JP2014515040A5 - - Google Patents
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- JP2014515040A5 JP2014515040A5 JP2014510929A JP2014510929A JP2014515040A5 JP 2014515040 A5 JP2014515040 A5 JP 2014515040A5 JP 2014510929 A JP2014510929 A JP 2014510929A JP 2014510929 A JP2014510929 A JP 2014510929A JP 2014515040 A5 JP2014515040 A5 JP 2014515040A5
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- Prior art keywords
- alkyl
- aryl
- independently
- drug
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 C**C(N)=C(***NC)I Chemical compound C**C(N)=C(***NC)I 0.000 description 3
- PZILMLQXTGDJCM-UHFFFAOYSA-N C(C1)NCCN1c1nnc(N2CCNCC2)nn1 Chemical compound C(C1)NCCN1c1nnc(N2CCNCC2)nn1 PZILMLQXTGDJCM-UHFFFAOYSA-N 0.000 description 1
- XSWILQCWFQOKIE-UHFFFAOYSA-N C1CC(c2nnc(C3NCCCC3)nn2)NCC1 Chemical compound C1CC(c2nnc(C3NCCCC3)nn2)NCC1 XSWILQCWFQOKIE-UHFFFAOYSA-N 0.000 description 1
- ITWARJUHZJXKNM-UHFFFAOYSA-N CC(C1)C=C(C)C=C1NC(OC1C=CCCCCC1)=O Chemical compound CC(C1)C=C(C)C=C1NC(OC1C=CCCCCC1)=O ITWARJUHZJXKNM-UHFFFAOYSA-N 0.000 description 1
- XLZCIYOGIKMDSG-UHFFFAOYSA-N CC(C1C2CCCCCC1)=NN=C2c1ccccn1 Chemical compound CC(C1C2CCCCCC1)=NN=C2c1ccccn1 XLZCIYOGIKMDSG-UHFFFAOYSA-N 0.000 description 1
- NGMHTEDSSHAFGW-UHFFFAOYSA-N Cc1c[nH]c(-c2nnc(-c3nc(C)c[nH]3)nn2)n1 Chemical compound Cc1c[nH]c(-c2nnc(-c3nc(C)c[nH]3)nn2)n1 NGMHTEDSSHAFGW-UHFFFAOYSA-N 0.000 description 1
- ASUZTNLCAHONDF-UHFFFAOYSA-N Cc1nnc(-c2ccccn2)nn1 Chemical compound Cc1nnc(-c2ccccn2)nn1 ASUZTNLCAHONDF-UHFFFAOYSA-N 0.000 description 1
- PMMSDMUGUYODMC-UHFFFAOYSA-N NCc1nnc(CN)nn1 Chemical compound NCc1nnc(CN)nn1 PMMSDMUGUYODMC-UHFFFAOYSA-N 0.000 description 1
- FOJXFFILELMRKJ-UHFFFAOYSA-N c1cnc(-c2nnc(-c3ncc[nH]3)nn2)[nH]1 Chemical compound c1cnc(-c2nnc(-c3ncc[nH]3)nn2)[nH]1 FOJXFFILELMRKJ-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (17)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11166241 | 2011-05-16 | ||
| EP11166241.7 | 2011-05-16 | ||
| EP11166942.0 | 2011-05-20 | ||
| EP11166942 | 2011-05-20 | ||
| US201161515432P | 2011-08-05 | 2011-08-05 | |
| US201161515458P | 2011-08-05 | 2011-08-05 | |
| US61/515,458 | 2011-08-05 | ||
| US61/515,432 | 2011-08-05 | ||
| EP11176741 | 2011-08-05 | ||
| EP11176736 | 2011-08-05 | ||
| EP11176736.4 | 2011-08-05 | ||
| EP11176741.4 | 2011-08-05 | ||
| EP11192572.3 | 2011-12-08 | ||
| EP11192577.2 | 2011-12-08 | ||
| EP11192572 | 2011-12-08 | ||
| EP11192577 | 2011-12-08 | ||
| PCT/IB2012/052446 WO2012156919A1 (en) | 2011-05-16 | 2012-05-16 | Bio-orthogonal drug activation |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016161617A Division JP2017014262A (ja) | 2011-05-16 | 2016-08-22 | 生体直交型薬物活性化 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014515040A JP2014515040A (ja) | 2014-06-26 |
| JP2014515040A5 true JP2014515040A5 (enExample) | 2016-03-03 |
| JP5993940B2 JP5993940B2 (ja) | 2016-09-21 |
Family
ID=47176369
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014510928A Active JP6215194B2 (ja) | 2011-05-16 | 2012-05-16 | 生体直交型薬物活性化 |
| JP2014510930A Active JP6482273B2 (ja) | 2011-05-16 | 2012-05-16 | 生体直交型薬物活性化 |
| JP2014510929A Active JP5993940B2 (ja) | 2011-05-16 | 2012-05-16 | 生体直交型薬物活性化 |
| JP2016161617A Ceased JP2017014262A (ja) | 2011-05-16 | 2016-08-22 | 生体直交型薬物活性化 |
| JP2018000737A Active JP6608467B2 (ja) | 2011-05-16 | 2018-01-05 | 生体直交型薬物活性化 |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014510928A Active JP6215194B2 (ja) | 2011-05-16 | 2012-05-16 | 生体直交型薬物活性化 |
| JP2014510930A Active JP6482273B2 (ja) | 2011-05-16 | 2012-05-16 | 生体直交型薬物活性化 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016161617A Ceased JP2017014262A (ja) | 2011-05-16 | 2016-08-22 | 生体直交型薬物活性化 |
| JP2018000737A Active JP6608467B2 (ja) | 2011-05-16 | 2018-01-05 | 生体直交型薬物活性化 |
Country Status (9)
| Country | Link |
|---|---|
| US (8) | US9421274B2 (enExample) |
| EP (4) | EP2709668A1 (enExample) |
| JP (5) | JP6215194B2 (enExample) |
| CN (4) | CN103732256A (enExample) |
| AU (3) | AU2012257416B8 (enExample) |
| CA (3) | CA2836338C (enExample) |
| DK (1) | DK2709667T3 (enExample) |
| ES (1) | ES2920373T3 (enExample) |
| WO (3) | WO2012156919A1 (enExample) |
Families Citing this family (90)
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| JP6215194B2 (ja) * | 2011-05-16 | 2017-10-18 | コーニンクレッカ フィリップス エヌ ヴェＫｏｎｉｎｋｌｉｊｋｅ Ｐｈｉｌｉｐｓ Ｎ．Ｖ． | 生体直交型薬物活性化 |
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