JP2014520863A - Ｂｒｕｔｏｎ型チロシンキナーゼの阻害剤 - Google Patents
Ｂｒｕｔｏｎ型チロシンキナーゼの阻害剤 Download PDFInfo
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
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Landscapes
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US201161507482P | 2011-07-13 | 2011-07-13 | |
| US61/507,482 | 2011-07-13 | ||
| PCT/US2012/046779 WO2013010136A2 (en) | 2011-07-13 | 2012-07-13 | Inhibitors of bruton's tyrosine kinase |
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| JP2014520863A true JP2014520863A (ja) | 2014-08-25 |
| JP2014520863A5 JP2014520863A5 (https=) | 2015-09-03 |
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| Country | Link |
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| US (2) | US9138436B2 (https=) |
| EP (1) | EP2731612A4 (https=) |
| JP (1) | JP2014520863A (https=) |
| KR (1) | KR20140048968A (https=) |
| CN (1) | CN103857396A (https=) |
| AU (1) | AU2012283775A1 (https=) |
| BR (1) | BR112014000653A2 (https=) |
| CA (1) | CA2841080A1 (https=) |
| EA (1) | EA201490265A1 (https=) |
| MX (1) | MX2014000518A (https=) |
| PH (1) | PH12014500122A1 (https=) |
| WO (1) | WO2013010136A2 (https=) |
| ZA (1) | ZA201400012B (https=) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016121953A1 (ja) * | 2015-01-30 | 2016-08-04 | 大鵬薬品工業株式会社 | 免疫疾患の予防及び／又は治療剤 |
| JP2018527384A (ja) * | 2015-09-16 | 2018-09-20 | ロクソ オンコロジー， インコーポレイテッドＬｏｘｏ Ｏｎｃｏｌｏｇｙ， Ｉｎｃ． | がんの治療のためのｂｔｋ阻害剤としてのピラゾロピリミジン誘導体 |
| JP2019507793A (ja) * | 2016-03-11 | 2019-03-22 | コーバス・ファーマシューティカルズ・インコーポレイテッド | ブルトン型チロシンキナーゼを調節する化合物及び方法 |
| JP2019535820A (ja) * | 2016-11-15 | 2019-12-12 | ハンヂョウ ハーツ ファーマシューティカル カンパニー リミテッド | 選択性ブルトン型チロシンキナーゼ阻害剤及びその使用 |
| JP2022523480A (ja) * | 2019-01-18 | 2022-04-25 | ミンフイ ファーマシューティカル （シャンハイ） リミテッド | ブルトン型チロシンキナーゼ阻害剤としての環状分子 |
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- 2012-07-13 PH PH1/2014/500122A patent/PH12014500122A1/en unknown
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- 2012-07-13 WO PCT/US2012/046779 patent/WO2013010136A2/en not_active Ceased
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- 2012-07-13 CA CA2841080A patent/CA2841080A1/en not_active Abandoned
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- 2012-07-13 US US13/549,267 patent/US9138436B2/en active Active
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| JP7849580B2 (ja) | 2020-10-05 | 2026-04-22 | デイナ ファーバー キャンサー インスティチュート，インコーポレイテッド | Ｈｅｒ２の強力かつ選択的な阻害剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2731612A2 (en) | 2014-05-21 |
| ZA201400012B (en) | 2016-01-27 |
| EP2731612A4 (en) | 2015-04-08 |
| AU2012283775A8 (en) | 2014-02-20 |
| EA201490265A1 (ru) | 2014-12-30 |
| CA2841080A1 (en) | 2013-01-17 |
| US20150329550A1 (en) | 2015-11-19 |
| MX2014000518A (es) | 2014-05-30 |
| AU2012283775A1 (en) | 2014-01-23 |
| CN103857396A (zh) | 2014-06-11 |
| US9862722B2 (en) | 2018-01-09 |
| BR112014000653A2 (pt) | 2017-02-14 |
| WO2013010136A3 (en) | 2013-07-04 |
| WO2013010136A2 (en) | 2013-01-17 |
| US20130018032A1 (en) | 2013-01-17 |
| PH12014500122A1 (en) | 2014-03-24 |
| US9138436B2 (en) | 2015-09-22 |
| KR20140048968A (ko) | 2014-04-24 |
| NZ619642A (en) | 2016-04-29 |
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