JP2012513410A - 抗ウイルス化合物 - Google Patents

抗ウイルス化合物 Download PDF

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Publication number
JP2012513410A
JP2012513410A JP2011542571A JP2011542571A JP2012513410A JP 2012513410 A JP2012513410 A JP 2012513410A JP 2011542571 A JP2011542571 A JP 2011542571A JP 2011542571 A JP2011542571 A JP 2011542571A JP 2012513410 A JP2012513410 A JP 2012513410A
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JP
Japan
Prior art keywords
independently
carbocyclyl
optionally
substituted
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011542571A
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English (en)
Japanese (ja)
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JP2012513410A5 (https=
Inventor
デイゴーイ，デイビツド・エイ
ドナー，パメラ・エル
ケイテイ，ウオーレン・エム
ハツチンス，チヤールズ・ダブリユ
クリユーガー，アラン・シー
ランドルフ，ジヨン・テイー
モツター，クリストフアー・イー
クリシユナン，プリーシ
ミストリー，ニータ・シー
パイロツト−マテイアス，タミ・ジエイ
パテル，サツチン・ブイ
リー，シヤオヤン
ソルトウエデル，トツド・エヌ
ネルソン，リサ・テイー
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Abbott Laboratories
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Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of JP2012513410A publication Critical patent/JP2012513410A/ja
Publication of JP2012513410A5 publication Critical patent/JP2012513410A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
JP2011542571A 2008-12-23 2009-12-22 抗ウイルス化合物 Pending JP2012513410A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14031808P 2008-12-23 2008-12-23
US61/140,318 2008-12-23
PCT/US2009/069188 WO2010075380A1 (en) 2008-12-23 2009-12-22 Anti-viral compounds

Publications (2)

Publication Number Publication Date
JP2012513410A true JP2012513410A (ja) 2012-06-14
JP2012513410A5 JP2012513410A5 (https=) 2013-02-14

Family

ID=42167446

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011542571A Pending JP2012513410A (ja) 2008-12-23 2009-12-22 抗ウイルス化合物

Country Status (10)

Country Link
US (2) US8546405B2 (https=)
EP (1) EP2367823A1 (https=)
JP (1) JP2012513410A (https=)
CN (1) CN102245604A (https=)
CA (1) CA2740195A1 (https=)
MX (1) MX2011006333A (https=)
RU (1) RU2505539C2 (https=)
SG (1) SG172353A1 (https=)
WO (1) WO2010075380A1 (https=)
ZA (1) ZA201105356B (https=)

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