JP2014518199A5 - - Google Patents

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JP2014518199A5
JP2014518199A5 JP2014513214A JP2014513214A JP2014518199A5 JP 2014518199 A5 JP2014518199 A5 JP 2014518199A5 JP 2014513214 A JP2014513214 A JP 2014513214A JP 2014513214 A JP2014513214 A JP 2014513214A JP 2014518199 A5 JP2014518199 A5 JP 2014518199A5
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Japan
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formula
compound
group
alkyl
reacting
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JP2014513214A
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Japanese (ja)
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JP6425540B2 (ja
JP2014518199A (ja
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Priority claimed from PCT/EP2012/060447 external-priority patent/WO2012164096A1/en
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Publication of JP2014518199A5 publication Critical patent/JP2014518199A5/ja
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JP2014513214A 2011-06-01 2012-06-01 エステトロール中間体を製造するための方法 Active JP6425540B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161492300P 2011-06-01 2011-06-01
EP11168561 2011-06-01
EP11168561.6 2011-06-01
US61/492,300 2011-06-01
PCT/EP2012/060447 WO2012164096A1 (en) 2011-06-01 2012-06-01 Process for the production of estetrol intermediates

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017155801A Division JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Publications (3)

Publication Number Publication Date
JP2014518199A JP2014518199A (ja) 2014-07-28
JP2014518199A5 true JP2014518199A5 (enExample) 2016-02-12
JP6425540B2 JP6425540B2 (ja) 2018-11-21

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JP2014513214A Active JP6425540B2 (ja) 2011-06-01 2012-06-01 エステトロール中間体を製造するための方法
JP2017155801A Active JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Family Applications After (1)

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JP2017155801A Active JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Country Status (24)

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US (1) US11053274B2 (enExample)
EP (1) EP2714710B1 (enExample)
JP (2) JP6425540B2 (enExample)
KR (1) KR101994805B1 (enExample)
CN (2) CN103703014A (enExample)
AU (1) AU2012264602B2 (enExample)
BR (1) BR112013030830B1 (enExample)
CA (1) CA2835981C (enExample)
CY (1) CY1118150T1 (enExample)
DK (1) DK2714710T3 (enExample)
EA (1) EA023991B1 (enExample)
ES (1) ES2579175T3 (enExample)
HR (1) HRP20160692T2 (enExample)
HU (1) HUE029252T2 (enExample)
ME (1) ME02454B (enExample)
MX (1) MX341561B (enExample)
PL (1) PL2714710T3 (enExample)
PT (1) PT2714710T (enExample)
RS (1) RS54880B1 (enExample)
SG (1) SG195118A1 (enExample)
SI (1) SI2714710T1 (enExample)
SM (1) SMT201600206B (enExample)
WO (1) WO2012164096A1 (enExample)
ZA (1) ZA201308446B (enExample)

Families Citing this family (20)

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US11053274B2 (en) 2011-06-01 2021-07-06 Estetra S.P.R.L. Process for the production of estetrol intermediates
CA2835979C (en) 2011-06-01 2018-05-01 Estetra S.A. Process for the production of estetrol intermediates
EP2383279A1 (en) 2011-07-19 2011-11-02 Pantarhei Bioscience B.V. Process for the preparation of estetrol
EP2764008B1 (en) 2011-10-07 2016-08-17 Estetra S.P.R.L. Process for the production of estetrol
JP6813150B2 (ja) 2015-06-18 2021-01-13 エステトラ ソシエテ プリーヴ ア レスポンサビリテ リミテ エステトロールを含有する口腔内崩壊錠
CN116077454A (zh) 2015-06-18 2023-05-09 埃斯特拉有限责任公司 含雌四醇组分的口腔分散剂量单位
US11147771B2 (en) 2015-06-18 2021-10-19 Estetra Sprl Orodispersible dosage unit containing an estetrol component
ES2877186T3 (es) 2015-06-18 2021-11-16 Estetra Sprl Comprimido orodispersable que contiene estetrol
CN105837424A (zh) * 2016-03-31 2016-08-10 常州大学 一种1-氯-3-甲基-3-丁烯-2-酮的合成方法
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JOP20200260A1 (ar) 2018-04-19 2019-10-19 Estetra Sprl مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث
TWI801561B (zh) 2018-04-19 2023-05-11 比利時商依思特拉私人有限責任公司 化合物及其用於緩解絕經相關症狀的用途
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IT201900021879A1 (it) 2019-11-22 2021-05-22 Ind Chimica Srl PROCESSO PER LA PREPARAZIONE DI (15α,16α,17β)-ESTRA-1,3,5(10)-TRIENE-3,15,16,17-TETROLO (ESTETROLO) ED INTERMEDI DI DETTO PROCESSO
UY38895A (es) 2019-09-27 2021-04-30 Ind Chimica Srl PROCESO PARA PREPARAR (15a,16a,17ß)-ESTRA-1,3,5(10)-TRIENO-3,15,16,17-TETROL (ESTETROL) E INTERMEDIOS DE DICHO PROCESO
TWI893101B (zh) 2020-04-16 2025-08-11 比利時商埃斯特拉有限責任公司 具有降低之副作用之避孕組成物
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WO2024160373A1 (en) 2023-02-02 2024-08-08 Industriale Chimica S.R.L. PROCESS FOR PREPARING (15α,16α,17β)-ESTRA-1,3,5(10)-TRIENE-3,15,16,17-TETROL (ESTETROL) MONOHYDRATE

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US11147771B2 (en) 2015-06-18 2021-10-19 Estetra Sprl Orodispersible dosage unit containing an estetrol component
ES2877186T3 (es) 2015-06-18 2021-11-16 Estetra Sprl Comprimido orodispersable que contiene estetrol
CN116077454A (zh) 2015-06-18 2023-05-09 埃斯特拉有限责任公司 含雌四醇组分的口腔分散剂量单位

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