JP2010531304A5 - - Google Patents

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Publication number
JP2010531304A5
JP2010531304A5 JP2010513237A JP2010513237A JP2010531304A5 JP 2010531304 A5 JP2010531304 A5 JP 2010531304A5 JP 2010513237 A JP2010513237 A JP 2010513237A JP 2010513237 A JP2010513237 A JP 2010513237A JP 2010531304 A5 JP2010531304 A5 JP 2010531304A5
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JP
Japan
Prior art keywords
group
hydrogen atom
alkyl
chemical formula
aralkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010513237A
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English (en)
Japanese (ja)
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JP2010531304A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/007594 external-priority patent/WO2008156783A2/en
Publication of JP2010531304A publication Critical patent/JP2010531304A/ja
Publication of JP2010531304A5 publication Critical patent/JP2010531304A5/ja
Pending legal-status Critical Current

Links

JP2010513237A 2007-06-18 2008-06-18 抗悪性腫瘍活性を有するpfkfb3阻害物質ファミリー Pending JP2010531304A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93603007P 2007-06-18 2007-06-18
PCT/US2008/007594 WO2008156783A2 (en) 2007-06-18 2008-06-18 Family of pfkfb3 inhibitors with anti-neoplastic activities

Publications (2)

Publication Number Publication Date
JP2010531304A JP2010531304A (ja) 2010-09-24
JP2010531304A5 true JP2010531304A5 (enExample) 2011-07-28

Family

ID=39735477

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010513237A Pending JP2010531304A (ja) 2007-06-18 2008-06-18 抗悪性腫瘍活性を有するpfkfb3阻害物質ファミリー

Country Status (5)

Country Link
US (1) US8088385B2 (enExample)
EP (1) EP2167058B1 (enExample)
JP (1) JP2010531304A (enExample)
AU (1) AU2008266856A1 (enExample)
WO (1) WO2008156783A2 (enExample)

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EP2525790B1 (en) 2009-10-21 2020-05-27 Agios Pharmaceuticals, Inc. Methods and compositions for cell-proliferation-related disorders
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US9492418B2 (en) 2011-05-10 2016-11-15 Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College Inhibitors of PFKFB3 for cancer therapy
RU2477723C2 (ru) 2011-06-16 2013-03-20 Общество С Ограниченной Ответственностью "Фьюжн Фарма" Ингибиторы протеинкиназ (варианты), их применение для лечения онкологических заболеваний и фармацевтическая композиция на их основе
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US10000449B2 (en) 2011-12-22 2018-06-19 Kancera Ab Bisarylsulfonamides useful in the treatment of inflammation and cancer
CN104168958B (zh) 2011-12-22 2017-12-01 坎塞拉有限公司 可用于治疗炎症和癌症的二芳基磺酰胺
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US8828998B2 (en) 2012-06-25 2014-09-09 Infinity Pharmaceuticals, Inc. Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors
KR102229478B1 (ko) 2012-11-01 2021-03-18 인피니티 파마슈티칼스, 인코포레이티드 Pi3 키나아제 동형단백질 조절인자를 사용하는 암의 치료
US8871754B2 (en) 2012-11-19 2014-10-28 Irm Llc Compounds and compositions for the treatment of parasitic diseases
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US9663486B2 (en) 2013-10-14 2017-05-30 Eisai R&D Management Co., Ltd. Selectively substituted quinoline compounds
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JP6543268B2 (ja) 2014-04-15 2019-07-10 バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated 嚢胞性線維症膜コンダクタンス調節因子が媒介する疾患を処置するための医薬組成物
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