JP2013519683A5 - - Google Patents

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Publication number
JP2013519683A5
JP2013519683A5 JP2012553046A JP2012553046A JP2013519683A5 JP 2013519683 A5 JP2013519683 A5 JP 2013519683A5 JP 2012553046 A JP2012553046 A JP 2012553046A JP 2012553046 A JP2012553046 A JP 2012553046A JP 2013519683 A5 JP2013519683 A5 JP 2013519683A5
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Japan
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pharmaceutical composition
treatment
pharmaceutically acceptable
composition according
compound according
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JP2012553046A
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English (en)
Japanese (ja)
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JP5928828B2 (ja
JP2013519683A (ja
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Priority claimed from PCT/US2011/024583 external-priority patent/WO2011100585A1/en
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Publication of JP2013519683A5 publication Critical patent/JP2013519683A5/ja
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JP2012553046A 2010-02-11 2011-02-11 Ｎｍｄａ受容体モジュレータを安定化させる二次構造及びその使用 Active JP5928828B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30347210P 2010-02-11 2010-02-11
US61/303,472 2010-02-11
PCT/US2011/024583 WO2011100585A1 (en) 2010-02-11 2011-02-11 Secondary structure stabilized nmda receptor modulators and uses thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016080043A Division JP6328169B2 (ja) 2010-02-11 2016-04-13 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物

Publications (3)

Publication Number Publication Date
JP2013519683A JP2013519683A (ja) 2013-05-30
JP2013519683A5 true JP2013519683A5 (enExample) 2014-03-27
JP5928828B2 JP5928828B2 (ja) 2016-06-01

Family

ID=44368160

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2012553046A Active JP5928828B2 (ja) 2010-02-11 2011-02-11 Ｎｍｄａ受容体モジュレータを安定化させる二次構造及びその使用
JP2016080043A Expired - Fee Related JP6328169B2 (ja) 2010-02-11 2016-04-13 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物
JP2018079295A Withdrawn JP2018119004A (ja) 2010-02-11 2018-04-17 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物
JP2020046041A Pending JP2020117510A (ja) 2010-02-11 2020-03-17 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP2016080043A Expired - Fee Related JP6328169B2 (ja) 2010-02-11 2016-04-13 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物
JP2018079295A Withdrawn JP2018119004A (ja) 2010-02-11 2018-04-17 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物
JP2020046041A Pending JP2020117510A (ja) 2010-02-11 2020-03-17 Ｎｍｄａ受容体モジュレータを安定化させる化合物及びそれを含む医薬組成物

Country Status (13)

Country Link
US (2) US9101612B2 (enExample)
EP (1) EP2542254B1 (enExample)
JP (4) JP5928828B2 (enExample)
CN (2) CN102933226A (enExample)
AU (1) AU2011215704B2 (enExample)
BR (1) BR112012020142A2 (enExample)
CA (1) CA2789331C (enExample)
ES (1) ES2706063T3 (enExample)
IL (1) IL221400A (enExample)
MX (1) MX2012009388A (enExample)
RU (1) RU2566821C2 (enExample)
SG (3) SG10201811584RA (enExample)
WO (1) WO2011100585A1 (enExample)

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JP6823083B2 (ja) 2016-05-19 2021-01-27 アプティニックス インコーポレイテッド スピロラクタム系ｎｍｄａ受容体モジュレーターおよびその使用
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SG11201900558RA (en) 2016-08-01 2019-02-27 Aptinyx Inc Spiro-lactam nmda receptor modulators and uses thereof
CN109843889B (zh) 2016-08-01 2022-03-15 阿普廷伊克斯股份有限公司 螺-内酰胺nmda调节剂和使用其的方法
BR112019001768A2 (pt) 2016-08-01 2019-06-11 Aptinyx Inc moduladores do receptor de spiro-lactamas nmda e usos dos mesmos
PE20210455A1 (es) 2018-01-31 2021-03-08 Aptinyx Inc Moduladores del receptor nmda espiro-lactama y usos de los mismos
BR112020015666A2 (pt) * 2018-01-31 2021-02-23 Aptinyx Inc. moduladores de espiro-lactamas de receptores nmda e usos dos mesmos
CN110003309B (zh) * 2019-04-09 2021-09-10 北京广为医药科技有限公司 调节nmda受体活性的化合物、其药物组合物及用途
JP2022543772A (ja) * 2019-08-01 2022-10-14 アプティニックス インコーポレイテッド Ｎｍｄａ受容体と相互作用する抗体のレベル上昇に関連する障害を治療する方法
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