JP2014532754A5 - - Google Patents
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- Publication number
- JP2014532754A5 JP2014532754A5 JP2014540612A JP2014540612A JP2014532754A5 JP 2014532754 A5 JP2014532754 A5 JP 2014532754A5 JP 2014540612 A JP2014540612 A JP 2014540612A JP 2014540612 A JP2014540612 A JP 2014540612A JP 2014532754 A5 JP2014532754 A5 JP 2014532754A5
- Authority
- JP
- Japan
- Prior art keywords
- oxo
- dihydro
- compound
- ylmethyl
- oxazolidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C(N(*)C(C(C1=O)=C2)=[U]C(C3**(BCC(CN4C5=IC(NC(C*6)=O)=C6C=C5)OC4=O)*3)=C2[Mn])=C1I#C Chemical compound *C(N(*)C(C(C1=O)=C2)=[U]C(C3**(BCC(CN4C5=IC(NC(C*6)=O)=C6C=C5)OC4=O)*3)=C2[Mn])=C1I#C 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IB2011054968 | 2011-11-08 | ||
| IBPCT/IB2011/054968 | 2011-11-08 | ||
| PCT/IB2012/056236 WO2013068948A1 (en) | 2011-11-08 | 2012-11-07 | 2-oxo-oxazolidin-3,5-diyl antibiotic derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014532754A JP2014532754A (ja) | 2014-12-08 |
| JP2014532754A5 true JP2014532754A5 (enExample) | 2015-12-03 |
| JP6030146B2 JP6030146B2 (ja) | 2016-11-24 |
Family
ID=47258051
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014540612A Expired - Fee Related JP6030146B2 (ja) | 2011-11-08 | 2012-11-07 | ２−オキソ−オキサゾリジン−３，５−ジイル抗生物質誘導体 |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US9079922B2 (enExample) |
| EP (1) | EP2776431B1 (enExample) |
| JP (1) | JP6030146B2 (enExample) |
| KR (1) | KR20140096337A (enExample) |
| AR (1) | AR088691A1 (enExample) |
| AU (1) | AU2012335207B2 (enExample) |
| BR (1) | BR112014011064A8 (enExample) |
| CA (1) | CA2854264A1 (enExample) |
| CL (1) | CL2014001154A1 (enExample) |
| ES (1) | ES2581056T3 (enExample) |
| HK (1) | HK1202288A1 (enExample) |
| IL (1) | IL232463A0 (enExample) |
| IN (1) | IN2014CN04126A (enExample) |
| MX (1) | MX344529B (enExample) |
| PH (1) | PH12014500831A1 (enExample) |
| PL (1) | PL2776431T3 (enExample) |
| RU (1) | RU2616609C2 (enExample) |
| SG (1) | SG11201401710PA (enExample) |
| TW (1) | TWI594996B (enExample) |
| WO (1) | WO2013068948A1 (enExample) |
| ZA (1) | ZA201404176B (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY158520A (en) | 2008-10-07 | 2016-10-14 | Actelion Pharmaceuticals Ltd | Tricyclic oxazolidinone antibiotic compounds |
| SG11201508479RA (en) | 2013-04-16 | 2015-11-27 | Actelion Pharmaceuticals Ltd | Antibacterial biaromatic derivatives |
| AR096135A1 (es) | 2013-05-02 | 2015-12-09 | Actelion Pharmaceuticals Ltd | Derivados de la quinolona |
| AR102256A1 (es) | 2014-10-15 | 2017-02-15 | Actelion Pharmaceuticals Ltd | Derivados biaromáticos básicos antibacterianos con sustitución de aminoalcoxi |
| MA41168A (fr) | 2014-12-17 | 2017-10-24 | Acraf | Nouveaux composés antibactériens |
| MA41169A (fr) | 2014-12-17 | 2017-10-24 | Acraf | Composés antibactériens à large spectre d'activité |
| SG11201806166WA (en) * | 2016-02-08 | 2018-08-30 | Redx Pharma Plc | Heterocyclic compounds, in particular 2-oxo-4,4,5,5,6,6,7,7-octahydrobenzoxazole derivatives, and their use as antibacterial compounds |
| WO2017137743A1 (en) * | 2016-02-08 | 2017-08-17 | Redx Pharma Plc | Antibacterial compounds |
| GB201602235D0 (en) * | 2016-02-08 | 2016-03-23 | Redx Pharma Plc | Antibacterial compounds |
| AU2017276627A1 (en) | 2016-06-08 | 2018-12-20 | Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A. | New antibacterial compounds |
| TW201833120A (zh) | 2017-02-17 | 2018-09-16 | 瑞士商愛杜西亞製藥有限公司 | 芳基噁唑啶酮抗生素化合物 |
| FI3634968T3 (fi) * | 2017-06-08 | 2023-04-26 | Bugworks Res Inc | Bakteerilääkkeinä käyttökelpoisia heterosyklisiä yhdisteitä ja menetelmä niiden valmistamiseksi |
| ES2952989T3 (es) * | 2017-11-29 | 2023-11-07 | Bugworks Res Inc | Compuestos heterocíclicos antibacterianos y su síntesis |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3149104A (en) | 1961-01-03 | 1964-09-15 | Sterling Drug Inc | 4-hydroxy-7-styryl-1, 8-naphthyridine-3-carboxylic acids and esters |
| DE2362553A1 (de) | 1972-12-18 | 1974-06-20 | Dainippon Pharmaceutical Co | Neue piperazinderivate |
| SE444566B (sv) | 1977-09-20 | 1986-04-21 | Bellon Labor Sa Roger | 7-dialkylamin-6-halogen-4-oxo-1,4-dihydrokinolin-3-karboxylsyra, forfarande for framstellning derav och farmaceutiskt preparat derav |
| GB1598915A (en) | 1977-09-20 | 1981-09-23 | Bellon Labor Sa Roger | 1,4-dihydro-quinoline-3-carboxylic acid derivatives process for their preparation and composition containing them |
| CS274601B2 (en) | 1983-07-27 | 1991-09-15 | Dainippon Pharmaceutical Co | Method of 1,8-naphthyridine derivative production |
| JPS62205060A (ja) | 1986-03-04 | 1987-09-09 | Kyorin Pharmaceut Co Ltd | ８位置換キノロンカルボン酸誘導体 |
| EP0241206A3 (en) | 1986-03-31 | 1989-05-10 | Sankyo Company Limited | Quinoline-3-carboxylic acid derivatives, their preparation and use |
| JP2631854B2 (ja) | 1987-12-23 | 1997-07-16 | 藤本製薬株式会社 | 新規な１，８−ナフチリジン誘導体 |
| DE4301246A1 (de) | 1993-01-19 | 1994-07-21 | Bayer Ag | Chinolon- und Naphthyridoncarbonsäurederivate |
| JPWO2004002973A1 (ja) | 2002-06-28 | 2005-10-27 | 株式会社カネカ | 光学活性１−置換アミノ−２，３−エポキシプロパンの製造方法並びにその合成中間体およびそれらの製造方法 |
| BRPI0409955A (pt) * | 2003-04-30 | 2006-04-25 | Morphochem Ag Komb Chemie | uso de antibióticos hìbridos de oxazolidinona - quinolina para o tratamento de antrax e outras infecções |
| MXPA06006769A (es) * | 2003-12-18 | 2006-12-19 | Morphochem Ag Komb Chemie | Antibioticos hibridos de oxazolidinona-quinolona. |
| WO2006024741A2 (fr) * | 2004-07-30 | 2006-03-09 | Palumed S.A. | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
| US8613657B2 (en) | 2004-09-01 | 2013-12-24 | Christian Richard | System and method for permitting identification and counting of gaming chips |
| US20090156577A1 (en) | 2004-09-09 | 2009-06-18 | Benjamin Davis | 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones |
| EP2007377A4 (en) | 2006-04-06 | 2011-08-17 | Glaxo Group Ltd | ANTIBACTERIAL ACTIVE SUBSTANCES |
| MX2009004764A (es) * | 2006-11-10 | 2009-05-21 | Actelion Pharmaceuticals Ltd | Derivados de 5-hidroximetil-oxazolidin-2-ona. |
| CL2008001003A1 (es) * | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| CL2008001002A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| MX2010006111A (es) * | 2007-12-18 | 2010-06-25 | Actelion Pharmaceuticals Ltd | Derivados de 5-aminociclilmetil-oxazolidin-2-ona y su uso como antibacteriales. |
| ES2398939T3 (es) * | 2008-02-22 | 2013-03-22 | Actelion Pharmaceuticals Ltd. | Derivados de oxazolidinona |
| MY158520A (en) | 2008-10-07 | 2016-10-14 | Actelion Pharmaceuticals Ltd | Tricyclic oxazolidinone antibiotic compounds |
| BRPI0920870A2 (pt) * | 2008-10-10 | 2018-06-26 | Actelion Pharmaceuticals Ltd | antibióticos de oxazolidinila. |
| CA2738775A1 (en) * | 2008-10-10 | 2010-04-15 | Actelion Pharmaceuticals Ltd | 2-benzothiophenyl-and 2-naphthyl-0xaz0lidin0nes and their azaisostere analogues as antibacterial agents |
| TW201121965A (en) | 2009-09-28 | 2011-07-01 | Lg Life Sciences Ltd | Use of a quinolone derivative containing 7-(4-aminomethyl-3-oxime)pyrrolidine group that is capable of inducing granulocyte colony stimulating factor for treatment of neutropenia and recovery of hematopoiesis |
| CN101792443A (zh) | 2010-03-09 | 2010-08-04 | 北京欧凯纳斯科技有限公司 | 氟代喹诺酮衍生物及其制备方法和用途 |
-
2012
- 2012-11-07 PL PL12791863.9T patent/PL2776431T3/pl unknown
- 2012-11-07 SG SG11201401710PA patent/SG11201401710PA/en unknown
- 2012-11-07 MX MX2014005637A patent/MX344529B/es active IP Right Grant
- 2012-11-07 PH PH1/2014/500831A patent/PH12014500831A1/en unknown
- 2012-11-07 AU AU2012335207A patent/AU2012335207B2/en not_active Ceased
- 2012-11-07 IN IN4126CHN2014 patent/IN2014CN04126A/en unknown
- 2012-11-07 HK HK15102622.5A patent/HK1202288A1/xx unknown
- 2012-11-07 CA CA2854264A patent/CA2854264A1/en not_active Abandoned
- 2012-11-07 KR KR1020147014957A patent/KR20140096337A/ko not_active Abandoned
- 2012-11-07 ES ES12791863.9T patent/ES2581056T3/es active Active
- 2012-11-07 TW TW101141423A patent/TWI594996B/zh not_active IP Right Cessation
- 2012-11-07 JP JP2014540612A patent/JP6030146B2/ja not_active Expired - Fee Related
- 2012-11-07 US US14/356,896 patent/US9079922B2/en not_active Expired - Fee Related
- 2012-11-07 AR ARP120104192A patent/AR088691A1/es unknown
- 2012-11-07 BR BR112014011064A patent/BR112014011064A8/pt not_active Application Discontinuation
- 2012-11-07 EP EP12791863.9A patent/EP2776431B1/en not_active Not-in-force
- 2012-11-07 WO PCT/IB2012/056236 patent/WO2013068948A1/en not_active Ceased
- 2012-11-07 RU RU2014123109A patent/RU2616609C2/ru not_active IP Right Cessation
-
2014
- 2014-04-30 CL CL2014001154A patent/CL2014001154A1/es unknown
- 2014-05-05 IL IL232463A patent/IL232463A0/en unknown
- 2014-06-06 ZA ZA2014/04176A patent/ZA201404176B/en unknown
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