JP2015520152A5 - - Google Patents

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Publication number
JP2015520152A5
JP2015520152A5 JP2015511772A JP2015511772A JP2015520152A5 JP 2015520152 A5 JP2015520152 A5 JP 2015520152A5 JP 2015511772 A JP2015511772 A JP 2015511772A JP 2015511772 A JP2015511772 A JP 2015511772A JP 2015520152 A5 JP2015520152 A5 JP 2015520152A5
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JP
Japan
Prior art keywords
aryl
membered heterocyclyl
membered
alkyl
carbazol
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JP2015511772A
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English (en)
Japanese (ja)
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JP2015520152A (ja
JP6377054B2 (ja
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Priority claimed from PCT/US2013/040604 external-priority patent/WO2013170186A1/en
Publication of JP2015520152A publication Critical patent/JP2015520152A/ja
Publication of JP2015520152A5 publication Critical patent/JP2015520152A5/ja
Application granted granted Critical
Publication of JP6377054B2 publication Critical patent/JP6377054B2/ja
Expired - Fee Related legal-status Critical Current
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JP2015511772A 2012-05-11 2013-05-10 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド Expired - Fee Related JP6377054B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261645918P 2012-05-11 2012-05-11
US61/645,918 2012-05-11
US201361778176P 2013-03-12 2013-03-12
US61/778,176 2013-03-12
PCT/US2013/040604 WO2013170186A1 (en) 2012-05-11 2013-05-10 Carbazole-containing sulfonamides as cryptochrome modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017140820A Division JP2017200946A (ja) 2012-05-11 2017-07-20 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド

Publications (3)

Publication Number Publication Date
JP2015520152A JP2015520152A (ja) 2015-07-16
JP2015520152A5 true JP2015520152A5 (https=) 2017-02-09
JP6377054B2 JP6377054B2 (ja) 2018-08-22

Family

ID=48444649

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2015511772A Expired - Fee Related JP6377054B2 (ja) 2012-05-11 2013-05-10 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2017140820A Withdrawn JP2017200946A (ja) 2012-05-11 2017-07-20 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2019015689A Withdrawn JP2019077722A (ja) 2012-05-11 2019-01-31 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2020159390A Withdrawn JP2020203948A (ja) 2012-05-11 2020-09-24 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2022166167A Pending JP2023002659A (ja) 2012-05-11 2022-10-17 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド

Family Applications After (4)

Application Number Title Priority Date Filing Date
JP2017140820A Withdrawn JP2017200946A (ja) 2012-05-11 2017-07-20 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2019015689A Withdrawn JP2019077722A (ja) 2012-05-11 2019-01-31 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2020159390A Withdrawn JP2020203948A (ja) 2012-05-11 2020-09-24 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド
JP2022166167A Pending JP2023002659A (ja) 2012-05-11 2022-10-17 クリプトクロム調節薬としてのカルバゾール含有スルホンアミド

Country Status (15)

Country Link
US (3) US9265772B2 (https=)
EP (1) EP2855458B1 (https=)
JP (5) JP6377054B2 (https=)
KR (1) KR102136431B1 (https=)
CN (2) CN107674071B (https=)
AR (1) AR092319A1 (https=)
AU (1) AU2013259294B2 (https=)
CA (1) CA2873214C (https=)
IL (1) IL235602A0 (https=)
MX (1) MX361457B (https=)
NZ (2) NZ701702A (https=)
RU (1) RU2654484C1 (https=)
SG (1) SG11201407402TA (https=)
TW (2) TWI643845B (https=)
WO (1) WO2013170186A1 (https=)

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CN107674071B (zh) * 2012-05-11 2021-12-31 同步制药公司 作为隐花色素调节剂的含有咔唑的磺酰胺类
GB201309333D0 (en) 2013-05-23 2013-07-10 Agency Science Tech & Res Purine diones as WNT pathway modulators
JP2016540001A (ja) * 2013-12-13 2016-12-22 アラーガン、インコーポレイテッドAllergan,Incorporated ステロイド様化合物の多形形態並びにその製造方法及びその用途
TWI690521B (zh) * 2014-04-07 2020-04-11 美商同步製藥公司 作為隱花色素調節劑之含有咔唑之醯胺類、胺基甲酸酯類及脲類
KR101542324B1 (ko) * 2014-04-09 2015-08-05 동아대학교 산학협력단 손상된 dna의 회복 속도 비교를 위한 정보 제공 방법
EP3152185B1 (en) * 2014-06-04 2023-10-04 Roche Diagnostics GmbH Method and usage of a salt for separating epimers by ion mobility spectrometry
JP6975184B2 (ja) 2016-07-04 2021-12-01 バイエル・クロップサイエンス・アクチェンゲゼルシャフト ベンゾスルタム類及び類似体、並びに、殺菌剤としてのそれらの使用
CN107941976B (zh) * 2017-09-28 2019-11-19 浙江新化化工股份有限公司 一种2-甲氧基环己胺的含量测定方法
JP7187152B2 (ja) * 2018-01-12 2022-12-12 三星電子株式会社 化合物、有機エレクトロルミネッセンス素子用材料、有機エレクトロルミネッセンス素子用組成物、有機エレクトロルミネッセンス素子、及び化合物の製造方法
US10947236B2 (en) 2018-08-14 2021-03-16 Osteoqc Inc. Pyrrolo-dipyridine compounds
US20220081433A1 (en) * 2018-09-05 2022-03-17 Assembly Biosciences, Inc. Cyclic sulfamide compounds for treatment of hbv
CN109232596B (zh) * 2018-09-05 2020-03-17 大连九信精细化工有限公司 一种二苯并呋喃咔唑的合成方法
US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
CN114854803A (zh) * 2022-04-21 2022-08-05 山东农业大学 镰刀菌对3,6-二氯咔唑生物降解的方法
CN115974763B (zh) * 2022-12-26 2025-03-11 常州大学 一种咔唑衍生物及其应用
CN116217467B (zh) * 2023-03-09 2026-03-10 烟台皓元生物医药科技有限公司 一种erdrp-0519的中间体及其制备方法
WO2025183207A1 (ja) * 2024-02-28 2025-09-04 国立大学法人京都大学 がん免疫を活性化するスペルミジン誘導体
WO2025239319A1 (ja) * 2024-05-13 2025-11-20 国立大学法人東海国立大学機構 概日時計タンパク質cryに作用するフェニルピラゾール骨格を有する化合物を含有する経粘膜摂取剤

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