JP2011510928A5 - - Google Patents
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- Publication number
- JP2011510928A5 JP2011510928A5 JP2010544413A JP2010544413A JP2011510928A5 JP 2011510928 A5 JP2011510928 A5 JP 2011510928A5 JP 2010544413 A JP2010544413 A JP 2010544413A JP 2010544413 A JP2010544413 A JP 2010544413A JP 2011510928 A5 JP2011510928 A5 JP 2011510928A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- independently
- haloalkyl
- alkoxy
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- -1 cyano, hydroxy Chemical group 0.000 claims 41
- 229910052736 halogen Inorganic materials 0.000 claims 23
- 150000002367 halogens Chemical class 0.000 claims 23
- 229910052799 carbon Inorganic materials 0.000 claims 19
- 125000001424 substituent group Chemical group 0.000 claims 15
- 125000000217 alkyl group Chemical group 0.000 claims 13
- 150000001721 carbon Chemical group 0.000 claims 13
- 125000004093 cyano group Chemical group *C#N 0.000 claims 13
- 125000003545 alkoxy group Chemical group 0.000 claims 12
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 12
- 125000004663 dialkyl amino group Chemical group 0.000 claims 11
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 claims 10
- 125000000753 cycloalkyl group Chemical group 0.000 claims 10
- 229910052739 hydrogen Inorganic materials 0.000 claims 10
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 10
- 125000005119 alkyl cycloalkyl group Chemical group 0.000 claims 9
- 125000005120 alkyl cycloalkyl alkyl group Chemical group 0.000 claims 8
- 150000001875 compounds Chemical class 0.000 claims 8
- 125000004665 trialkylsilyl group Chemical group 0.000 claims 8
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 7
- 125000003282 alkyl amino group Chemical group 0.000 claims 7
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims 7
- 125000004438 haloalkoxy group Chemical group 0.000 claims 7
- 125000001188 haloalkyl group Chemical group 0.000 claims 7
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 7
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 7
- 229910052760 oxygen Inorganic materials 0.000 claims 7
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 7
- 125000002813 thiocarbonyl group Chemical group *C(*)=S 0.000 claims 7
- 125000005347 halocycloalkyl group Chemical group 0.000 claims 6
- 125000001624 naphthyl group Chemical group 0.000 claims 6
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims 6
- 125000004183 alkoxy alkyl group Chemical group 0.000 claims 5
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 claims 5
- 125000004414 alkyl thio group Chemical group 0.000 claims 5
- 125000004122 cyclic group Chemical group 0.000 claims 5
- 125000000000 cycloalkoxy group Chemical group 0.000 claims 5
- 125000004858 cycloalkoxyalkyl group Chemical group 0.000 claims 5
- 125000004985 dialkyl amino alkyl group Chemical group 0.000 claims 5
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 4
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 4
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 4
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 4
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 4
- 125000005081 alkoxyalkoxyalkyl group Chemical group 0.000 claims 4
- 125000005078 alkoxycarbonylalkyl group Chemical group 0.000 claims 4
- 125000000278 alkyl amino alkyl group Chemical group 0.000 claims 4
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 claims 4
- 125000004687 alkyl sulfinyl alkyl group Chemical group 0.000 claims 4
- 125000004688 alkyl sulfonyl alkyl group Chemical group 0.000 claims 4
- 125000006350 alkyl thio alkyl group Chemical group 0.000 claims 4
- 125000005112 cycloalkylalkoxy group Chemical group 0.000 claims 4
- 125000004994 halo alkoxy alkyl group Chemical group 0.000 claims 4
- 125000000262 haloalkenyl group Chemical group 0.000 claims 4
- 125000005203 haloalkylcarbonyloxy group Chemical group 0.000 claims 4
- 125000004461 halocycloalkylalkyl group Chemical group 0.000 claims 4
- 229910052717 sulfur Inorganic materials 0.000 claims 4
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 3
- 125000003118 aryl group Chemical group 0.000 claims 3
- 125000002619 bicyclic group Chemical group 0.000 claims 3
- 125000004432 carbon atom Chemical group C* 0.000 claims 3
- 125000006254 cycloalkyl carbonyl group Chemical group 0.000 claims 3
- 125000006448 cycloalkyl cycloalkyl group Chemical group 0.000 claims 3
- 125000005167 cycloalkylaminocarbonyl group Chemical group 0.000 claims 3
- 125000005201 cycloalkylcarbonyloxy group Chemical group 0.000 claims 3
- 125000005366 cycloalkylthio group Chemical group 0.000 claims 3
- 125000000232 haloalkynyl group Chemical group 0.000 claims 3
- 125000006769 halocycloalkoxy group Chemical group 0.000 claims 3
- 125000005842 heteroatom Chemical group 0.000 claims 3
- 125000000623 heterocyclic group Chemical group 0.000 claims 3
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims 3
- 125000002757 morpholinyl group Chemical group 0.000 claims 3
- 125000003386 piperidinyl group Chemical group 0.000 claims 3
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 3
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims 2
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims 2
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims 2
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims 2
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 2
- 125000006771 (C1-C6) haloalkylthio group Chemical group 0.000 claims 2
- 125000006766 (C2-C6) alkynyloxy group Chemical group 0.000 claims 2
- 125000006765 (C2-C6) haloalkenyloxy group Chemical group 0.000 claims 2
- XTFIVUDBNACUBN-UHFFFAOYSA-N 1,3,5-trinitro-1,3,5-triazinane Chemical compound [O-][N+](=O)N1CN([N+]([O-])=O)CN([N+]([O-])=O)C1 XTFIVUDBNACUBN-UHFFFAOYSA-N 0.000 claims 2
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- 125000002853 C1-C4 hydroxyalkyl group Chemical group 0.000 claims 2
- 125000003320 C2-C6 alkenyloxy group Chemical group 0.000 claims 2
- 125000004648 C2-C8 alkenyl group Chemical group 0.000 claims 2
- 125000004649 C2-C8 alkynyl group Chemical group 0.000 claims 2
- 125000005083 alkoxyalkoxy group Chemical group 0.000 claims 2
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims 2
- 125000000304 alkynyl group Chemical group 0.000 claims 2
- 125000006615 aromatic heterocyclic group Chemical group 0.000 claims 2
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 2
- 125000000392 cycloalkenyl group Chemical group 0.000 claims 2
- 125000006310 cycloalkyl amino group Chemical group 0.000 claims 2
- 125000005144 cycloalkylsulfonyl group Chemical group 0.000 claims 2
- 125000005221 halo alkyl carbonyl amino group Chemical group 0.000 claims 2
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 claims 2
- 229910052757 nitrogen Inorganic materials 0.000 claims 2
- 125000000719 pyrrolidinyl group Chemical group 0.000 claims 2
- 229920006395 saturated elastomer Polymers 0.000 claims 2
- 125000006729 (C2-C5) alkenyl group Chemical group 0.000 claims 1
- 125000006825 (C2-C5) haloalkyl group Chemical group 0.000 claims 1
- 125000006767 (C2-C6) haloalkynyloxy group Chemical group 0.000 claims 1
- 125000004198 2-fluorophenyl group Chemical group [H]C1=C([H])C(F)=C(*)C([H])=C1[H] 0.000 claims 1
- 150000001204 N-oxides Chemical class 0.000 claims 1
- 241000233654 Oomycetes Species 0.000 claims 1
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical group C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 claims 1
- 125000003342 alkenyl group Chemical group 0.000 claims 1
- 125000004450 alkenylene group Chemical group 0.000 claims 1
- 125000003302 alkenyloxy group Chemical group 0.000 claims 1
- 125000004702 alkoxy alkyl carbonyl group Chemical group 0.000 claims 1
- 125000005082 alkoxyalkenyl group Chemical group 0.000 claims 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims 1
- 125000005085 alkoxycarbonylalkoxy group Chemical group 0.000 claims 1
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 claims 1
- 125000004949 alkyl amino carbonyl amino group Chemical group 0.000 claims 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 claims 1
- 125000005130 alkyl carbonyl thio group Chemical group 0.000 claims 1
- 125000004656 alkyl sulfonylamino group Chemical group 0.000 claims 1
- 125000005133 alkynyloxy group Chemical group 0.000 claims 1
- 125000004103 aminoalkyl group Chemical group 0.000 claims 1
- 230000000844 anti-bacterial effect Effects 0.000 claims 1
- 125000004429 atom Chemical group 0.000 claims 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims 1
- 125000004966 cyanoalkyl group Chemical group 0.000 claims 1
- 125000004465 cycloalkenyloxy group Chemical group 0.000 claims 1
- 125000005149 cycloalkylsulfinyl group Chemical group 0.000 claims 1
- 125000004983 dialkoxyalkyl group Chemical group 0.000 claims 1
- 125000004472 dialkylaminosulfonyl group Chemical group 0.000 claims 1
- 201000010099 disease Diseases 0.000 claims 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 244000000004 fungal plant pathogen Species 0.000 claims 1
- 125000005291 haloalkenyloxy group Chemical group 0.000 claims 1
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 claims 1
- 125000004443 haloalkoxycarbonylamino group Chemical group 0.000 claims 1
- 125000004992 haloalkylamino group Chemical group 0.000 claims 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 claims 1
- 125000004664 haloalkylsulfonylamino group Chemical group 0.000 claims 1
- 125000004995 haloalkylthio group Chemical group 0.000 claims 1
- 125000005292 haloalkynyloxy group Chemical group 0.000 claims 1
- 125000000842 isoxazolyl group Chemical group 0.000 claims 1
- AGYVSBQQNSDGIS-UHFFFAOYSA-N methyl n-(2,5-dimethylphenyl)-4-[4-[5-(2-oxo-1,3-benzoxazol-3-yl)-4,5-dihydro-1,2-oxazol-3-yl]-1,3-thiazol-2-yl]piperidine-1-carboximidate Chemical compound C1CC(C=2SC=C(N=2)C=2CC(ON=2)N2C(OC3=CC=CC=C32)=O)CCN1C(OC)=NC1=CC(C)=CC=C1C AGYVSBQQNSDGIS-UHFFFAOYSA-N 0.000 claims 1
- 125000004674 methylcarbonyl group Chemical group CC(=O)* 0.000 claims 1
- MHHBHSAYGWOQIM-UHFFFAOYSA-N n'-(2,5-dimethylphenyl)-4-[4-(5-phenyl-4,5-dihydro-1,2-oxazol-3-yl)-1,3-thiazol-2-yl]piperidine-1-carboximidamide Chemical compound CC1=CC=C(C)C(NC(=N)N2CCC(CC2)C=2SC=C(N=2)C=2CC(ON=2)C=2C=CC=CC=2)=C1 MHHBHSAYGWOQIM-UHFFFAOYSA-N 0.000 claims 1
- 125000006574 non-aromatic ring group Chemical group 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- XCJZAEBHRKDWQG-UHFFFAOYSA-N CC(C1)=NOC1c(c(OC)cc(OC)c1)c1OC Chemical compound CC(C1)=NOC1c(c(OC)cc(OC)c1)c1OC XCJZAEBHRKDWQG-UHFFFAOYSA-N 0.000 description 1
- 0 CC(C1)=NOC1c1c(C)cc(*)cc1C Chemical compound CC(C1)=NOC1c1c(C)cc(*)cc1C 0.000 description 1
- KPHATKPOJFGEAO-UHFFFAOYSA-N CC(C1)=NOC1c1ccccc1 Chemical compound CC(C1)=NOC1c1ccccc1 KPHATKPOJFGEAO-UHFFFAOYSA-N 0.000 description 1
- WCKLKDXFQHATPQ-UHFFFAOYSA-N CC(C1)=NOC1c1ccccc1C(OC)=O Chemical compound CC(C1)=NOC1c1ccccc1C(OC)=O WCKLKDXFQHATPQ-UHFFFAOYSA-N 0.000 description 1
- REDZCUVHHXAOGE-GFCCVEGCSA-N CC(C1)=NO[C@]1(c(cccc1)c1N1CI)C1=O Chemical compound CC(C1)=NO[C@]1(c(cccc1)c1N1CI)C1=O REDZCUVHHXAOGE-GFCCVEGCSA-N 0.000 description 1
- LBZIXNGCDVMNGZ-GFCCVEGCSA-N CC(C1)=NO[C@]1(c1c2cccc1)N(C)C2=O Chemical compound CC(C1)=NO[C@]1(c1c2cccc1)N(C)C2=O LBZIXNGCDVMNGZ-GFCCVEGCSA-N 0.000 description 1
- KBCUKLBCFHQJRI-NSHDSACASA-N CC(C1)=NO[C@]1(c1ccccc1)C#N Chemical compound CC(C1)=NO[C@]1(c1ccccc1)C#N KBCUKLBCFHQJRI-NSHDSACASA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6239508P | 2008-01-25 | 2008-01-25 | |
| US61/062,395 | 2008-01-25 | ||
| PCT/US2009/031686 WO2009094445A2 (en) | 2008-01-25 | 2009-01-22 | Fungicidal hetercyclic compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011510928A JP2011510928A (ja) | 2011-04-07 |
| JP2011510928A5 true JP2011510928A5 (https=) | 2012-02-23 |
| JP5529044B2 JP5529044B2 (ja) | 2014-06-25 |
Family
ID=40791139
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010544413A Expired - Fee Related JP5529044B2 (ja) | 2008-01-25 | 2009-01-22 | 殺菌性複素環化合物 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8349870B2 (https=) |
| EP (2) | EP2402332A3 (https=) |
| JP (1) | JP5529044B2 (https=) |
| KR (2) | KR20100119552A (https=) |
| CN (2) | CN103965187A (https=) |
| AU (1) | AU2009206468B2 (https=) |
| BR (1) | BRPI0905759A2 (https=) |
| MX (1) | MX2010008102A (https=) |
| WO (1) | WO2009094445A2 (https=) |
Families Citing this family (63)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9090604B2 (en) | 2006-07-27 | 2015-07-28 | E I Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| WO2008013622A2 (en) | 2006-07-27 | 2008-01-31 | E. I. Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| PE20110368A1 (es) * | 2008-08-18 | 2011-06-13 | Univ Yale | Moduladores de mif |
| US9643922B2 (en) | 2008-08-18 | 2017-05-09 | Yale University | MIF modulators |
| US9540322B2 (en) | 2008-08-18 | 2017-01-10 | Yale University | MIF modulators |
| AU2009322486A1 (en) | 2008-12-02 | 2010-06-10 | E. I. Du Pont De Nemours And Company | Fungicidal heterocyclic compounds |
| CN102292334A (zh) | 2008-12-11 | 2011-12-21 | 拜尔农作物科学股份公司 | 噻唑基肟醚和腙植物保护剂 |
| US20100267706A1 (en) * | 2009-04-20 | 2010-10-21 | Institute For Oneworld Health | Compounds, Compositions and Methods Comprising Pyridazine Derivatives |
| AR076687A1 (es) * | 2009-05-18 | 2011-06-29 | Infinity Pharmaceuticals Inc | Isoxazolinas como inhibidores de la amidahidrolasa de acidos grasos y com-posiciones farmaceuticas que los contienen |
| US9149465B2 (en) | 2009-05-18 | 2015-10-06 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| US8927551B2 (en) | 2009-05-18 | 2015-01-06 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| EP2464643A1 (en) * | 2009-08-12 | 2012-06-20 | Syngenta Participations AG | Microbiocidal heterocycles |
| KR20120101019A (ko) | 2009-10-30 | 2012-09-12 | 바이엘 크롭사이언스 아게 | 헤테로아릴피페리딘 및 -피페라진 유도체 |
| EP2509978A1 (en) * | 2009-12-11 | 2012-10-17 | E.I. Du Pont De Nemours And Company | Azocyclic inhibitors of fatty acid amide hydrolase |
| MX2012007200A (es) | 2009-12-21 | 2012-07-10 | Bayer Cropscience Ag | Bis(difluorometil)pirazoles como fungicidas. |
| BR112012016733A2 (pt) * | 2010-01-07 | 2015-09-01 | Du Pont | "composto, composição fungicida e método" |
| BR112012027762B1 (pt) | 2010-04-28 | 2018-06-05 | Bayer Intellectual Property Gmbh | Derivados de cetoheteroarilpiperidina e - piperazina como fungicidas |
| US8815775B2 (en) | 2010-05-18 | 2014-08-26 | Bayer Cropscience Ag | Bis(difluoromethyl)pyrazoles as fungicides |
| BR112012026708A2 (pt) | 2010-05-20 | 2015-09-22 | Du Pont | composto selecionado, composição fungicida e método para controlar doenças vegetais |
| EP2576539B1 (de) | 2010-05-27 | 2017-12-13 | Bayer CropScience AG | Pyridinylcarbonsäure derivate als fungizide |
| US20120122928A1 (en) | 2010-08-11 | 2012-05-17 | Bayer Cropscience Ag | Heteroarylpiperidine and -Piperazine Derivatives as Fungicides |
| AU2015261660B2 (en) * | 2010-08-25 | 2017-01-05 | Bayer Cropscience Aktiengesellschaft | Heteroarylpiperidine and -piperazine derivatives as fungicides |
| US8759527B2 (en) | 2010-08-25 | 2014-06-24 | Bayer Cropscience Ag | Heteroarylpiperidine and -piperazine derivatives as fungicides |
| EP2423210A1 (de) | 2010-08-25 | 2012-02-29 | Bayer CropScience AG | Heteroarylpiperidin- und -piperazinderivate als Fungizide |
| EP2632922B1 (de) * | 2010-10-27 | 2019-02-27 | Bayer CropScience Aktiengesellschaft | Heteroarylpiperidin und -piperazinderivate als fungizide |
| JP5695397B2 (ja) * | 2010-11-25 | 2015-04-01 | 日本エンバイロケミカルズ株式会社 | 防カビ剤、それを用いる防カビ方法、生育阻止剤およびそれを用いる生育阻止方法 |
| CN103384470A (zh) * | 2010-12-17 | 2013-11-06 | 纳幕尔杜邦公司 | 杀真菌偶氮环酰胺 |
| WO2012104273A1 (de) | 2011-02-01 | 2012-08-09 | Bayer Cropscience Ag | Heteroarylpiperidin und -piperazinderivate als fungizide |
| EP2532233A1 (en) | 2011-06-07 | 2012-12-12 | Bayer CropScience AG | Active compound combinations |
| US10004232B2 (en) | 2011-09-15 | 2018-06-26 | Bayer Intellectual Property Gmbh | Piperidine pyrazoles as fungicides |
| DK2797899T3 (en) | 2011-12-27 | 2016-04-04 | Bayer Ip Gmbh | Heteroarylpiperidin and -piperazinderivater as fungicides |
| US9266876B2 (en) | 2012-02-02 | 2016-02-23 | Actelion Pharmaceuticals Ltd. | 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives |
| MX360174B (es) * | 2012-02-27 | 2018-10-12 | Bayer Ip Gmbh | Combinaciones de compuestos activos que contienen una tiazolilisoxazolina y un fungicida. |
| EP2864326A1 (en) | 2012-06-22 | 2015-04-29 | E. I. Du Pont de Nemours and Company | Fungicidal heterocyclic compounds |
| MX355542B (es) | 2012-08-30 | 2018-04-20 | Bayer Cropscience Ag | Procedimiento de descarboxilacion de derivados de acido 3,5-bis(haloalquil)-pirazol-4-carboxilico. |
| EP2801575A1 (en) | 2013-05-07 | 2014-11-12 | Bayer CropScience AG | Heteroaryldihydropyridine derivatives as fungicides |
| WO2014206896A1 (en) | 2013-06-24 | 2014-12-31 | Bayer Cropscience Ag | Piperidinecarboxylic acid derivatives as fungicides |
| EA030067B1 (ru) | 2013-07-22 | 2018-06-29 | Идорсиа Фармасьютиклз Лтд | Производные 1-(пиперазин-1-ил)-2-([1,2,4]триазол-1-ил)этанона |
| US9924721B2 (en) | 2013-08-28 | 2018-03-27 | Bayer Cropscience Aktiengesellschaft | Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides |
| AR099789A1 (es) | 2014-03-24 | 2016-08-17 | Actelion Pharmaceuticals Ltd | Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina |
| PT3122746T (pt) | 2014-03-24 | 2018-07-27 | Bayer Cropscience Ag | Derivados de fenilpiperidinacarboxamida como fungicidas |
| WO2015181097A1 (en) * | 2014-05-28 | 2015-12-03 | Bayer Cropscience Ag | Process for preparing thiazole derivatives |
| TWI665192B (zh) * | 2014-05-28 | 2019-07-11 | 德商拜耳作物科學股份有限公司 | 製備二氫異唑衍生物之方法 |
| WO2016024350A1 (ja) | 2014-08-13 | 2016-02-18 | 株式会社エス・ディー・エス バイオテック | 縮合１１員環化合物及びそれらを含有する農園芸用殺菌剤 |
| BR112017002359B1 (pt) * | 2014-08-13 | 2023-03-28 | Nippon Soda Co., Ltd | Composto, agentes de controle de organismo nocivo e de parasita externo, inseticida ou acaricida, e, expelente ou agente de controle de parasita interno |
| JP6337218B2 (ja) | 2015-01-15 | 2018-06-06 | イドーシア ファーマシューティカルズ リミテッドＩｄｏｒｓｉａ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ | Ｃｘｃｒ３受容体調節剤としてのヒドロキシアルキル−ピペラジン誘導体 |
| AR103399A1 (es) | 2015-01-15 | 2017-05-10 | Actelion Pharmaceuticals Ltd | Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3 |
| WO2016202761A1 (en) | 2015-06-17 | 2016-12-22 | Bayer Cropscience Aktiengesellschaft | Active compound combinations |
| CN105541830B (zh) * | 2015-12-14 | 2018-04-27 | 北京迪尔乐农业高新技术研发中心 | 一种杀菌化合物、制备方法及其应用 |
| KR102605762B1 (ko) * | 2016-02-08 | 2023-11-27 | 고완 크롭 프로텍션 리미티드 | 살균성 조성물 |
| CN108602765B (zh) | 2016-02-08 | 2022-05-03 | 高文有限公司 | 1,2-苯二甲醇化合物的制造方法 |
| TW201838974A (zh) | 2017-04-19 | 2018-11-01 | 印度商Ｐｉ工業公司 | 具殺菌性質之雜環化合物 |
| CA3073637A1 (en) * | 2017-09-08 | 2019-03-14 | Pi Industries Ltd | Novel fungicidal heterocyclic compounds |
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| CN109516962A (zh) * | 2018-12-13 | 2019-03-26 | 天津雅奥泰克科技有限公司 | 一种合成2,6-二氟苯基-1-(4,5-二氢异恶唑)-3-乙基酮的新方法 |
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| EP4578854A4 (en) * | 2022-08-26 | 2025-12-03 | Jiangsu Flag Chem Ind Co Ltd | COMPOUND CONTAINING A CHAIN-FORMED CARBOXYLIC ACID AMIDE STRUCTURE, ITS PREPARATION PROCESS, ITS USE AND BACTERICIDAL ACTION |
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| WO2025098238A1 (zh) * | 2023-11-07 | 2025-05-15 | 江苏中旗科技股份有限公司 | 含哌嗪环结构的化合物及其制备方法和应用、一种杀菌剂 |
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2009
- 2009-01-22 US US12/863,875 patent/US8349870B2/en not_active Expired - Fee Related
- 2009-01-22 AU AU2009206468A patent/AU2009206468B2/en not_active Ceased
- 2009-01-22 KR KR1020107018519A patent/KR20100119552A/ko not_active Ceased
- 2009-01-22 JP JP2010544413A patent/JP5529044B2/ja not_active Expired - Fee Related
- 2009-01-22 MX MX2010008102A patent/MX2010008102A/es active IP Right Grant
- 2009-01-22 CN CN201410221847.2A patent/CN103965187A/zh active Pending
- 2009-01-22 BR BRPI0905759-5A patent/BRPI0905759A2/pt not_active Application Discontinuation
- 2009-01-22 KR KR1020157014513A patent/KR20150065958A/ko not_active Ceased
- 2009-01-22 EP EP11007851.6A patent/EP2402332A3/en not_active Withdrawn
- 2009-01-22 EP EP09704518A patent/EP2260032A2/en not_active Withdrawn
- 2009-01-22 CN CN200980105521.0A patent/CN101970432B/zh not_active Expired - Fee Related
- 2009-01-22 WO PCT/US2009/031686 patent/WO2009094445A2/en not_active Ceased
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