JP2011529033A5 - - Google Patents
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- JP2011529033A5 JP2011529033A5 JP2011519189A JP2011519189A JP2011529033A5 JP 2011529033 A5 JP2011529033 A5 JP 2011529033A5 JP 2011519189 A JP2011519189 A JP 2011519189A JP 2011519189 A JP2011519189 A JP 2011519189A JP 2011529033 A5 JP2011529033 A5 JP 2011529033A5
- Authority
- JP
- Japan
- Prior art keywords
- cancer
- pyridin
- mol
- added
- prostate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13592008P | 2008-07-25 | 2008-07-25 | |
| US61/135,920 | 2008-07-25 | ||
| US22068509P | 2009-06-26 | 2009-06-26 | |
| US61/220,685 | 2009-06-26 | ||
| PCT/EP2009/059605 WO2010010191A1 (en) | 2008-07-25 | 2009-07-24 | Novel compounds useful for the treatment of degenerative and inflammatory diseases. |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011529033A JP2011529033A (ja) | 2011-12-01 |
| JP2011529033A5 true JP2011529033A5 (cg-RX-API-DMAC7.html) | 2012-09-06 |
| JP5480261B2 JP5480261B2 (ja) | 2014-04-23 |
Family
ID=41021059
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011519189A Active JP5480261B2 (ja) | 2008-07-25 | 2009-07-24 | 変性及び炎症性疾患の治療に有用な新規化合物 |
| JP2011519188A Active JP5559168B2 (ja) | 2008-07-25 | 2009-07-24 | 変性及び炎症性疾患の治療に有用な新規化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011519188A Active JP5559168B2 (ja) | 2008-07-25 | 2009-07-24 | 変性及び炎症性疾患の治療に有用な新規化合物 |
Country Status (35)
Families Citing this family (86)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0719803D0 (en) | 2007-10-10 | 2007-11-21 | Cancer Rec Tech Ltd | Therapeutic compounds and their use |
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| AU2010254806C1 (en) | 2009-06-05 | 2016-07-07 | Cephalon, Inc. | Preparation and uses of 1,2,4-triazolo [1,5a] pyridine derivatives |
| TWI462920B (zh) * | 2009-06-26 | 2014-12-01 | 葛萊伯格有限公司 | 用於治療退化性及發炎疾病之新穎化合物 |
| JO3030B1 (ar) * | 2009-06-26 | 2016-09-05 | Galapagos Nv | مركب جديد مفيد لمعالجة الامراض التنكسية والالتهابات |
| US20100331222A1 (en) * | 2009-06-26 | 2010-12-30 | Basf Se | Process for producing cellulose beads from solutions of cellulose in ionic liquid |
| US8877795B2 (en) | 2010-05-07 | 2014-11-04 | The Board Of Trustees Of The Leland Stanford Junior University | Identification of stabilizers of multimeric proteins |
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| MX367055B (es) | 2012-06-26 | 2019-08-02 | Del Mar Pharmaceuticals | El uso de una composición que comprende dianhidrogalactitol, diacetildianhidrogalactitol, y dibromodulcitol, y análogos o derivados de cada uno para el tratamiento de malignidades resistentes a inhibidores de tirosina cinasa. |
| US9169214B2 (en) * | 2012-12-21 | 2015-10-27 | The Board Of Trustees Of The Leland Stanford Junior University | Compounds and compositions that bind and stabilize transthyretin and their use for inhibiting transthyretin amyloidosis and protein-protein interactions |
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| BR112017021583A2 (pt) * | 2015-04-13 | 2018-07-03 | Galapagos Nv | métodos para o tratamento de transtornos inflamatórios |
| PL3290418T3 (pl) * | 2015-04-29 | 2019-11-29 | Wuxi Fortune Pharmaceutical Co Ltd | Inhibitory kinaz janusowych (jak) |
| AU2016257892A1 (en) * | 2015-05-05 | 2017-11-09 | Concert Pharmaceuticals, Inc. | Deuterated filgotinib |
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| WO2017012771A1 (en) | 2015-07-23 | 2017-01-26 | Ratiopharm Gmbh | Crystalline filgotinib sulfonic acid addition salts |
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| TWI712604B (zh) | 2016-03-01 | 2020-12-11 | 日商日本新藥股份有限公司 | 具jak抑制作用之化合物之結晶 |
| KR102492378B1 (ko) | 2016-07-26 | 2023-01-27 | 톈진 롱보진 파마시우티컬 씨오., 엘티디. | 선택적 jak 저해제로서 화합물, 및 이의 염 및 치료학적 용도 |
| JOP20190024A1 (ar) | 2016-08-26 | 2019-02-19 | Gilead Sciences Inc | مركبات بيروليزين بها استبدال واستخداماتها |
| CN107880038B (zh) * | 2016-09-30 | 2021-09-28 | 中国医药研究开发中心有限公司 | [1,2,4]三唑并[1,5-a]吡啶类化合物及其制备方法和医药用途 |
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| EA036903B1 (ru) * | 2016-10-26 | 2021-01-13 | Янссен Фармацевтика Нв | Соединения конденсированных бициклических пиридинов и их применение в качестве модуляторов ampa-рецептора |
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| EA039344B1 (ru) * | 2017-01-19 | 2022-01-17 | Сучжоу Лонгбайотек Фармасьютикалз Ко., Лтд. | Гетероциклическое соединение в качестве ингибитора jak и его соли и терапевтическое применение |
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| US12214216B1 (en) | 2019-10-16 | 2025-02-04 | Helen Feng | Photon enhanced bone growth system and method |
| CN111072655B (zh) * | 2019-12-30 | 2021-12-10 | 深圳市坤健创新药物研究院 | 一种三氮唑并吡啶类化合物及其制备方法和药用组合物与应用 |
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| WO2021226261A1 (en) | 2020-05-06 | 2021-11-11 | Ajax Therapeutics, Inc. | 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors |
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2009
- 2009-07-12 JO JOP/2009/0259A patent/JO3041B1/ar active
- 2009-07-22 AR ARP090102793A patent/AR072875A1/es active IP Right Grant
- 2009-07-23 TW TW098124908A patent/TWI447118B/zh not_active IP Right Cessation
- 2009-07-23 CL CL2009001637A patent/CL2009001637A1/es unknown
- 2009-07-24 BR BRPI0916862A patent/BRPI0916862B8/pt not_active IP Right Cessation
- 2009-07-24 BR BRPI0916659A patent/BRPI0916659B8/pt active IP Right Grant
- 2009-07-24 EP EP09781073A patent/EP2346864B1/en active Active
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