JP2014518199A5 - - Google Patents

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Publication number
JP2014518199A5
JP2014518199A5 JP2014513214A JP2014513214A JP2014518199A5 JP 2014518199 A5 JP2014518199 A5 JP 2014518199A5 JP 2014513214 A JP2014513214 A JP 2014513214A JP 2014513214 A JP2014513214 A JP 2014513214A JP 2014518199 A5 JP2014518199 A5 JP 2014518199A5
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Japan
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formula
compound
group
alkyl
reacting
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JP2014513214A
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Japanese (ja)
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JP6425540B2 (ja
JP2014518199A (ja
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Priority claimed from PCT/EP2012/060447 external-priority patent/WO2012164096A1/en
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Publication of JP2014518199A5 publication Critical patent/JP2014518199A5/ja
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JP2014513214A 2011-06-01 2012-06-01 エステトロール中間体を製造するための方法 Active JP6425540B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161492300P 2011-06-01 2011-06-01
US61/492,300 2011-06-01
EP11168561.6 2011-06-01
EP11168561 2011-06-01
PCT/EP2012/060447 WO2012164096A1 (en) 2011-06-01 2012-06-01 Process for the production of estetrol intermediates

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017155801A Division JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Publications (3)

Publication Number Publication Date
JP2014518199A JP2014518199A (ja) 2014-07-28
JP2014518199A5 true JP2014518199A5 (enExample) 2016-02-12
JP6425540B2 JP6425540B2 (ja) 2018-11-21

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JP2014513214A Active JP6425540B2 (ja) 2011-06-01 2012-06-01 エステトロール中間体を製造するための方法
JP2017155801A Active JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Family Applications After (1)

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JP2017155801A Active JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Country Status (24)

Country Link
US (1) US11053274B2 (enExample)
EP (1) EP2714710B1 (enExample)
JP (2) JP6425540B2 (enExample)
KR (1) KR101994805B1 (enExample)
CN (2) CN103703014A (enExample)
AU (1) AU2012264602B2 (enExample)
BR (1) BR112013030830B1 (enExample)
CA (1) CA2835981C (enExample)
CY (1) CY1118150T1 (enExample)
DK (1) DK2714710T3 (enExample)
EA (1) EA023991B1 (enExample)
ES (1) ES2579175T3 (enExample)
HR (1) HRP20160692T2 (enExample)
HU (1) HUE029252T2 (enExample)
ME (1) ME02454B (enExample)
MX (1) MX341561B (enExample)
PL (1) PL2714710T3 (enExample)
PT (1) PT2714710T (enExample)
RS (1) RS54880B1 (enExample)
SG (1) SG195118A1 (enExample)
SI (1) SI2714710T1 (enExample)
SM (1) SMT201600206B (enExample)
WO (1) WO2012164096A1 (enExample)
ZA (1) ZA201308446B (enExample)

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WO2012164096A1 (en) 2011-06-01 2012-12-06 Estetra S.A. Process for the production of estetrol intermediates
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EP2383279A1 (en) 2011-07-19 2011-11-02 Pantarhei Bioscience B.V. Process for the preparation of estetrol
EP2764008B1 (en) 2011-10-07 2016-08-17 Estetra S.P.R.L. Process for the production of estetrol
NZ737945A (en) 2015-06-18 2023-06-30 Estetra Sprl Orodispersible dosage unit containing an estetrol component
LT3310345T (lt) 2015-06-18 2021-06-25 Estetra Sprl Burnoje disperguojama tabletė, turinti estetrolio
WO2016203044A1 (en) 2015-06-18 2016-12-22 Mithra Pharmaceuticals S.A. Orodispersible tablet containing estetrol
RS57328B1 (sr) 2015-06-18 2018-08-31 Mithra Pharmaceuticals S A Orodisperzibilna dozna jedinica koja sadrži estetrolsku komponentu
CN105837424A (zh) * 2016-03-31 2016-08-10 常州大学 一种1-氯-3-甲基-3-丁烯-2-酮的合成方法
CA3178291A1 (en) 2016-08-05 2018-04-12 Estetra Srl Method for the management of dysmenorrhea and menstrual pain
JP6935766B2 (ja) 2018-02-15 2021-09-15 日本精工株式会社 スピンドル装置
CR20200486A (es) 2018-04-19 2021-01-27 Estetra Sprl Compuestos y sus usos para aliviar los síntomas asociados a la menopausa
TWI801561B (zh) 2018-04-19 2023-05-11 比利時商依思特拉私人有限責任公司 化合物及其用於緩解絕經相關症狀的用途
IT201900017414A1 (it) 2019-09-27 2021-03-27 Ind Chimica Srl Processo per la preparazione di (15α,16α,17β)-estra-1,3,5(10)-triene-3,15,16,17-tetrolo (Estetrolo) ed intermedi di detto processo
IT201900021879A1 (it) 2019-11-22 2021-05-22 Ind Chimica Srl PROCESSO PER LA PREPARAZIONE DI (15α,16α,17β)-ESTRA-1,3,5(10)-TRIENE-3,15,16,17-TETROLO (ESTETROLO) ED INTERMEDI DI DETTO PROCESSO
CN114514237B (zh) 2019-09-27 2024-07-26 工业化学有限公司 用于制备(15α,16α,17β)-雌-1,3,5(10)-三烯-3,15,16,17-四醇(雌四醇)的工艺及所述工艺的中间体
TWI893101B (zh) 2020-04-16 2025-08-11 比利時商埃斯特拉有限責任公司 具有降低之副作用之避孕組成物
WO2023021026A1 (en) 2021-08-17 2023-02-23 Aspen Oss B.V. A synthetic pathway to estra-1,3,5(10)-triene-3,15a,16a,17b-tetrol
GB2626482B (en) 2021-10-01 2025-04-30 Ind Chimica Srl Process for preparing (15alpha,16alpha,17beta)-estra-1,3,5-(10)-triene-3,15,16,17-tetrol(estetrol) monohydrate
CN120958008A (zh) 2023-02-02 2025-11-14 工业化学有限公司 制备(15α,16α,17β)-雌甾-1,3,5(10)-三烯-3,15,16,17-四醇(雌四醇)一水合物的方法
JP7711145B2 (ja) 2023-10-30 2025-07-22 ヤマハ発動機株式会社 報知システム、報知方法およびコンピュータプログラム

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