JP2011522827A5 - - Google Patents

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Publication number
JP2011522827A5
JP2011522827A5 JP2011512645A JP2011512645A JP2011522827A5 JP 2011522827 A5 JP2011522827 A5 JP 2011522827A5 JP 2011512645 A JP2011512645 A JP 2011512645A JP 2011512645 A JP2011512645 A JP 2011512645A JP 2011522827 A5 JP2011522827 A5 JP 2011522827A5
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JP
Japan
Prior art keywords
medicament
mammals
mammals use
purity
pharmaceutical composition
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Application number
JP2011512645A
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English (en)
Japanese (ja)
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JP2011522827A (ja
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Priority claimed from PCT/US2009/046256 external-priority patent/WO2009149258A2/en
Publication of JP2011522827A publication Critical patent/JP2011522827A/ja
Publication of JP2011522827A5 publication Critical patent/JP2011522827A5/ja
Pending legal-status Critical Current

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JP2011512645A 2008-06-04 2009-06-04 ６−［（４ｓ）−２−メチル−４−（２−ナフチル）−１，２，３，４−テトラヒドロイソキノリン−７−イル］ピリダジン−３−アミンの結晶形 Pending JP2011522827A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5871708P 2008-06-04 2008-06-04
US61/058,717 2008-06-04
PCT/US2009/046256 WO2009149258A2 (en) 2008-06-04 2009-06-04 Crystalline form of 6-[(4s)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine

Publications (2)

Publication Number Publication Date
JP2011522827A JP2011522827A (ja) 2011-08-04
JP2011522827A5 true JP2011522827A5 (OSRAM) 2012-08-09

Family

ID=41277466

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011512646A Expired - Fee Related JP5567557B2 (ja) 2008-06-04 2009-06-04 テトラヒドロイソキノリンの製造方法
JP2011512645A Pending JP2011522827A (ja) 2008-06-04 2009-06-04 ６−［（４ｓ）−２−メチル−４−（２−ナフチル）−１，２，３，４−テトラヒドロイソキノリン−７−イル］ピリダジン−３−アミンの結晶形
JP2014100580A Pending JP2014169312A (ja) 2008-06-04 2014-05-14 テトラヒドロイソキノリンの製造方法

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2011512646A Expired - Fee Related JP5567557B2 (ja) 2008-06-04 2009-06-04 テトラヒドロイソキノリンの製造方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2014100580A Pending JP2014169312A (ja) 2008-06-04 2014-05-14 テトラヒドロイソキノリンの製造方法

Country Status (9)

Country Link
US (4) US8445494B2 (OSRAM)
EP (2) EP2280955B8 (OSRAM)
JP (3) JP5567557B2 (OSRAM)
KR (1) KR20110011653A (OSRAM)
CN (2) CN102112464A (OSRAM)
AR (1) AR071997A1 (OSRAM)
ES (1) ES2652462T3 (OSRAM)
TW (1) TW201002682A (OSRAM)
WO (2) WO2009149258A2 (OSRAM)

Families Citing this family (15)

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CN103880827B (zh) 2004-07-15 2017-01-04 阿尔巴尼分子研究公司 芳基和杂芳基取代的四氢异喹啉及其阻断去甲肾上腺素、多巴胺和血清素的重摄取的应用
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US9156812B2 (en) 2008-06-04 2015-10-13 Bristol-Myers Squibb Company Crystalline form of 6-[(4S)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine
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US8815894B2 (en) 2009-05-12 2014-08-26 Bristol-Myers Squibb Company Crystalline forms of (S)-7-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydroisoquinoline and use thereof
EP2429295B1 (en) 2009-05-12 2013-12-25 Albany Molecular Research, Inc. Aryl, heteroaryl, and heterocycle substituted tetrahydroisoquinolines and use thereof
KR101830447B1 (ko) * 2009-05-12 2018-02-20 알바니 몰레큘라 리써치, 인크. 7-(［1,2,4］트리아졸로［1,5-α］피리딘-6-일)-4-(3,4-디클로로페닐)-1,2,3,4-테트라하이드로이소퀴놀린 및 이의 용도
EP2606049A4 (en) 2010-08-17 2014-01-08 Albany Molecular Res Inc 2,5-METHANO- AND 2,5-ETHANO-TETRAHYDROBENZAZEPINE DERIVATIVES AND USES THEREOF FOR BLOCKING NOREPINEPHRINE, DOPAMINE, AND SEROTONIN REUPTAKE
NO2686520T3 (OSRAM) 2011-06-06 2018-03-17
EP3610890A1 (en) 2012-11-14 2020-02-19 The Johns Hopkins University Methods and compositions for treating schizophrenia
WO2014159501A2 (en) * 2013-03-14 2014-10-02 Bristol-Myers Squibb Company Processes for preparing tetrahydroisoquinolines
CN103601699A (zh) * 2013-11-04 2014-02-26 南京大学 一类1,3,4-噻二唑-2-酰胺衍生物及其制备方法
SG10202012791TA (en) 2013-11-15 2021-01-28 Akebia Therapeutics Inc Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino}acetic acid, compositions, and uses thereof
MX2020011845A (es) 2018-05-09 2021-01-15 Akebia Therapeutics Inc Proceso para preparar acido 2-[[5-(3-clorofenil)-3-hidroxipiridina -2-carbonil]amino]acetico.
US11524939B2 (en) 2019-11-13 2022-12-13 Akebia Therapeutics, Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino} acetic acid

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