JP2012527442A5 - - Google Patents

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Publication number
JP2012527442A5
JP2012527442A5 JP2012511355A JP2012511355A JP2012527442A5 JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5 JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5
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JP
Japan
Prior art keywords
salt
diffraction pattern
pharmaceutical composition
powder diffraction
ray powder
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JP2012511355A
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English (en)
Japanese (ja)
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JP5717727B2 (ja
JP2012527442A (ja
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Priority claimed from GBGB0908772.7A external-priority patent/GB0908772D0/en
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Publication of JP2012527442A5 publication Critical patent/JP2012527442A5/ja
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Publication of JP5717727B2 publication Critical patent/JP5717727B2/ja
Expired - Fee Related legal-status Critical Current
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JP2012511355A 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩 Expired - Fee Related JP5717727B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0908772.7A GB0908772D0 (en) 2009-05-21 2009-05-21 New salts 756
GB0908772.7 2009-05-21
PCT/GB2010/050822 WO2010133882A1 (en) 2009-05-21 2010-05-20 Disaccharin, difumaric acid, di-l-hydroxy-2-naphthoic acid and mono-benzoic acid salts of 4- (dimethylamin0)butyl 2- (4- ( (2-amino-4-methyl-6- (pentylamino) pyrimidin- 5 -yl) methyl) phenyl)acetate

Publications (3)

Publication Number Publication Date
JP2012527442A JP2012527442A (ja) 2012-11-08
JP2012527442A5 true JP2012527442A5 (enExample) 2013-07-04
JP5717727B2 JP5717727B2 (ja) 2015-05-13

Family

ID=40862774

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012511355A Expired - Fee Related JP5717727B2 (ja) 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩

Country Status (30)

Country Link
US (1) US8476288B2 (enExample)
EP (1) EP2435412B1 (enExample)
JP (1) JP5717727B2 (enExample)
KR (1) KR101709363B1 (enExample)
CN (1) CN102596917B (enExample)
AR (1) AR076597A1 (enExample)
AU (1) AU2010250920B2 (enExample)
BR (1) BRPI1012198A8 (enExample)
CA (1) CA2760765A1 (enExample)
CL (1) CL2011002941A1 (enExample)
CO (1) CO6440532A2 (enExample)
CR (1) CR20110611A (enExample)
CU (1) CU24053B1 (enExample)
DO (1) DOP2011000360A (enExample)
EA (1) EA021854B1 (enExample)
EC (1) ECSP11011469A (enExample)
ES (1) ES2566912T3 (enExample)
GB (1) GB0908772D0 (enExample)
HN (1) HN2011003072A (enExample)
IL (1) IL216280A0 (enExample)
MX (1) MX2011012344A (enExample)
NI (1) NI201100205A (enExample)
NZ (1) NZ596118A (enExample)
PE (1) PE20120989A1 (enExample)
SA (1) SA110310402B1 (enExample)
SG (1) SG175322A1 (enExample)
TW (1) TW201100389A (enExample)
UY (1) UY32649A (enExample)
WO (1) WO2010133882A1 (enExample)
ZA (1) ZA201109383B (enExample)

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TW201639852A (zh) 2008-12-09 2016-11-16 吉李德科學股份有限公司 用於製備可用作類鐸受體調節劑之化合物的中間體化合物
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ES2886973T3 (es) 2016-11-28 2021-12-21 Jiangsu Hengrui Medicine Co Derivado pirazolo-heteroarilo, método de preparación y uso médico del mismo
EP3636646A4 (en) 2017-05-18 2020-12-09 Jiangsu Hengrui Medicine Co., Ltd. HETEROARYL PYRAZOL DERIVATIVE AND MANUFACTURING METHOD FOR IT AND MEDICAL USES THEREOF
CN111819178B (zh) 2018-05-25 2022-04-12 江苏恒瑞医药股份有限公司 一种吡唑并杂芳基类衍生物盐酸盐的晶型及制备方法

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