JP2012527442A5 - - Google Patents

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Publication number
JP2012527442A5
JP2012527442A5 JP2012511355A JP2012511355A JP2012527442A5 JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5 JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5
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JP
Japan
Prior art keywords
salt
diffraction pattern
pharmaceutical composition
powder diffraction
ray powder
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JP2012511355A
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English (en)
Japanese (ja)
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JP5717727B2 (ja
JP2012527442A (ja
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Priority claimed from GBGB0908772.7A external-priority patent/GB0908772D0/en
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Publication of JP2012527442A publication Critical patent/JP2012527442A/ja
Publication of JP2012527442A5 publication Critical patent/JP2012527442A5/ja
Application granted granted Critical
Publication of JP5717727B2 publication Critical patent/JP5717727B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012511355A 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩 Expired - Fee Related JP5717727B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0908772.7 2009-05-21
GBGB0908772.7A GB0908772D0 (en) 2009-05-21 2009-05-21 New salts 756
PCT/GB2010/050822 WO2010133882A1 (en) 2009-05-21 2010-05-20 Disaccharin, difumaric acid, di-l-hydroxy-2-naphthoic acid and mono-benzoic acid salts of 4- (dimethylamin0)butyl 2- (4- ( (2-amino-4-methyl-6- (pentylamino) pyrimidin- 5 -yl) methyl) phenyl)acetate

Publications (3)

Publication Number Publication Date
JP2012527442A JP2012527442A (ja) 2012-11-08
JP2012527442A5 true JP2012527442A5 (enExample) 2013-07-04
JP5717727B2 JP5717727B2 (ja) 2015-05-13

Family

ID=40862774

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012511355A Expired - Fee Related JP5717727B2 (ja) 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩

Country Status (30)

Country Link
US (1) US8476288B2 (enExample)
EP (1) EP2435412B1 (enExample)
JP (1) JP5717727B2 (enExample)
KR (1) KR101709363B1 (enExample)
CN (1) CN102596917B (enExample)
AR (1) AR076597A1 (enExample)
AU (1) AU2010250920B2 (enExample)
BR (1) BRPI1012198A8 (enExample)
CA (1) CA2760765A1 (enExample)
CL (1) CL2011002941A1 (enExample)
CO (1) CO6440532A2 (enExample)
CR (1) CR20110611A (enExample)
CU (1) CU24053B1 (enExample)
DO (1) DOP2011000360A (enExample)
EA (1) EA021854B1 (enExample)
EC (1) ECSP11011469A (enExample)
ES (1) ES2566912T3 (enExample)
GB (1) GB0908772D0 (enExample)
HN (1) HN2011003072A (enExample)
IL (1) IL216280A0 (enExample)
MX (1) MX2011012344A (enExample)
NI (1) NI201100205A (enExample)
NZ (1) NZ596118A (enExample)
PE (1) PE20120989A1 (enExample)
SA (1) SA110310402B1 (enExample)
SG (1) SG175322A1 (enExample)
TW (1) TW201100389A (enExample)
UY (1) UY32649A (enExample)
WO (1) WO2010133882A1 (enExample)
ZA (1) ZA201109383B (enExample)

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SI3166607T1 (sl) 2014-07-11 2023-01-31 Gilead Sciences, Inc. Modulatorji toličnih receptorjev za zdravljenje HIV-a
CN110305133A (zh) 2014-09-16 2019-10-08 吉利德科学公司 Toll样受体调节剂的固体形式
KR20190084991A (ko) 2016-11-28 2019-07-17 지앙수 헨그루이 메디슨 컴퍼니 리미티드 피라졸로-헤테로아릴 유도체, 이의 제조 방법 및 의학적 용도
JP2020520379A (ja) 2017-05-18 2020-07-09 江▲蘇▼恒瑞医▲薬▼股▲フン▼有限公司Ｊｉａｎｇｓｕ Ｈｅｎｇｒｕｉ Ｍｅｄｉｃｉｎｅ Ｃｏ．， Ｌｔｄ． ヘテロアリール−ピラゾール誘導体ならびにその調製方法および医学的適用
MX2020012651A (es) 2018-05-25 2021-02-02 Jiangsu Hengrui Medicine Co Forma de cristal de clorhidrato de derivado de pirazoloheteroarilo, y metodo de preparacion.
CN113924114A (zh) 2019-05-22 2022-01-11 吉利德科学公司 Tlr7调节化合物和hiv疫苗的组合

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