JP2012513410A - 抗ウイルス化合物 - Google Patents

抗ウイルス化合物 Download PDF

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Publication number
JP2012513410A
JP2012513410A JP2011542571A JP2011542571A JP2012513410A JP 2012513410 A JP2012513410 A JP 2012513410A JP 2011542571 A JP2011542571 A JP 2011542571A JP 2011542571 A JP2011542571 A JP 2011542571A JP 2012513410 A JP2012513410 A JP 2012513410A
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JP
Japan
Prior art keywords
independently
carbocyclyl
optionally
substituted
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011542571A
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English (en)
Japanese (ja)
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JP2012513410A5 (https=
Inventor
デイゴーイ，デイビツド・エイ
ドナー，パメラ・エル
ケイテイ，ウオーレン・エム
ハツチンス，チヤールズ・ダブリユ
クリユーガー，アラン・シー
ランドルフ，ジヨン・テイー
モツター，クリストフアー・イー
クリシユナン，プリーシ
ミストリー，ニータ・シー
パイロツト−マテイアス，タミ・ジエイ
パテル，サツチン・ブイ
リー，シヤオヤン
ソルトウエデル，トツド・エヌ
ネルソン，リサ・テイー
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Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of JP2012513410A publication Critical patent/JP2012513410A/ja
Publication of JP2012513410A5 publication Critical patent/JP2012513410A5/ja
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2011542571A 2008-12-23 2009-12-22 抗ウイルス化合物 Pending JP2012513410A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14031808P 2008-12-23 2008-12-23
US61/140,318 2008-12-23
PCT/US2009/069188 WO2010075380A1 (en) 2008-12-23 2009-12-22 Anti-viral compounds

Publications (2)

Publication Number Publication Date
JP2012513410A true JP2012513410A (ja) 2012-06-14
JP2012513410A5 JP2012513410A5 (https=) 2013-02-14

Family

ID=42167446

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011542571A Pending JP2012513410A (ja) 2008-12-23 2009-12-22 抗ウイルス化合物

Country Status (10)

Country Link
US (2) US8546405B2 (https=)
EP (1) EP2367823A1 (https=)
JP (1) JP2012513410A (https=)
CN (1) CN102245604A (https=)
CA (1) CA2740195A1 (https=)
MX (1) MX2011006333A (https=)
RU (1) RU2505539C2 (https=)
SG (1) SG172353A1 (https=)
WO (1) WO2010075380A1 (https=)
ZA (1) ZA201105356B (https=)

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