JP2012505836A5 - - Google Patents
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- Publication number
- JP2012505836A5 JP2012505836A5 JP2011531305A JP2011531305A JP2012505836A5 JP 2012505836 A5 JP2012505836 A5 JP 2012505836A5 JP 2011531305 A JP2011531305 A JP 2011531305A JP 2011531305 A JP2011531305 A JP 2011531305A JP 2012505836 A5 JP2012505836 A5 JP 2012505836A5
- Authority
- JP
- Japan
- Prior art keywords
- amino
- benzofuran
- oxadiazol
- diol
- propane
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2008905369 | 2008-10-17 | ||
| AU2008905369A AU2008905369A0 (en) | 2008-10-17 | S1P Receptors Modulators and Their use Thereof | |
| AU2009903644 | 2009-08-05 | ||
| AU2009903644A AU2009903644A0 (en) | 2009-08-05 | S1P Receptors Modulators and their use Thereof | |
| PCT/AU2009/001371 WO2010043000A1 (en) | 2008-10-17 | 2009-10-19 | S1p receptors modulators and their use thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014192502A Division JP5963823B2 (ja) | 2008-10-17 | 2014-09-22 | S1p受容体モジュレーターおよびそれらの使用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2012505836A JP2012505836A (ja) | 2012-03-08 |
| JP2012505836A5 true JP2012505836A5 (OSRAM) | 2013-02-07 |
Family
ID=42106136
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011531305A Pending JP2012505836A (ja) | 2008-10-17 | 2009-10-19 | S1p受容体モジュレーターおよびそれらの使用 |
| JP2014192502A Active JP5963823B2 (ja) | 2008-10-17 | 2014-09-22 | S1p受容体モジュレーターおよびそれらの使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014192502A Active JP5963823B2 (ja) | 2008-10-17 | 2014-09-22 | S1p受容体モジュレーターおよびそれらの使用 |
Country Status (9)
| Country | Link |
|---|---|
| US (3) | US8592399B2 (OSRAM) |
| EP (1) | EP2344484B1 (OSRAM) |
| JP (2) | JP2012505836A (OSRAM) |
| CN (1) | CN102186845B (OSRAM) |
| AU (1) | AU2009304598B2 (OSRAM) |
| CA (1) | CA2740484C (OSRAM) |
| ES (1) | ES2590904T3 (OSRAM) |
| NZ (1) | NZ592748A (OSRAM) |
| WO (1) | WO2010043000A1 (OSRAM) |
Families Citing this family (39)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2344484B1 (en) * | 2008-10-17 | 2016-06-08 | Akaal Pharma Pty Ltd | S1p receptors modulators and use thereof |
| AU2009304596A1 (en) | 2008-10-17 | 2010-04-22 | Akaal Pharma Pty Ltd | S1P receptors modulators |
| KR20110117706A (ko) * | 2009-02-10 | 2011-10-27 | 아보트 러보러터리즈 | S1p5 수용체의 효능제 및 길항제, 및 이들의 사용 방법 |
| EA023283B1 (ru) * | 2010-11-30 | 2016-05-31 | Адэссо Эдванст Материалс Уси Ко., Лтд. | Новые вещества для повторно перерабатываемых эпоксидных смол |
| EP2697195A1 (en) * | 2011-04-14 | 2014-02-19 | Allergan, Inc. | Phenyl bicyclic methyl azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| CN102993027B (zh) * | 2011-09-08 | 2014-08-13 | 中化蓝天集团有限公司 | 4-氟-n-异丙基苯胺的定向单烷基化制备方法 |
| AU2012354695B2 (en) | 2011-12-23 | 2016-11-03 | Meiji Seika Pharma Co., Ltd. | Novel S1P receptor modulator |
| US9376409B2 (en) | 2012-05-09 | 2016-06-28 | Boehringer Ingelheim International Gmbh | Methods for making oxetan-3-ylmethanamines |
| NZ703851A (en) * | 2012-07-27 | 2017-01-27 | Biogen Ma Inc | Compounds that are s1p modulating agents and/or atx modulating agents |
| US8859598B2 (en) | 2012-10-04 | 2014-10-14 | Allergan, Inc. | 1, 2, 4-oxadiazoles azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| WO2014063199A1 (en) * | 2012-10-26 | 2014-05-01 | Akaal Pharma Pty Ltd | Organic compounds |
| CN104870446B (zh) | 2012-11-07 | 2019-08-13 | 内尔维阿诺医学科学有限公司 | 取代的嘧啶基和吡啶基吡咯并吡啶酮类、其制备方法及其作为激酶抑制剂的用途 |
| US8735433B1 (en) * | 2012-11-14 | 2014-05-27 | Allergan, Inc. | Aryl oxadiazole derivatives as sphingosine 1-phosphate (S1P) receptor modulators |
| CN103304503B (zh) * | 2013-06-02 | 2015-03-04 | 张远强 | 抗糖尿病化合物、其制备方法和用途 |
| CN103304499B (zh) * | 2013-06-02 | 2015-03-04 | 张远强 | 抗糖尿病化合物、其制备方法和用途 |
| WO2015023839A1 (en) * | 2013-08-15 | 2015-02-19 | Allergan, Inc. | Aryl azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| EP3112347B1 (en) | 2014-02-28 | 2018-10-31 | Kissei Pharmaceutical Co., Ltd. | Novel aniline derivative, pharmaceutical composition containing same, and use thereof |
| BR112017019453A2 (pt) | 2015-03-13 | 2018-05-15 | Forma Therapeutics Inc | compostos e composições de alfa-cinamida como inibidores de hdac8 |
| HK1254769A1 (zh) * | 2015-08-11 | 2019-07-26 | 阿卡制药有限公司 | 包含s1p受体调节剂的组合物 |
| AU2017218889A1 (en) | 2016-02-09 | 2018-08-30 | Pharmakea, Inc. | Quinolinone lysyl oxidase-like 2 inhibitors and uses thereof |
| US11472776B2 (en) | 2016-12-20 | 2022-10-18 | Oligomerix, Inc. | Quinazolinones that inhibit the formation of tau oligomers and their method of use |
| JP7273722B2 (ja) | 2016-12-20 | 2023-05-15 | オリゴメリックス インコーポレイテッド | タウオリゴマーの形成を阻害する新規ベンゾフラン、ベンゾチオフェン及びインドール類似体並びにそれらの使用方法 |
| EP3638235A4 (en) | 2017-06-14 | 2021-06-09 | Trevena, Inc. | COMPOUNDS FOR MODULATING S1P1 ACTIVITY AND METHODS OF USING IT |
| KR102017324B1 (ko) | 2018-04-30 | 2019-09-02 | 경북대학교 산학협력단 | 신규한 asm 활성 직접 억제 화합물 2-아미노-2-(1,2,3-트리아졸-4-일)프로판-1,3-디올 유도체 및 이의 용도 |
| US11801242B2 (en) | 2018-10-09 | 2023-10-31 | Duke University | Compositions and methods for adjuvant cancer therapeutics |
| WO2020114477A1 (zh) * | 2018-12-06 | 2020-06-11 | 上海济煜医药科技有限公司 | 作为免疫调节剂的化合物及其制备方法和应用 |
| CN109824685B (zh) * | 2019-04-03 | 2021-03-23 | 辽宁中医药大学 | 马齿苋中化合物oleracone G及其提取分离方法与应用 |
| KR20220079546A (ko) * | 2019-09-05 | 2022-06-13 | 트레베나, 인코포레이티드. | 간질 치료 방법 |
| JP2023502123A (ja) | 2019-11-19 | 2023-01-20 | トレベナ・インコーポレイテッド | S1p1モジュレーター化合物及び化合物を調製する方法 |
| US20230094545A1 (en) * | 2020-02-28 | 2023-03-30 | Akaal Pharma Pty Ltd | S1p receptor modulators |
| TW202300178A (zh) | 2021-03-18 | 2023-01-01 | 美商西根公司 | 內化的生物活性化合物偶聯物選擇性釋放藥物 |
| TW202430514A (zh) | 2022-09-30 | 2024-08-01 | 瑞士商先正達農作物保護股份公司 | 殺微生物之吡唑衍生物 |
| TW202430031A (zh) | 2022-09-30 | 2024-08-01 | 瑞士商先正達農作物保護股份公司 | 殺微生物之吡唑衍生物 |
| CN120282962A (zh) | 2022-11-30 | 2025-07-08 | 先正达农作物保护股份公司 | 杀微生物的四氢异喹啉衍生物 |
| WO2025114167A1 (en) | 2023-11-28 | 2025-06-05 | Syngenta Crop Protection Ag | Microbiocidal pyrazole derivatives |
| WO2025191053A1 (en) | 2024-03-14 | 2025-09-18 | Syngenta Crop Protection Ag | Microbiocidal pyrazole derivatives |
| WO2025210096A1 (en) | 2024-04-03 | 2025-10-09 | Syngenta Crop Protection Ag | Fungicidal compositions |
| WO2025210095A1 (en) | 2024-04-03 | 2025-10-09 | Syngenta Crop Protection Ag | Microbiocidal tetrahydroisoquinoline compounds |
| CN118878551A (zh) * | 2024-07-08 | 2024-11-01 | 安徽大学 | 一种4-溴噻吩并[2,3-c]吡啶-2-羧酸乙酯的制备方法 |
Family Cites Families (55)
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|---|---|---|---|---|
| US2550646A (en) | 1947-08-21 | 1951-04-24 | Commercial Solvents Corp | Polyamino alcohols and method for preparing them |
| JP2829451B2 (ja) * | 1990-11-30 | 1998-11-25 | 大塚製薬株式会社 | 活性酸素抑制剤 |
| CN1114834A (zh) * | 1993-09-28 | 1996-01-10 | 大塚制药株式会社 | 抗糖尿病剂 |
| FR2719044B1 (fr) * | 1994-04-26 | 1996-05-31 | Cird Galderma | Nouveaux composés bi-aromatiques acétylénés à groupement adamantyle, compositions pharmaceutiques et cosmétiques les contenant et utilisations. |
| US5883106A (en) * | 1994-10-18 | 1999-03-16 | Pfizer Inc. | 5-lipoxygenase inhibitors |
| JP3964478B2 (ja) | 1995-06-30 | 2007-08-22 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ヘテロ環含有カルボン酸誘導体及びそれを含有する医薬 |
| US6221865B1 (en) * | 1995-11-06 | 2001-04-24 | University Of Pittsburgh | Inhibitors of protein isoprenyl transferases |
| FR2741876B1 (fr) | 1995-12-01 | 1998-01-09 | Cird Galderma | Composes biaromatiques portant un groupement adamantyl en para, compositions pharmaceutiques et cosmetiques les contenant et utilisations |
| JPH10158192A (ja) | 1996-10-03 | 1998-06-16 | Eisai Co Ltd | 移植片対宿主疾患(gvhd)の治療および臓器移植時の移植片拒絶反応抑制のための医薬組成物 |
| US6228868B1 (en) * | 1998-07-27 | 2001-05-08 | Abbott Laboratories | Oxazoline antiproliferative agents |
| KR20010081117A (ko) * | 1998-12-18 | 2001-08-27 | 추후기재 | 신규한 바이사이클릭 화합물 |
| EP1250332A1 (en) * | 1999-12-17 | 2002-10-23 | Abbott Laboratories | Inhibitors of interleukin 5 gene expression |
| WO2002074758A2 (en) * | 2001-03-16 | 2002-09-26 | Abbott Laboratories | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
| US20040106794A1 (en) * | 2001-04-16 | 2004-06-03 | Schering Corporation | 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
| AR037714A1 (es) * | 2001-12-06 | 2004-12-01 | Maxia Pharmaceuticals Inc | Derivados de tiazolidinona y oxazolidinona 2-sustituidos para la inhibicion de fosfatasas y el tratamiento de cancer |
| AU2003302218A1 (en) * | 2002-05-16 | 2004-06-18 | Genelabs Technologies, Inc | Aryl and heteroaryl compounds as antibacterial and antifungal agents |
| CN1747949A (zh) | 2002-12-20 | 2006-03-15 | 法马西亚公司 | 无环吡唑化合物 |
| DK1602660T3 (da) * | 2003-02-18 | 2011-05-23 | Kyorin Seiyaku Kk | Aminophosphonsyrederivater, additionssalte deraf og S1P-receptormodulatorer |
| ES2379169T3 (es) * | 2003-05-19 | 2012-04-23 | Irm Llc | Composiciones y compuestos inmunosupresores |
| ES2527117T3 (es) | 2003-08-29 | 2015-01-20 | Ono Pharmaceutical Co., Ltd. | Compuesto capaz de unirse a receptor SIP y uso farmacéutico del mismo |
| CN1859904A (zh) | 2003-10-03 | 2006-11-08 | 默克公司 | 用于治疗阿尔茨海默氏病的苄醚和苄氨基β-分泌酶抑制剂 |
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| JP4874958B2 (ja) * | 2005-03-30 | 2012-02-15 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピリジン誘導体を含有する抗真菌剤 |
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| EP2014653A1 (en) * | 2007-06-15 | 2009-01-14 | Bioprojet | Novel dicarboxylic acid derivatives as S1P1 receptor agonists |
| US20090118349A1 (en) * | 2007-08-16 | 2009-05-07 | Onco-Pharmakon Incorporated | Bis-alkylating agents and their use in cancer therapy |
| AR072184A1 (es) * | 2008-06-20 | 2010-08-11 | Glaxo Group Ltd | Derivados de oxadiazol como agonistas del receptor s1p1 |
| AU2009304596A1 (en) | 2008-10-17 | 2010-04-22 | Akaal Pharma Pty Ltd | S1P receptors modulators |
| EP2344484B1 (en) * | 2008-10-17 | 2016-06-08 | Akaal Pharma Pty Ltd | S1p receptors modulators and use thereof |
| US20100160369A1 (en) | 2008-12-04 | 2010-06-24 | Exelixis, Inc. | S1P1 Agonists and Methods of Making And Using |
| CA2743397C (en) | 2008-12-18 | 2017-02-28 | Mathilde Muzerelle | Oxadiazole fused heterocyclic derivatives useful for the treatment of multiple sclerosis |
| WO2014063199A1 (en) * | 2012-10-26 | 2014-05-01 | Akaal Pharma Pty Ltd | Organic compounds |
-
2009
- 2009-10-19 EP EP09820119.7A patent/EP2344484B1/en active Active
- 2009-10-19 WO PCT/AU2009/001371 patent/WO2010043000A1/en not_active Ceased
- 2009-10-19 JP JP2011531305A patent/JP2012505836A/ja active Pending
- 2009-10-19 AU AU2009304598A patent/AU2009304598B2/en active Active
- 2009-10-19 CA CA2740484A patent/CA2740484C/en active Active
- 2009-10-19 US US13/124,549 patent/US8592399B2/en active Active
- 2009-10-19 NZ NZ592748A patent/NZ592748A/xx unknown
- 2009-10-19 ES ES09820119.7T patent/ES2590904T3/es active Active
- 2009-10-19 CN CN200980141188.9A patent/CN102186845B/zh active Active
-
2013
- 2013-10-29 US US14/066,276 patent/US9193716B2/en active Active
-
2014
- 2014-09-22 JP JP2014192502A patent/JP5963823B2/ja active Active
-
2015
- 2015-10-22 US US14/920,780 patent/US9707205B2/en active Active
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