NZ708821A - Lfa-1 inhibitor formulations - Google Patents

Lfa-1 inhibitor formulations

Info

Publication number
NZ708821A
NZ708821A NZ708821A NZ70882113A NZ708821A NZ 708821 A NZ708821 A NZ 708821A NZ 708821 A NZ708821 A NZ 708821A NZ 70882113 A NZ70882113 A NZ 70882113A NZ 708821 A NZ708821 A NZ 708821A
Authority
NZ
New Zealand
Prior art keywords
lfa
inhibitor formulations
compound
formula
treatment
Prior art date
Application number
NZ708821A
Other languages
English (en)
Inventor
Mary Newman
William Hunke
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50979140&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ708821(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NZ708821A publication Critical patent/NZ708821A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
NZ708821A 2012-12-19 2013-12-18 Lfa-1 inhibitor formulations NZ708821A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261739609P 2012-12-19 2012-12-19
US201361758147P 2013-01-29 2013-01-29
PCT/US2013/076041 WO2014100135A1 (en) 2012-12-19 2013-12-18 Lfa-1 inhibitor formulations

Publications (1)

Publication Number Publication Date
NZ708821A true NZ708821A (en) 2020-03-27

Family

ID=50979140

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ708821A NZ708821A (en) 2012-12-19 2013-12-18 Lfa-1 inhibitor formulations

Country Status (20)

Country Link
US (2) US11058677B2 (enExample)
EP (2) EP3827823A1 (enExample)
JP (1) JP6373867B2 (enExample)
KR (1) KR101891144B1 (enExample)
CN (1) CN104955453B (enExample)
AU (1) AU2013361579B2 (enExample)
BR (1) BR112015014367B1 (enExample)
CA (1) CA2894170C (enExample)
DK (1) DK2934510T3 (enExample)
EA (2) EA201791321A1 (enExample)
ES (1) ES2846724T3 (enExample)
HU (1) HUE052299T2 (enExample)
IL (1) IL239490B (enExample)
MX (2) MX391620B (enExample)
NZ (1) NZ708821A (enExample)
PL (1) PL2934510T3 (enExample)
PT (1) PT2934510T (enExample)
SI (1) SI2934510T1 (enExample)
WO (1) WO2014100135A1 (enExample)
ZA (2) ZA201504404B (enExample)

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EP3842032A1 (en) 2019-12-24 2021-06-30 Warszawskie Zaklady Farmaceutyczne Polfa S.A. A pharmaceutical formulation
CN116635032A (zh) * 2020-10-21 2023-08-22 阿祖拉眼科有限公司 用于治疗眼部病症的化合物和方法
CN116211796A (zh) * 2022-12-30 2023-06-06 新领先(重庆)医药科技有限公司 一种立他司特滴眼液及其制备方法
KR20240109779A (ko) * 2023-01-05 2024-07-12 주식회사 종근당 리피테그라스트와 토코페롤을 함유하는 건성안 예방 또는 치료용 약제학적 조성물
KR20250033790A (ko) 2023-09-01 2025-03-10 주식회사 와이에스생명과학 리피테그라스트 함유 점안 조성물
KR20260109029A (ko) 2023-11-02 2026-07-09 노바리크 게엠베하 리피테그라스트를 포함하는 세미플루오르화 알칸 조성물
CN122349415A (zh) * 2023-11-17 2026-07-07 博士伦爱尔兰有限公司 用于治疗眼部病症的半氟化烷烃小分子lfa-1拮抗剂复方组合物
CN117771174B (zh) * 2023-12-29 2025-07-29 鲁南贝特制药有限公司 一种立他司特滴眼液及其制备方法

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KR20120085330A (ko) * 2009-11-23 2012-07-31 알러간, 인코포레이티드 결정형 ｉｉ의 ７?〔３,５?다이하이드록시?２?(３?하이드록시?５?페닐?펜트?１?에닐)?사이클로펜틸〕?ｎ?에틸?헵트?５?엔아마이드(비마토프로스트), 그의 제조방법 및 이용방법
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Also Published As

Publication number Publication date
PT2934510T (pt) 2021-01-13
CA2894170C (en) 2021-08-10
EP2934510A4 (en) 2016-08-17
HK1214963A1 (en) 2016-08-12
MX368876B (es) 2019-10-21
ES2846724T3 (es) 2021-07-29
EP3827823A1 (en) 2021-06-02
IL239490B (en) 2018-12-31
JP2016503058A (ja) 2016-02-01
US20220000859A1 (en) 2022-01-06
EA028008B1 (ru) 2017-09-29
CN104955453B (zh) 2018-09-18
CN104955453A (zh) 2015-09-30
BR112015014367B1 (pt) 2022-11-22
IL239490A0 (en) 2015-08-31
ZA201608069B (en) 2017-11-29
KR101891144B1 (ko) 2018-08-23
WO2014100135A1 (en) 2014-06-26
HK1214536A1 (zh) 2016-07-29
AU2013361579A1 (en) 2015-06-18
EP2934510B1 (en) 2020-10-28
PL2934510T3 (pl) 2021-07-05
EA201791321A1 (ru) 2018-04-30
US20150320737A1 (en) 2015-11-12
CA2894170A1 (en) 2014-06-26
SI2934510T1 (sl) 2021-02-26
JP6373867B2 (ja) 2018-08-15
BR112015014367A2 (pt) 2017-07-11
US11058677B2 (en) 2021-07-13
KR20150100763A (ko) 2015-09-02
DK2934510T3 (da) 2021-01-25
ZA201504404B (en) 2020-01-29
EA201591180A1 (ru) 2015-12-30
MX391620B (es) 2025-03-19
MX2019012375A (es) 2020-01-20
MX2015007540A (es) 2016-04-13
AU2013361579B2 (en) 2018-05-24
HUE052299T2 (hu) 2021-04-28
EP2934510A1 (en) 2015-10-28

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Legal Events

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ASS Change of ownership

Owner name: NOVARTIS AG, CH

Effective date: 20200217

PSEA Patent sealed
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Effective date: 20201119

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Owner name: BAUSCH + LOMB IRELAND LIMITED, IE

Effective date: 20231222

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