JP2013520466A5 - - Google Patents

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Publication number
JP2013520466A5
JP2013520466A5 JP2012554332A JP2012554332A JP2013520466A5 JP 2013520466 A5 JP2013520466 A5 JP 2013520466A5 JP 2012554332 A JP2012554332 A JP 2012554332A JP 2012554332 A JP2012554332 A JP 2012554332A JP 2013520466 A5 JP2013520466 A5 JP 2013520466A5
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JP
Japan
Prior art keywords
alkyl
alkylene
pyrrolidin
pyridin
oxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012554332A
Other languages
English (en)
Japanese (ja)
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JP2013520466A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2011/052662 external-priority patent/WO2011104266A1/en
Publication of JP2013520466A publication Critical patent/JP2013520466A/ja
Publication of JP2013520466A5 publication Critical patent/JP2013520466A5/ja
Pending legal-status Critical Current

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JP2012554332A 2010-02-25 2011-02-23 二量体ｉａｐ阻害剤 Pending JP2013520466A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US30811410P 2010-02-25 2010-02-25
US61/308,114 2010-02-25
US33392710P 2010-05-12 2010-05-12
US61/333,927 2010-05-12
US38841010P 2010-09-30 2010-09-30
US61/388,410 2010-09-30
PCT/EP2011/052662 WO2011104266A1 (en) 2010-02-25 2011-02-23 Dimeric iap inhibitors

Publications (2)

Publication Number Publication Date
JP2013520466A JP2013520466A (ja) 2013-06-06
JP2013520466A5 true JP2013520466A5 (https=) 2014-03-20

Family

ID=44476672

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012554332A Pending JP2013520466A (ja) 2010-02-25 2011-02-23 二量体ｉａｐ阻害剤

Country Status (13)

Country Link
US (1) US8445440B2 (https=)
EP (1) EP2539333A1 (https=)
JP (1) JP2013520466A (https=)
KR (1) KR20130010894A (https=)
CN (1) CN102834389A (https=)
AR (1) AR080253A1 (https=)
BR (1) BR112012021291A2 (https=)
CA (1) CA2790302A1 (https=)
EA (1) EA201201177A1 (https=)
MX (1) MX2012009894A (https=)
TW (1) TW201141846A (https=)
UY (1) UY33236A (https=)
WO (1) WO2011104266A1 (https=)

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US9453048B2 (en) 2012-08-09 2016-09-27 Bristol-Myers Squibb Company IAP antagonists
CA2930030A1 (en) * 2012-11-09 2014-05-15 Ensemble Therapeutics Corporation Macrocyclic compounds for inhibition of inhibitors of apoptosis
KR20160030099A (ko) 2013-06-25 2016-03-16 더 월터 앤드 엘리자 홀 인스티튜트 오브 메디컬 리서치 세포내 감염의 치료 방법
WO2016079527A1 (en) 2014-11-19 2016-05-26 Tetralogic Birinapant Uk Ltd Combination therapy
WO2016097773A1 (en) 2014-12-19 2016-06-23 Children's Cancer Institute Therapeutic iap antagonists for treating proliferative disorders
CN109705191B (zh) * 2017-10-25 2022-04-29 广东东阳光药业有限公司 Iap抑制剂及其在药物中的应用

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