JP2011529033A5 - - Google Patents
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- JP2011529033A5 JP2011529033A5 JP2011519189A JP2011519189A JP2011529033A5 JP 2011529033 A5 JP2011529033 A5 JP 2011529033A5 JP 2011519189 A JP2011519189 A JP 2011519189A JP 2011519189 A JP2011519189 A JP 2011519189A JP 2011529033 A5 JP2011529033 A5 JP 2011529033A5
- Authority
- JP
- Japan
- Prior art keywords
- cancer
- pyridin
- mol
- added
- prostate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13592008P | 2008-07-25 | 2008-07-25 | |
| US61/135,920 | 2008-07-25 | ||
| US22068509P | 2009-06-26 | 2009-06-26 | |
| US61/220,685 | 2009-06-26 | ||
| PCT/EP2009/059605 WO2010010191A1 (en) | 2008-07-25 | 2009-07-24 | Novel compounds useful for the treatment of degenerative and inflammatory diseases. |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011529033A JP2011529033A (ja) | 2011-12-01 |
| JP2011529033A5 true JP2011529033A5 (OSRAM) | 2012-09-06 |
| JP5480261B2 JP5480261B2 (ja) | 2014-04-23 |
Family
ID=41021059
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011519189A Active JP5480261B2 (ja) | 2008-07-25 | 2009-07-24 | 変性及び炎症性疾患の治療に有用な新規化合物 |
| JP2011519188A Active JP5559168B2 (ja) | 2008-07-25 | 2009-07-24 | 変性及び炎症性疾患の治療に有用な新規化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011519188A Active JP5559168B2 (ja) | 2008-07-25 | 2009-07-24 | 変性及び炎症性疾患の治療に有用な新規化合物 |
Country Status (35)
| Country | Link |
|---|---|
| US (5) | US8242274B2 (OSRAM) |
| EP (2) | EP2361251B1 (OSRAM) |
| JP (2) | JP5480261B2 (OSRAM) |
| KR (2) | KR101711911B1 (OSRAM) |
| CN (2) | CN102105472B (OSRAM) |
| AR (1) | AR072875A1 (OSRAM) |
| AU (2) | AU2009273144B2 (OSRAM) |
| BR (2) | BRPI0916659B8 (OSRAM) |
| CA (2) | CA2730762C (OSRAM) |
| CL (1) | CL2009001637A1 (OSRAM) |
| CO (1) | CO6361925A2 (OSRAM) |
| CR (1) | CR20110092A (OSRAM) |
| CY (2) | CY1113945T1 (OSRAM) |
| DK (2) | DK2361251T3 (OSRAM) |
| DO (1) | DOP2011000022A (OSRAM) |
| EA (2) | EA018080B1 (OSRAM) |
| ES (2) | ES2406691T3 (OSRAM) |
| HR (2) | HRP20140681T1 (OSRAM) |
| IL (2) | IL210262A (OSRAM) |
| JO (1) | JO3041B1 (OSRAM) |
| MA (1) | MA32551B1 (OSRAM) |
| ME (1) | ME02046B (OSRAM) |
| MX (2) | MX2011000758A (OSRAM) |
| MY (1) | MY157615A (OSRAM) |
| NZ (1) | NZ590646A (OSRAM) |
| PE (1) | PE20100152A1 (OSRAM) |
| PL (2) | PL2346864T3 (OSRAM) |
| PT (2) | PT2346864E (OSRAM) |
| RS (2) | RS52823B (OSRAM) |
| SI (2) | SI2361251T1 (OSRAM) |
| SM (2) | SMT201300051B (OSRAM) |
| TW (1) | TWI447118B (OSRAM) |
| UY (1) | UY32006A (OSRAM) |
| WO (2) | WO2010010191A1 (OSRAM) |
| ZA (2) | ZA201100396B (OSRAM) |
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| CA2763900A1 (en) | 2009-06-05 | 2010-12-09 | Cephalon, Inc. | Preparation and uses of 1,2,4-triazolo [1,5a] pyridine derivatives |
| TWI462920B (zh) | 2009-06-26 | 2014-12-01 | 葛萊伯格有限公司 | 用於治療退化性及發炎疾病之新穎化合物 |
| US20100331222A1 (en) * | 2009-06-26 | 2010-12-30 | Basf Se | Process for producing cellulose beads from solutions of cellulose in ionic liquid |
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| EP2566333A4 (en) | 2010-05-07 | 2014-04-02 | Univ Leland Stanford Junior | IDENTIFICATION OF STABILIZERS OF MULTIMEDER PROTEINS |
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| AU2013280644B2 (en) | 2012-06-26 | 2018-08-02 | Jeffrey A. BACHA | Methods for treating tyrosine-kinase-inhibitor-resistant malignancies in patients with genetic polymorphisms or AHI1 dysregulations or mutations employing dianhydrogalactitol, diacetyldianhydrogalactitol, dibromodulcitol, or analogs or derivatives thereof |
| US9169214B2 (en) * | 2012-12-21 | 2015-10-27 | The Board Of Trustees Of The Leland Stanford Junior University | Compounds and compositions that bind and stabilize transthyretin and their use for inhibiting transthyretin amyloidosis and protein-protein interactions |
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| EP3179857B1 (en) | 2014-08-14 | 2021-09-08 | Mamoun M. Alhamadsheh | Conjugation of pharmaceutically active agents with transthyretin ligands through adjustable linkers to increase serum half-life |
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| CN107531695B (zh) * | 2015-04-29 | 2020-03-27 | 无锡福祈制药有限公司 | Jak抑制剂 |
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| ES2443307T3 (es) * | 2009-02-02 | 2014-02-18 | Basf Se | Absorbente que comprende aminas cíclicas para la eliminación de gases ácidos |
| CA2763900A1 (en) | 2009-06-05 | 2010-12-09 | Cephalon, Inc. | Preparation and uses of 1,2,4-triazolo [1,5a] pyridine derivatives |
| JO3030B1 (ar) | 2009-06-26 | 2016-09-05 | Galapagos Nv | مركب جديد مفيد لمعالجة الامراض التنكسية والالتهابات |
| TWI462920B (zh) | 2009-06-26 | 2014-12-01 | 葛萊伯格有限公司 | 用於治療退化性及發炎疾病之新穎化合物 |
| WO2013173506A2 (en) | 2012-05-16 | 2013-11-21 | Rigel Pharmaceuticals, Inc. | Method of treating muscular degradation |
| EP2863950B1 (en) | 2012-06-22 | 2018-07-18 | Galapagos NV | Aminotriazolopyridine for use in the treatment of inflammation, and pharmaceutical compositions thereof |
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