JP2012527442A5 - - Google Patents

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Publication number
JP2012527442A5
JP2012527442A5 JP2012511355A JP2012511355A JP2012527442A5 JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5 JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5
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JP
Japan
Prior art keywords
salt
diffraction pattern
pharmaceutical composition
powder diffraction
ray powder
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JP2012511355A
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English (en)
Japanese (ja)
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JP2012527442A (ja
JP5717727B2 (ja
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Priority claimed from GBGB0908772.7A external-priority patent/GB0908772D0/en
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Publication of JP2012527442A publication Critical patent/JP2012527442A/ja
Publication of JP2012527442A5 publication Critical patent/JP2012527442A5/ja
Application granted granted Critical
Publication of JP5717727B2 publication Critical patent/JP5717727B2/ja
Expired - Fee Related legal-status Critical Current
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JP2012511355A 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩 Expired - Fee Related JP5717727B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0908772.7A GB0908772D0 (en) 2009-05-21 2009-05-21 New salts 756
GB0908772.7 2009-05-21
PCT/GB2010/050822 WO2010133882A1 (en) 2009-05-21 2010-05-20 Disaccharin, difumaric acid, di-l-hydroxy-2-naphthoic acid and mono-benzoic acid salts of 4- (dimethylamin0)butyl 2- (4- ( (2-amino-4-methyl-6- (pentylamino) pyrimidin- 5 -yl) methyl) phenyl)acetate

Publications (3)

Publication Number Publication Date
JP2012527442A JP2012527442A (ja) 2012-11-08
JP2012527442A5 true JP2012527442A5 (enExample) 2013-07-04
JP5717727B2 JP5717727B2 (ja) 2015-05-13

Family

ID=40862774

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012511355A Expired - Fee Related JP5717727B2 (ja) 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩

Country Status (30)

Country Link
US (1) US8476288B2 (enExample)
EP (1) EP2435412B1 (enExample)
JP (1) JP5717727B2 (enExample)
KR (1) KR101709363B1 (enExample)
CN (1) CN102596917B (enExample)
AR (1) AR076597A1 (enExample)
AU (1) AU2010250920B2 (enExample)
BR (1) BRPI1012198A8 (enExample)
CA (1) CA2760765A1 (enExample)
CL (1) CL2011002941A1 (enExample)
CO (1) CO6440532A2 (enExample)
CR (1) CR20110611A (enExample)
CU (1) CU24053B1 (enExample)
DO (1) DOP2011000360A (enExample)
EA (1) EA021854B1 (enExample)
EC (1) ECSP11011469A (enExample)
ES (1) ES2566912T3 (enExample)
GB (1) GB0908772D0 (enExample)
HN (1) HN2011003072A (enExample)
IL (1) IL216280A0 (enExample)
MX (1) MX2011012344A (enExample)
NI (1) NI201100205A (enExample)
NZ (1) NZ596118A (enExample)
PE (1) PE20120989A1 (enExample)
SA (1) SA110310402B1 (enExample)
SG (1) SG175322A1 (enExample)
TW (1) TW201100389A (enExample)
UY (1) UY32649A (enExample)
WO (1) WO2010133882A1 (enExample)
ZA (1) ZA201109383B (enExample)

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JP5978226B2 (ja) 2010-12-17 2016-08-24 大日本住友製薬株式会社 プリン誘導体
AU2013261267B2 (en) 2012-05-18 2017-06-29 Sumitomo Pharma Co., Ltd. Carboxylic acid compounds
EP4140485A1 (en) 2014-07-11 2023-03-01 Gilead Sciences, Inc. Modulators of toll-like receptors for the treatment of hiv
EA201790369A1 (ru) 2014-09-16 2017-10-31 Джилид Сайэнс, Инк. Твердые формы модулятора толл-подобного рецептора
ES2886973T3 (es) 2016-11-28 2021-12-21 Jiangsu Hengrui Medicine Co Derivado pirazolo-heteroarilo, método de preparación y uso médico del mismo
TW201900647A (zh) 2017-05-18 2019-01-01 大陸商江蘇恒瑞醫藥股份有限公司 雜芳基并吡唑類衍生物、其製備方法及其在醫藥上的應用
JP2021526520A (ja) 2018-05-25 2021-10-07 江▲蘇▼恒瑞医▲薬▼股▲フン▼有限公司Ｊｉａｎｇｓｕ Ｈｅｎｇｒｕｉ Ｍｅｄｉｃｉｎｅ Ｃｏ．， Ｌｔｄ． ピラゾロヘテロアリール誘導体の塩酸塩の結晶形および調製方法

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