JP2011509294A5 - - Google Patents
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- Publication number
- JP2011509294A5 JP2011509294A5 JP2010542266A JP2010542266A JP2011509294A5 JP 2011509294 A5 JP2011509294 A5 JP 2011509294A5 JP 2010542266 A JP2010542266 A JP 2010542266A JP 2010542266 A JP2010542266 A JP 2010542266A JP 2011509294 A5 JP2011509294 A5 JP 2011509294A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- aryl
- heterocyclyl
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- HRJDRCMGALFOLA-GDLZYMKVSA-N N[C@H](CCc1ccccc1)C(NOCc1ccc(CNC(CN2CCN(CC(O)=O)CCN(CC(O)=O)CCN(CC(O)=O)CC2)=O)cc1)=O Chemical compound N[C@H](CCc1ccccc1)C(NOCc1ccc(CNC(CN2CCN(CC(O)=O)CCN(CC(O)=O)CCN(CC(O)=O)CC2)=O)cc1)=O HRJDRCMGALFOLA-GDLZYMKVSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1962708P | 2008-01-08 | 2008-01-08 | |
| US61/019,627 | 2008-01-08 | ||
| PCT/US2009/000096 WO2009089022A1 (en) | 2008-01-08 | 2009-01-08 | N-alkoxyamide conjugates as imaging agents |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015079425A Division JP6087386B2 (ja) | 2008-01-08 | 2015-04-08 | 造影剤としてのｎ−アルコキシアミド抱合体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011509294A JP2011509294A (ja) | 2011-03-24 |
| JP2011509294A5 true JP2011509294A5 (https=) | 2012-02-23 |
| JP5730581B2 JP5730581B2 (ja) | 2015-06-10 |
Family
ID=40456854
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010542266A Expired - Fee Related JP5730581B2 (ja) | 2008-01-08 | 2009-01-08 | 造影剤としてのｎ−アルコキシアミド抱合体 |
| JP2015079425A Expired - Fee Related JP6087386B2 (ja) | 2008-01-08 | 2015-04-08 | 造影剤としてのｎ−アルコキシアミド抱合体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015079425A Expired - Fee Related JP6087386B2 (ja) | 2008-01-08 | 2015-04-08 | 造影剤としてのｎ−アルコキシアミド抱合体 |
Country Status (14)
| Country | Link |
|---|---|
| US (4) | US8361438B2 (https=) |
| EP (1) | EP2240206B1 (https=) |
| JP (2) | JP5730581B2 (https=) |
| KR (2) | KR101595324B1 (https=) |
| CN (2) | CN101970015B (https=) |
| AU (2) | AU2009204427B2 (https=) |
| BR (1) | BRPI0907612A2 (https=) |
| CA (1) | CA2711426C (https=) |
| ES (1) | ES2629340T3 (https=) |
| IL (1) | IL206846A (https=) |
| MX (1) | MX2010007501A (https=) |
| TW (1) | TWI465251B (https=) |
| WO (1) | WO2009089022A1 (https=) |
| ZA (1) | ZA201005130B (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3209821B2 (ja) | 1993-03-31 | 2001-09-17 | 日立ビアメカニクス株式会社 | 消耗電極式ガスシールドアーク溶接の出力制御方法およびその溶接装置 |
| US8361438B2 (en) | 2008-01-08 | 2013-01-29 | Lantheus Medical Imaging, Inc. | N-alkoxyamide conjugates as imaging agents |
| CA2803520C (en) * | 2009-07-08 | 2019-10-22 | Lantheus Medical Imaging, Inc. | N-alkoxyamide conjugates as imaging agents |
| PL3050878T3 (pl) | 2013-09-24 | 2022-01-24 | Fujifilm Corporation | Zawierający atom azotu związek lub jego sól, lub ich kompleks z metalem |
Family Cites Families (39)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5122885A (en) * | 1974-08-13 | 1976-02-23 | Sagami Chem Res | Ashiru ll aminosan oo chikanhidorokisamidono seizohoho |
| JPS5910322B2 (ja) | 1975-07-30 | 1984-03-08 | 三井東圧化学株式会社 | 殺草剤 |
| HU175152B (hu) * | 1976-12-30 | 1980-05-28 | Richter Gedeon Vegyeszet | Sposob poluchenija peptidov s gastrin-aktivnost'ju, soderzhahhikh amino-oksi-kisloty |
| US4859777A (en) * | 1981-07-01 | 1989-08-22 | Eastman Kodak Company | Terpyridine chelating agents |
| US4957939A (en) * | 1981-07-24 | 1990-09-18 | Schering Aktiengesellschaft | Sterile pharmaceutical compositions of gadolinium chelates useful enhancing NMR imaging |
| EP0247156B1 (en) * | 1985-11-18 | 1993-06-23 | Access Pharmaceuticals Inc. | Polychelating agents for image and spectral enhancement (and spectral shift) |
| EP0233607B1 (en) | 1986-02-18 | 1991-03-13 | E.R. Squibb & Sons, Inc. | [(2,2,2-Trichloroethoxy) methoxy]amine |
| US5064956A (en) * | 1987-06-24 | 1991-11-12 | The Dow Chemical Company | Process for preparing mono-n-alkylated polyazamacrocycles |
| JP2573006B2 (ja) | 1987-12-17 | 1997-01-16 | 富士薬品工業株式会社 | 新規なヒドロキサム酸誘導体 |
| IT1224627B (it) * | 1988-04-12 | 1990-10-04 | Guidotti & C Spa Labor | Ammidi di acidi ciclometilen_1,2_dicarbossilici adattivita' terapeutica, procedimenti per la loro preparazione e composizioni farmaceutiche che le contengono. |
| US5087440A (en) * | 1989-07-31 | 1992-02-11 | Salutar, Inc. | Heterocyclic derivatives of DTPA used for magnetic resonance imaging |
| US5089043A (en) * | 1989-11-09 | 1992-02-18 | Shionogi & Co., Ltd. | Heterocyclic oxy-phenoxyacetic acid derivatives and their use as herbicides |
| JPH0491070A (ja) * | 1990-08-06 | 1992-03-24 | Kanebo Ltd | カリックスアレーン誘導体 |
| US5225173A (en) * | 1991-06-12 | 1993-07-06 | Idaho Research Foundation, Inc. | Methods and devices for the separation of radioactive rare earth metal isotopes from their alkaline earth metal precursors |
| US5274129A (en) * | 1991-06-12 | 1993-12-28 | Idaho Research Foundation, Inc. | Hydroxamic acid crown ethers |
| GB9115375D0 (en) * | 1991-07-17 | 1991-09-04 | Salutar Inc | Compounds |
| US5639746A (en) * | 1994-12-29 | 1997-06-17 | The Procter & Gamble Company | Hydroxamic acid-containing inhibitors of matrix metalloproteases |
| TW319763B (https=) * | 1995-02-01 | 1997-11-11 | Epix Medical Inc | |
| EP0955044B1 (en) | 1995-06-26 | 2005-11-16 | Chelator LLC | Method of inhibiting bacterial or fungal growth using a complexing agent |
| NZ305940A (en) | 1995-07-26 | 1999-05-28 | Pfizer | N-(aroyl)glycine hydroxamic acid derivatives and related compounds that inhibit the production of tnf and are useful in treating asthma |
| US6461587B1 (en) * | 1999-03-22 | 2002-10-08 | Schering Aktiengesellschaft | Perfluoroalkylamides, their production and their use in diagnosis |
| US6989139B2 (en) * | 2000-02-15 | 2006-01-24 | Bristol-Myers Squibb Pharma Company | Matrix metalloproteinase inhibitors |
| US6656448B1 (en) * | 2000-02-15 | 2003-12-02 | Bristol-Myers Squibb Pharma Company | Matrix metalloproteinase inhibitors |
| US20020002152A1 (en) * | 2000-04-14 | 2002-01-03 | Craig Richard A. | Hydrazide and alkoxyamide angiogenesis inhibitors |
| EP1377321A4 (en) * | 2001-02-23 | 2006-01-11 | Bristol Myers Squibb Co | RECOVERY ANTAGONISTS RECEIVING DETECTABLE MACROPHAGE RECEPTORS FOR THE IDENTIFICATION OF ATHEROSCLEROSIS AND VULNERABLE PLAQUE BY IMAGING |
| JP4590157B2 (ja) * | 2001-03-21 | 2010-12-01 | アイシス イノヴェイション リミテッド | アッセイ、方法および手段 |
| TWI240632B (en) | 2001-07-30 | 2005-10-01 | Epix Medical Inc | Purified peptides for peptide-based multimeric targeted contrast agents |
| WO2005001415A2 (en) | 2003-05-23 | 2005-01-06 | Epix Pharmaceuticals, Inc. | Optically pure and enriched isomers of chelating ligands and contrast agents |
| JP2007521254A (ja) * | 2003-06-25 | 2007-08-02 | ゲルベ | 診断画像用化合物 |
| WO2005020973A2 (en) | 2003-08-29 | 2005-03-10 | The University Of Houston System | Compositions having antimycrobial activity including a hydroxamate or a hydroxamate and a hydroxylamine |
| US20050106100A1 (en) * | 2003-09-03 | 2005-05-19 | Harris Thomas D. | Compounds containing matrix metalloproteinase substrates and methods of their use |
| WO2005084179A2 (en) | 2003-12-01 | 2005-09-15 | Immunomedics, Inc. | Improved method for preparing conjugates of proteins and chelating agents |
| US20070142417A1 (en) * | 2005-05-11 | 2007-06-21 | Aventis Pharmaceuticals Inc | Substantially Pure 2-{[2-(2-Methylamino-Pyrimidin-4-YL)-1H-Indole-5-Carbonyl]-Amino}-3-Phenylpyridin-2-YL-Amino)-Propionic Acid as an IkB Kinase Inhibitor |
| WO2007005491A1 (en) * | 2005-06-30 | 2007-01-11 | Bristol-Myers Squibb Pharma Company | Hydrazide conjugates as imaging agents |
| US7618957B2 (en) * | 2005-07-15 | 2009-11-17 | Bayer Schering Pharma Aktiengesellschaft | Perfluoroalkyl-containing complexes, process for their production as well as their use |
| DE102005033902B3 (de) | 2005-07-15 | 2007-04-05 | Schering Ag | Perfluoralkylhaltige Komplexe, Verfahren zu deren Herstellung, sowie deren Verwendung und diese enthaltende pharmazeutische Mittel |
| US8361438B2 (en) | 2008-01-08 | 2013-01-29 | Lantheus Medical Imaging, Inc. | N-alkoxyamide conjugates as imaging agents |
| WO2011000532A2 (de) | 2009-07-03 | 2011-01-06 | Archimica Gmbh | Verfahren zur enantioselektiven addition von organometallischen kohlenstoffnukleophilen an trifluormethylketone und verwendung des verfahrens in der synthese von hiv reverse transcriptase inhibitoren |
| CA2803520C (en) | 2009-07-08 | 2019-10-22 | Lantheus Medical Imaging, Inc. | N-alkoxyamide conjugates as imaging agents |
-
2009
- 2009-01-08 US US12/350,628 patent/US8361438B2/en active Active
- 2009-01-08 KR KR1020107017602A patent/KR101595324B1/ko not_active Expired - Fee Related
- 2009-01-08 CA CA2711426A patent/CA2711426C/en active Active
- 2009-01-08 JP JP2010542266A patent/JP5730581B2/ja not_active Expired - Fee Related
- 2009-01-08 AU AU2009204427A patent/AU2009204427B2/en not_active Ceased
- 2009-01-08 MX MX2010007501A patent/MX2010007501A/es active IP Right Grant
- 2009-01-08 TW TW098100454A patent/TWI465251B/zh not_active IP Right Cessation
- 2009-01-08 BR BRPI0907612-3A patent/BRPI0907612A2/pt not_active Application Discontinuation
- 2009-01-08 EP EP09700768.6A patent/EP2240206B1/en active Active
- 2009-01-08 ES ES09700768.6T patent/ES2629340T3/es active Active
- 2009-01-08 CN CN200980108357.9A patent/CN101970015B/zh not_active Expired - Fee Related
- 2009-01-08 KR KR1020167003565A patent/KR101861025B1/ko not_active Expired - Fee Related
- 2009-01-08 CN CN201410136402.4A patent/CN103965128B/zh not_active Expired - Fee Related
- 2009-01-08 WO PCT/US2009/000096 patent/WO2009089022A1/en not_active Ceased
-
2010
- 2010-07-06 IL IL206846A patent/IL206846A/en active IP Right Grant
- 2010-07-19 ZA ZA2010/05130A patent/ZA201005130B/en unknown
-
2012
- 2012-12-21 US US13/723,333 patent/US8852553B2/en active Active
-
2014
- 2014-01-02 AU AU2014200012A patent/AU2014200012C1/en not_active Ceased
- 2014-09-02 US US14/474,566 patent/US9266846B2/en active Active
-
2015
- 2015-04-08 JP JP2015079425A patent/JP6087386B2/ja not_active Expired - Fee Related
- 2015-12-21 US US14/977,249 patent/US9732047B2/en active Active
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