JP2011524376A5 - - Google Patents

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Publication number
JP2011524376A5
JP2011524376A5 JP2011513822A JP2011513822A JP2011524376A5 JP 2011524376 A5 JP2011524376 A5 JP 2011524376A5 JP 2011513822 A JP2011513822 A JP 2011513822A JP 2011513822 A JP2011513822 A JP 2011513822A JP 2011524376 A5 JP2011524376 A5 JP 2011524376A5
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JP
Japan
Prior art keywords
protected form
solid support
group
reduction reaction
reducing agent
Prior art date
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Pending
Application number
JP2011513822A
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English (en)
Japanese (ja)
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JP2011524376A (ja
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Priority claimed from PCT/AU2009/000786 external-priority patent/WO2009152577A1/en
Publication of JP2011524376A publication Critical patent/JP2011524376A/ja
Publication of JP2011524376A5 publication Critical patent/JP2011524376A5/ja
Pending legal-status Critical Current

Links

JP2011513822A 2008-06-20 2009-06-19 N−脱メチル化モルフィナン化合物を合成する方法 Pending JP2011524376A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AU2008903154A AU2008903154A0 (en) 2008-06-20 Process
AU2008903154 2008-06-20
PCT/AU2009/000786 WO2009152577A1 (en) 2008-06-20 2009-06-19 Process for the synthesis of n-demethylated morphinane compounds

Publications (2)

Publication Number Publication Date
JP2011524376A JP2011524376A (ja) 2011-09-01
JP2011524376A5 true JP2011524376A5 (https=) 2012-08-02

Family

ID=41433601

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011513822A Pending JP2011524376A (ja) 2008-06-20 2009-06-19 N−脱メチル化モルフィナン化合物を合成する方法

Country Status (9)

Country Link
US (1) US20110306766A1 (https=)
EP (1) EP2297160B1 (https=)
JP (1) JP2011524376A (https=)
CN (1) CN102089310A (https=)
AU (1) AU2009260121C1 (https=)
CA (1) CA2727944A1 (https=)
NZ (1) NZ589867A (https=)
WO (1) WO2009152577A1 (https=)
ZA (1) ZA201009078B (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8829020B2 (en) 2009-07-16 2014-09-09 Mallinckrodt Llc Compounds and compositions for use in phototherapy and in treatment of ocular neovascular disease and cancers
CN103275005B (zh) * 2013-06-17 2015-05-20 苏州立新制药有限公司 ent-3-甲氧基-17-甲基吗喃-10-酮的制备方法
WO2017184979A1 (en) * 2016-04-22 2017-10-26 Noramco, Inc. N-demethylation of morphinan alkaloids
US20230242547A1 (en) * 2020-06-10 2023-08-03 Research Center Pharmaceutical Engineering Gmbh Processes for preparing nor-opioid compounds and opioid antagonists by electrochemical n-demethylation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0732877B2 (ja) * 1990-07-10 1995-04-12 工業技術院長 固定化金属錯体
JPH05115787A (ja) * 1991-10-30 1993-05-14 Tosoh Corp アスコルビン酸の酸化触媒物質
AUPQ968300A0 (en) * 2000-08-25 2000-09-21 Glaxo Wellcome Australia Ltd Chemical methods
JP4674995B2 (ja) * 2001-05-31 2011-04-20 大阪瓦斯株式会社 担体−錯体複合体、アルカン酸化触媒およびアルカノール合成方法
US7087686B2 (en) * 2001-08-06 2006-08-08 Bp Chemicals Limited Chain growth reaction process
CA2539659C (en) * 2003-09-22 2013-03-26 Johnson Matthey Public Limited Company Process for the synthesis of morphinane compounds and intermediates thereof
CN1785976A (zh) * 2005-12-15 2006-06-14 南京大学 一类n-烃基青藤碱及其制备方法

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