 2019-04-18 2022-01-10 아주라 오프탈믹스 엘티디 안구 장애의 치료를 위한 화합물 및 방법
EP3842032A1 (en) 2019-12-24 2021-06-30 Warszawskie Zaklady Farmaceutyczne Polfa S.A. A pharmaceutical formulation
CN116635032A (zh) * 2020-10-21 2023-08-22 阿祖拉眼科有限公司 用于治疗眼部病症的化合物和方法
CN116211796A (zh) * 2022-12-30 2023-06-06 新领先(重庆)医药科技有限公司 一种立他司特滴眼液及其制备方法
KR20240109779A (ko) * 2023-01-05 2024-07-12 주식회사 종근당 리피테그라스트와 토코페롤을 함유하는 건성안 예방 또는 치료용 약제학적 조성물
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WO2025093739A1 (en) 2023-11-02 2025-05-08 Novaliq Gmbh Semifluorinated alkane compositions comprising lifitegrast
US20250161294A1 (en) * 2023-11-17 2025-05-22 Bausch + Lomb Ireland Limited Compositions and methods for treatment of ocular disorders
CN117771174B (zh) * 2023-12-29 2025-07-29 鲁南贝特制药有限公司 一种立他司特滴眼液及其制备方法

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