AU2012283775A1 - Inhibitors of Bruton's tyrosine kinase - Google Patents
Inhibitors of Bruton's tyrosine kinase Download PDFInfo
- Publication number
- AU2012283775A1 AU2012283775A1 AU2012283775A AU2012283775A AU2012283775A1 AU 2012283775 A1 AU2012283775 A1 AU 2012283775A1 AU 2012283775 A AU2012283775 A AU 2012283775A AU 2012283775 A AU2012283775 A AU 2012283775A AU 2012283775 A1 AU2012283775 A1 AU 2012283775A1
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- Prior art keywords
- substituted
- alkyl
- compound
- unsubstituted
- oph
- Prior art date
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- Abandoned
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Classifications
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
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-
2012
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- 2012-07-13 PH PH1/2014/500122A patent/PH12014500122A1/en unknown
- 2012-07-13 KR KR20147003521A patent/KR20140048968A/ko not_active Withdrawn
- 2012-07-13 EA EA201490265A patent/EA201490265A1/ru unknown
- 2012-07-13 WO PCT/US2012/046779 patent/WO2013010136A2/en not_active Ceased
- 2012-07-13 CN CN201280044640.1A patent/CN103857396A/zh active Pending
- 2012-07-13 CA CA2841080A patent/CA2841080A1/en not_active Abandoned
- 2012-07-13 EP EP20120811600 patent/EP2731612A4/en not_active Withdrawn
- 2012-07-13 US US13/549,267 patent/US9138436B2/en active Active
- 2012-07-13 BR BR112014000653A patent/BR112014000653A2/pt not_active IP Right Cessation
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| EP2731612A2 (en) | 2014-05-21 |
| ZA201400012B (en) | 2016-01-27 |
| EP2731612A4 (en) | 2015-04-08 |
| JP2014520863A (ja) | 2014-08-25 |
| AU2012283775A8 (en) | 2014-02-20 |
| EA201490265A1 (ru) | 2014-12-30 |
| CA2841080A1 (en) | 2013-01-17 |
| US20150329550A1 (en) | 2015-11-19 |
| MX2014000518A (es) | 2014-05-30 |
| CN103857396A (zh) | 2014-06-11 |
| US9862722B2 (en) | 2018-01-09 |
| BR112014000653A2 (pt) | 2017-02-14 |
| WO2013010136A3 (en) | 2013-07-04 |
| WO2013010136A2 (en) | 2013-01-17 |
| US20130018032A1 (en) | 2013-01-17 |
| PH12014500122A1 (en) | 2014-03-24 |
| US9138436B2 (en) | 2015-09-22 |
| KR20140048968A (ko) | 2014-04-24 |
| NZ619642A (en) | 2016-04-29 |
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