MX391620B - Formulaciones del inhibidor del antígeno-1 asociado a la función de linfocitos (lfa-1). - Google Patents

Formulaciones del inhibidor del antígeno-1 asociado a la función de linfocitos (lfa-1).

Info

Publication number
MX391620B
MX391620B MX2019012375A MX2019012375A MX391620B MX 391620 B MX391620 B MX 391620B MX 2019012375 A MX2019012375 A MX 2019012375A MX 2019012375 A MX2019012375 A MX 2019012375A MX 391620 B MX391620 B MX 391620B
Authority
MX
Mexico
Prior art keywords
lfa
associated antigen
lymphocyte function
inhibitor formulations
compound
Prior art date
Application number
MX2019012375A
Other languages
English (en)
Spanish (es)
Other versions
MX2019012375A (es
Inventor
Mary Newman
William Hunke
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50979140&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX391620(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2019012375A publication Critical patent/MX2019012375A/es
Publication of MX391620B publication Critical patent/MX391620B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
MX2019012375A 2012-12-19 2013-12-18 Formulaciones del inhibidor del antígeno-1 asociado a la función de linfocitos (lfa-1). MX391620B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261739609P 2012-12-19 2012-12-19
US201361758147P 2013-01-29 2013-01-29
PCT/US2013/076041 WO2014100135A1 (en) 2012-12-19 2013-12-18 Lfa-1 inhibitor formulations

Publications (2)

Publication Number Publication Date
MX2019012375A MX2019012375A (es) 2020-01-20
MX391620B true MX391620B (es) 2025-03-19

Family

ID=50979140

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2019012375A MX391620B (es) 2012-12-19 2013-12-18 Formulaciones del inhibidor del antígeno-1 asociado a la función de linfocitos (lfa-1).
MX2015007540A MX368876B (es) 2012-12-19 2013-12-18 Formulaciones del inhibidor del antígeno-1 asociado a la función de linfocitos (lfa-1).

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2015007540A MX368876B (es) 2012-12-19 2013-12-18 Formulaciones del inhibidor del antígeno-1 asociado a la función de linfocitos (lfa-1).

Country Status (20)

Country Link
US (2) US11058677B2 (enExample)
EP (2) EP3827823A1 (enExample)
JP (1) JP6373867B2 (enExample)
KR (1) KR101891144B1 (enExample)
CN (1) CN104955453B (enExample)
AU (1) AU2013361579B2 (enExample)
BR (1) BR112015014367B1 (enExample)
CA (1) CA2894170C (enExample)
DK (1) DK2934510T3 (enExample)
EA (2) EA201791321A1 (enExample)
ES (1) ES2846724T3 (enExample)
HU (1) HUE052299T2 (enExample)
IL (1) IL239490B (enExample)
MX (2) MX391620B (enExample)
NZ (1) NZ708821A (enExample)
PL (1) PL2934510T3 (enExample)
PT (1) PT2934510T (enExample)
SI (1) SI2934510T1 (enExample)
WO (1) WO2014100135A1 (enExample)
ZA (2) ZA201504404B (enExample)

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WO2019171260A1 (en) * 2018-03-09 2019-09-12 Mankind Pharma Ltd. Pharmaceutical composition of lifitegrast
JP7700045B2 (ja) * 2019-04-18 2025-06-30 アズーラ オフサルミックス エルティーディー. 眼障害を処置するための化合物および方法
EP3842032A1 (en) 2019-12-24 2021-06-30 Warszawskie Zaklady Farmaceutyczne Polfa S.A. A pharmaceutical formulation
CN116635032A (zh) * 2020-10-21 2023-08-22 阿祖拉眼科有限公司 用于治疗眼部病症的化合物和方法
CN116211796A (zh) * 2022-12-30 2023-06-06 新领先(重庆)医药科技有限公司 一种立他司特滴眼液及其制备方法
KR20240109779A (ko) * 2023-01-05 2024-07-12 주식회사 종근당 리피테그라스트와 토코페롤을 함유하는 건성안 예방 또는 치료용 약제학적 조성물
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WO2025093739A1 (en) 2023-11-02 2025-05-08 Novaliq Gmbh Semifluorinated alkane compositions comprising lifitegrast
US20250161294A1 (en) * 2023-11-17 2025-05-22 Bausch + Lomb Ireland Limited Compositions and methods for treatment of ocular disorders
CN117771174B (zh) * 2023-12-29 2025-07-29 鲁南贝特制药有限公司 一种立他司特滴眼液及其制备方法

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Also Published As

Publication number Publication date
AU2013361579B2 (en) 2018-05-24
IL239490B (en) 2018-12-31
BR112015014367A2 (pt) 2017-07-11
JP2016503058A (ja) 2016-02-01
NZ708821A (en) 2020-03-27
MX2019012375A (es) 2020-01-20
EA201591180A1 (ru) 2015-12-30
CA2894170C (en) 2021-08-10
KR101891144B1 (ko) 2018-08-23
KR20150100763A (ko) 2015-09-02
ZA201504404B (en) 2020-01-29
PT2934510T (pt) 2021-01-13
ZA201608069B (en) 2017-11-29
US20150320737A1 (en) 2015-11-12
DK2934510T3 (da) 2021-01-25
HK1214536A1 (zh) 2016-07-29
HUE052299T2 (hu) 2021-04-28
SI2934510T1 (sl) 2021-02-26
MX368876B (es) 2019-10-21
CA2894170A1 (en) 2014-06-26
JP6373867B2 (ja) 2018-08-15
CN104955453B (zh) 2018-09-18
IL239490A0 (en) 2015-08-31
EP2934510A1 (en) 2015-10-28
US20220000859A1 (en) 2022-01-06
MX2015007540A (es) 2016-04-13
ES2846724T3 (es) 2021-07-29
CN104955453A (zh) 2015-09-30
EA201791321A1 (ru) 2018-04-30
EP3827823A1 (en) 2021-06-02
EP2934510A4 (en) 2016-08-17
HK1214963A1 (en) 2016-08-12
AU2013361579A1 (en) 2015-06-18
EP2934510B1 (en) 2020-10-28
US11058677B2 (en) 2021-07-13
PL2934510T3 (pl) 2021-07-05
EA028008B1 (ru) 2017-09-29
BR112015014367B1 (pt) 2022-11-22
WO2014100135A1 (en) 2014-06-26

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