ATE301653T1 - Pyrazolopyridine - Google Patents

Pyrazolopyridine

Info

Publication number
ATE301653T1
ATE301653T1 AT01987095T AT01987095T ATE301653T1 AT E301653 T1 ATE301653 T1 AT E301653T1 AT 01987095 T AT01987095 T AT 01987095T AT 01987095 T AT01987095 T AT 01987095T AT E301653 T1 ATE301653 T1 AT E301653T1
Authority
AT
Austria
Prior art keywords
pyrazolopyridines
same
variables
preparing
processes
Prior art date
Application number
AT01987095T
Other languages
English (en)
Inventor
Stanley D Chamberlain
Kristjan Gudmundsson
Brian A Johns
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE301653T1 publication Critical patent/ATE301653T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
AT01987095T 2000-12-15 2001-11-26 Pyrazolopyridine ATE301653T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US25576300P 2000-12-15 2000-12-15
US27428401P 2001-03-08 2001-03-08
US31508901P 2001-08-27 2001-08-27
PCT/US2001/044210 WO2002048147A2 (en) 2000-12-15 2001-11-26 Pyrazolopyridines

Publications (1)

Publication Number Publication Date
ATE301653T1 true ATE301653T1 (de) 2005-08-15

Family

ID=27400896

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01987095T ATE301653T1 (de) 2000-12-15 2001-11-26 Pyrazolopyridine

Country Status (8)

Country Link
US (3) US6919352B2 (de)
EP (1) EP1341788B1 (de)
JP (1) JP2004518651A (de)
AT (1) ATE301653T1 (de)
AU (1) AU2002239344A1 (de)
DE (1) DE60112609T2 (de)
ES (1) ES2245380T3 (de)
WO (1) WO2002048147A2 (de)

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EP4141002A1 (de) 2015-11-19 2023-03-01 Incyte Corporation Heterocyclische verbindungen als immunmodulatoren
PL3394033T3 (pl) 2015-12-22 2021-05-31 Incyte Corporation Związki heterocykliczne jako immunomodulatory
TW201808950A (zh) 2016-05-06 2018-03-16 英塞特公司 作為免疫調節劑之雜環化合物
MA45116A (fr) 2016-05-26 2021-06-02 Incyte Corp Composés hétérocycliques comme immunomodulateurs
MX2018016273A (es) 2016-06-20 2019-07-04 Incyte Corp Compuestos heterociclicos como inmunomoduladores.
EP3484866B1 (de) 2016-07-14 2022-09-07 Incyte Corporation Heterocyclische verbindungen als immunmodulatoren
MA46045A (fr) 2016-08-29 2021-04-28 Incyte Corp Composés hétérocycliques utilisés comme immunomodulateurs
CN110582493B (zh) 2016-12-22 2024-03-08 因赛特公司 作为免疫调节剂的苯并噁唑衍生物
EP3558989B1 (de) 2016-12-22 2021-04-14 Incyte Corporation Triazolo[1,5-a]pyridin-derivate als immunmodulatoren
MD3558990T2 (ro) 2016-12-22 2023-02-28 Incyte Corp Derivați tetrahidro imidazo[4,5-c]piridină ca inductori de internalizare a PD-L1
ES2899402T3 (es) 2016-12-22 2022-03-11 Incyte Corp Derivados de piridina como inmunomoduladores
SG11202009440WA (en) 2018-03-30 2020-10-29 Incyte Corp Heterocyclic compounds as immunomodulators
DK3790877T3 (da) 2018-05-11 2023-04-24 Incyte Corp Tetrahydro-imidazo[4,5-c]pyridinderivater som pd-l1-immunmodulatorer
WO2021030162A1 (en) 2019-08-09 2021-02-18 Incyte Corporation Salts of a pd-1/pd-l1 inhibitor
US11401279B2 (en) 2019-09-30 2022-08-02 Incyte Corporation Pyrido[3,2-d]pyrimidine compounds as immunomodulators
TW202120504A (zh) 2019-11-11 2021-06-01 美商英塞特公司 Pd-1/pd-l1 抑制劑之鹽及結晶型
DE102020125641A1 (de) * 2020-09-25 2022-03-31 Creative Therapeutics Gmbh Wirkstoffe und Arzneimittel für die Therapie von Viruserkrankungen, insbesondere Corona-Infektionen, insbesondere COVID-19
AU2021373044A1 (en) 2020-11-06 2023-06-08 Incyte Corporation Process for making a pd-1/pd-l1 inhibitor and salts and crystalline forms thereof
WO2022099018A1 (en) 2020-11-06 2022-05-12 Incyte Corporation Process of preparing a pd-1/pd-l1 inhibitor
TW202233615A (zh) 2020-11-06 2022-09-01 美商英塞特公司 Ｐｄ—１／ｐｄ—ｌ１抑制劑之結晶形式

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Also Published As

Publication number Publication date
WO2002048147A3 (en) 2003-03-27
US7087618B2 (en) 2006-08-08
US20050182080A1 (en) 2005-08-18
US20050171133A1 (en) 2005-08-04
WO2002048147A2 (en) 2002-06-20
EP1341788B1 (de) 2005-08-10
US6919352B2 (en) 2005-07-19
AU2002239344A1 (en) 2002-06-24
DE60112609T2 (de) 2006-01-19
EP1341788A2 (de) 2003-09-10
DE60112609D1 (en) 2005-09-15
US7160897B2 (en) 2007-01-09
US20040072853A1 (en) 2004-04-15
ES2245380T3 (es) 2006-01-01
JP2004518651A (ja) 2004-06-24

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