JP2016503058A5 - - Google Patents
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- Publication number
- JP2016503058A5 JP2016503058A5 JP2015549612A JP2015549612A JP2016503058A5 JP 2016503058 A5 JP2016503058 A5 JP 2016503058A5 JP 2015549612 A JP2015549612 A JP 2015549612A JP 2015549612 A JP2015549612 A JP 2015549612A JP 2016503058 A5 JP2016503058 A5 JP 2016503058A5
- Authority
- JP
- Japan
- Prior art keywords
- composition
- formula
- compound
- thiosulfate
- amount
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261739609P | 2012-12-19 | 2012-12-19 | |
| US61/739,609 | 2012-12-19 | ||
| US201361758147P | 2013-01-29 | 2013-01-29 | |
| US61/758,147 | 2013-01-29 | ||
| PCT/US2013/076041 WO2014100135A1 (en) | 2012-12-19 | 2013-12-18 | Lfa-1 inhibitor formulations |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016503058A JP2016503058A (ja) | 2016-02-01 |
| JP2016503058A5 true JP2016503058A5 (enExample) | 2016-07-28 |
| JP6373867B2 JP6373867B2 (ja) | 2018-08-15 |
Family
ID=50979140
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015549612A Active JP6373867B2 (ja) | 2012-12-19 | 2013-12-18 | Ｌｆａ−１阻害剤製剤 |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US11058677B2 (enExample) |
| EP (2) | EP3827823A1 (enExample) |
| JP (1) | JP6373867B2 (enExample) |
| KR (1) | KR101891144B1 (enExample) |
| CN (1) | CN104955453B (enExample) |
| AU (1) | AU2013361579B2 (enExample) |
| BR (1) | BR112015014367B1 (enExample) |
| CA (1) | CA2894170C (enExample) |
| DK (1) | DK2934510T3 (enExample) |
| EA (2) | EA201791321A1 (enExample) |
| ES (1) | ES2846724T3 (enExample) |
| HU (1) | HUE052299T2 (enExample) |
| IL (1) | IL239490B (enExample) |
| MX (2) | MX391620B (enExample) |
| NZ (1) | NZ708821A (enExample) |
| PL (1) | PL2934510T3 (enExample) |
| PT (1) | PT2934510T (enExample) |
| SI (1) | SI2934510T1 (enExample) |
| WO (1) | WO2014100135A1 (enExample) |
| ZA (2) | ZA201504404B (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN106995439B (zh) * | 2016-01-26 | 2019-09-20 | 镇江圣安医药有限公司 | 氘取代3-(甲磺酰基)-l-苯丙氨酸衍生物及其药物组合物、药物制剂和用途 |
| WO2019171260A1 (en) * | 2018-03-09 | 2019-09-12 | Mankind Pharma Ltd. | Pharmaceutical composition of lifitegrast |
| CN114025759A (zh) * | 2019-04-18 | 2022-02-08 | 阿祖拉眼科有限公司 | 用于治疗眼病的化合物和方法 |
| EP3842032A1 (en) | 2019-12-24 | 2021-06-30 | Warszawskie Zaklady Farmaceutyczne Polfa S.A. | A pharmaceutical formulation |
| US20230399317A1 (en) * | 2020-10-21 | 2023-12-14 | Azura Ophthalmics Ltd. | Compounds and methods for the treatment of ocular disorders |
| CN116211796A (zh) * | 2022-12-30 | 2023-06-06 | 新领先(重庆)医药科技有限公司 | 一种立他司特滴眼液及其制备方法 |
| KR20240109779A (ko) * | 2023-01-05 | 2024-07-12 | 주식회사 종근당 | 리피테그라스트와 토코페롤을 함유하는 건성안 예방 또는 치료용 약제학적 조성물 |
| KR20250033790A (ko) | 2023-09-01 | 2025-03-10 | 주식회사 와이에스생명과학 | 리피테그라스트 함유 점안 조성물 |
| WO2025093739A1 (en) | 2023-11-02 | 2025-05-08 | Novaliq Gmbh | Semifluorinated alkane compositions comprising lifitegrast |
| WO2025104294A1 (en) * | 2023-11-17 | 2025-05-22 | Bausch + Lomb Ireland Limited | Semifluorinated alkane small molecule lfa-1 antagonist combination compositions for treatment of ocular disorders |
| CN117771174B (zh) * | 2023-12-29 | 2025-07-29 | 鲁南贝特制药有限公司 | 一种立他司特滴眼液及其制备方法 |
Family Cites Families (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2694719A (en) | 1949-02-12 | 1954-11-16 | Opplt Jan | Method of stabilizing ascorbic acid with alkali-thiosulfate-carbamide-complexes |
| ES2098739T3 (es) * | 1992-05-13 | 1997-05-01 | Sandoz Ltd | Composiciones oftalmicas conteniendo una cyclosporin. |
| US5429819A (en) * | 1992-10-14 | 1995-07-04 | Matsushita Electric Industrial Co., Ltd. | Antiviral composition |
| IT1277707B1 (it) * | 1995-12-22 | 1997-11-11 | Chemedica Sa | Formulazione oftalmica a base di ialuronato di sodio per uso nella chirurgia oculare |
| JP4138910B2 (ja) * | 1997-07-02 | 2008-08-27 | 帝國製薬株式会社 | 経皮吸収性が良好で且つ皮膚刺激性の少ない塩酸アゼラスチン含有経皮製剤 |
| RU2149611C1 (ru) * | 1998-04-06 | 2000-05-27 | Московская медицинская академия им. И.М. Сеченова | Капли для лечения воспалительных заболеваний глаз (варианты) |
| DE19954516A1 (de) * | 1999-11-12 | 2001-05-17 | Boehringer Ingelheim Int | Epinastin-haltige Lösungen |
| US6258814B1 (en) * | 2000-10-13 | 2001-07-10 | Schering Corporation | Method of using cetirizine and pharmaceutical compositions containing the same for inducing sleep |
| US8877168B1 (en) * | 2002-07-31 | 2014-11-04 | Senju Pharmaceuticals Co., Ltd. | Aqueous liquid preparations and light-stabilized aqueous liquid preparations |
| JP2007528857A (ja) * | 2003-07-11 | 2007-10-18 | ミリアド ジェネティクス， インコーポレイテッド | アルツハイマー病の処置のための薬学的方法、投与レジメンおよび投薬形態 |
| FI119361B (fi) | 2003-09-26 | 2008-10-31 | Raute Oyj | Menetelmä viilun sorvaamiseksi |
| US20060073172A1 (en) * | 2004-10-01 | 2006-04-06 | Schneider L W | Stabilized ophthalmic solution for the treatment of glaucoma and lowering intraocular pressure |
| CN102617557A (zh) * | 2005-05-17 | 2012-08-01 | 萨可德生物科学公司 | 治疗眼病的组合物和方法 |
| JP5315051B2 (ja) * | 2005-07-08 | 2013-10-16 | 千寿製薬株式会社 | オロパタジンを含む眼科用経皮吸収型製剤 |
| US7544893B2 (en) | 2007-07-25 | 2009-06-09 | Thomas & Betts International, Inc. | Extruded wire duct end cap |
| ITRM20080182A1 (it) * | 2008-04-07 | 2009-10-08 | Medivis S R L | Preparato oftalmico a base di dorzolamide e latanoprost per il trattamento topico del glaucoma. |
| CN102056485A (zh) | 2008-04-15 | 2011-05-11 | 萨可德公司 | 用于局部治疗免疫相关疾病的局部lfa-1拮抗剂 |
| US8080562B2 (en) * | 2008-04-15 | 2011-12-20 | Sarcode Bioscience Inc. | Crystalline pharmaceutical and methods of preparation and use thereof |
| JP2011518155A (ja) * | 2008-04-15 | 2011-06-23 | サーコード コーポレイション | 免疫関連障害の局所治療に使用するためのエアゾール化ｌｆａ−１アンタゴニスト |
| US20120028929A1 (en) * | 2008-09-19 | 2012-02-02 | Alacrity Bioscience, Inc. | Tetracycline stabilizing formulations |
| EP2346520B1 (en) * | 2008-11-17 | 2014-11-26 | Laila Pharmaceuticals Pvt. Ltd. | Curcuminoids and its metabolites for the application in ocular diseases |
| UA104320C2 (ru) * | 2009-06-10 | 2014-01-27 | Общество С Ограниченной Ответственностью "Мимотех" | Фармацевтическая композиция на основе митохондриально-адресованного антиоксиданта для применения в медицинской и ветеринарной офтальмологии |
| KR20110001103A (ko) * | 2009-06-29 | 2011-01-06 | 에스케이케미칼주식회사 | 보관 안정성이 향상된 톨테로딘 함유 경피 투여 조성물 |
| NZ600263A (en) * | 2009-11-23 | 2014-08-29 | Allergan Inc | 7-[3,5-dihydroxy-2- (3-hydroxy-5-phenyl-pent-1-enyl)- cyclopentyl]-n-ethyl-hept-5-enamide (bimatoprost) in crystalline form ii, methods for preparation, and methods for use thereof |
| US20120190653A1 (en) * | 2011-01-20 | 2012-07-26 | Dow Pharmaceutical Sciences, Inc. | Therapeutic eye drop comprising doxycycline and a stabilizer |
| WO2012111029A2 (en) * | 2011-02-18 | 2012-08-23 | M/S. Appasamy Associates | Ophthalmic composition for enabling dilation of pupils |
| WO2013003825A1 (en) * | 2011-06-29 | 2013-01-03 | Allergan, Inc. | Alcaftadine for use in the treatment of urticaria |
| ES2978927T3 (es) * | 2012-03-29 | 2024-09-23 | Epion Therapeutics Inc | Soluciones de tratamiento ocular, dispositivos de administración y métodos de aumento de la administración |
| CN103230583A (zh) * | 2013-05-17 | 2013-08-07 | 江西省创欣药业集团有限公司 | 兽用治疗肠道疾病的烟酸诺氟沙星复方注射液及制备方法 |
-
2013
- 2013-12-18 US US14/650,955 patent/US11058677B2/en active Active
- 2013-12-18 NZ NZ708821A patent/NZ708821A/en unknown
- 2013-12-18 PT PT138657572T patent/PT2934510T/pt unknown
- 2013-12-18 EA EA201791321A patent/EA201791321A1/ru unknown
- 2013-12-18 EP EP20204080.4A patent/EP3827823A1/en not_active Withdrawn
- 2013-12-18 EA EA201591180A patent/EA028008B1/ru unknown
- 2013-12-18 ES ES13865757T patent/ES2846724T3/es active Active
- 2013-12-18 CA CA2894170A patent/CA2894170C/en active Active
- 2013-12-18 DK DK13865757.2T patent/DK2934510T3/da active
- 2013-12-18 WO PCT/US2013/076041 patent/WO2014100135A1/en not_active Ceased
- 2013-12-18 CN CN201380071760.5A patent/CN104955453B/zh active Active
- 2013-12-18 BR BR112015014367-9A patent/BR112015014367B1/pt active IP Right Grant
- 2013-12-18 MX MX2019012375A patent/MX391620B/es unknown
- 2013-12-18 JP JP2015549612A patent/JP6373867B2/ja active Active
- 2013-12-18 MX MX2015007540A patent/MX368876B/es active IP Right Grant
- 2013-12-18 AU AU2013361579A patent/AU2013361579B2/en active Active
- 2013-12-18 PL PL13865757T patent/PL2934510T3/pl unknown
- 2013-12-18 EP EP13865757.2A patent/EP2934510B1/en active Active
- 2013-12-18 HU HUE13865757A patent/HUE052299T2/hu unknown
- 2013-12-18 KR KR1020157019352A patent/KR101891144B1/ko active Active
- 2013-12-18 SI SI201331833T patent/SI2934510T1/sl unknown
-
2015
- 2015-06-18 IL IL239490A patent/IL239490B/en active IP Right Grant
- 2015-06-18 ZA ZA2015/04404A patent/ZA201504404B/en unknown
-
2016
- 2016-11-22 ZA ZA2016/08069A patent/ZA201608069B/en unknown
-
2021
- 2021-06-09 US US17/342,631 patent/US20220000859A1/en not_active Abandoned
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