JP2013503823A5 - - Google Patents

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Publication number
JP2013503823A5
JP2013503823A5 JP2012527196A JP2012527196A JP2013503823A5 JP 2013503823 A5 JP2013503823 A5 JP 2013503823A5 JP 2012527196 A JP2012527196 A JP 2012527196A JP 2012527196 A JP2012527196 A JP 2012527196A JP 2013503823 A5 JP2013503823 A5 JP 2013503823A5
Authority
JP
Japan
Prior art keywords
duloxetine
crystalline duloxetine
crystalline
process according
range
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012527196A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013503823A (ja
Filing date
Publication date
Priority claimed from CZ2009-584A external-priority patent/CZ304602B6/cs
Application filed filed Critical
Publication of JP2013503823A publication Critical patent/JP2013503823A/ja
Publication of JP2013503823A5 publication Critical patent/JP2013503823A5/ja
Pending legal-status Critical Current

Links

JP2012527196A 2009-09-02 2010-09-02 (s)‐n‐メチル‐3‐(1‐ナフチルオキシ)‐3‐(2‐チエニル)プロピルアミン塩酸塩(デュロキセチン)の結晶化方法 Pending JP2013503823A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CZ2009-584A CZ304602B6 (cs) 2009-09-02 2009-09-02 Způsob krystalizace hydrochloridu (S)-N-methyl-3-(1-naftyloxy)-3-(2-thienyl)propylaminu (hydrochloridu duloxetinu)
CZPV-2009-584 2009-09-02
PCT/CZ2010/000099 WO2011026449A1 (en) 2009-09-02 2010-09-02 A method of crystallization of (s)-n-methyl-3-(1-naphthyloxy)-3- (2-thienyl)propylamine hydrochloride (duloxetine)

Publications (2)

Publication Number Publication Date
JP2013503823A JP2013503823A (ja) 2013-02-04
JP2013503823A5 true JP2013503823A5 (enExample) 2013-09-05

Family

ID=43413356

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012527196A Pending JP2013503823A (ja) 2009-09-02 2010-09-02 (s)‐n‐メチル‐3‐(1‐ナフチルオキシ)‐3‐(2‐チエニル)プロピルアミン塩酸塩(デュロキセチン)の結晶化方法

Country Status (11)

Country Link
EP (1) EP2473497A1 (enExample)
JP (1) JP2013503823A (enExample)
KR (1) KR20120047262A (enExample)
CN (1) CN102482254A (enExample)
BR (1) BR112012004862A2 (enExample)
CZ (1) CZ304602B6 (enExample)
EA (1) EA021528B1 (enExample)
IL (1) IL218329A0 (enExample)
MX (1) MX2012002621A (enExample)
WO (1) WO2011026449A1 (enExample)
ZA (1) ZA201201570B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103626735A (zh) * 2012-08-28 2014-03-12 石药集团中奇制药技术(石家庄)有限公司 一种盐酸度洛西汀晶型及其制备方法
CN104478849A (zh) * 2014-02-14 2015-04-01 广东东阳光药业有限公司 制备去甲肾上腺素再摄取双重抑制剂的方法
CN106265528A (zh) * 2015-05-12 2017-01-04 法德生技药品股份有限公司 制备药物凝集体的方法
JP2016222628A (ja) * 2015-06-03 2016-12-28 株式会社トクヤマ デュロキセチン塩酸塩の製造方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR880007433A (ko) 1986-12-22 1988-08-27 메리 앤 터커 3-아릴옥시-3-치환된 프로판아민
US5362886A (en) 1993-10-12 1994-11-08 Eli Lilly And Company Asymmetric synthesis
DE10212301A1 (de) 2002-03-20 2003-10-02 Bayer Ag Verfahren zur Herstellung von Aryl-aminopropanolen
PT1539673E (pt) 2002-07-09 2007-11-14 Lonza Ag Processo para preparação de beta-aminoálcoois nmonossubstituídos
GB0410470D0 (en) * 2004-05-11 2004-06-16 Cipla Ltd Pharmaceutical compound and polymorphs thereof
CZ297560B6 (cs) 2004-10-26 2007-02-07 Zentiva, A. S. Zpusob výroby hydrochloridu (S)-N-methyl-3-(1-naftyloxy)-3-(2-thienyl)propylaminu (duloxetinu)
TW200639161A (en) * 2005-03-14 2006-11-16 Teva Pharma Process for the purification of duloxetine hydrochloride
EP1820800A1 (en) * 2006-02-17 2007-08-22 KRKA, tovarna zdravil, d.d., Novo mesto Crystalline forms of duloxetine hydrochloride and processes for their preparation
GB0612508D0 (en) * 2006-06-23 2006-08-02 Arrow Int Ltd Crystalline duloxetine hydrochloride
GB0612509D0 (en) * 2006-06-23 2006-08-02 Arrow Int Ltd Crystalline duloxetine hydrochloride
CZ300116B6 (cs) * 2006-12-05 2009-02-11 Zentiva, A. S. Zpusob cištení hydrochloridu (S)-N-methyl-3-(1-naftyloxy)-3-(2-thienyl)propylaminu
WO2008107911A2 (en) * 2007-03-05 2008-09-12 Lupin Limited Novel process for preparation of duloxetine hydrochloride

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