JP2010531304A5 - - Google Patents

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Publication number
JP2010531304A5
JP2010531304A5 JP2010513237A JP2010513237A JP2010531304A5 JP 2010531304 A5 JP2010531304 A5 JP 2010531304A5 JP 2010513237 A JP2010513237 A JP 2010513237A JP 2010513237 A JP2010513237 A JP 2010513237A JP 2010531304 A5 JP2010531304 A5 JP 2010531304A5
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JP
Japan
Prior art keywords
group
hydrogen atom
alkyl
chemical formula
aralkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010513237A
Other languages
English (en)
Japanese (ja)
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JP2010531304A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/007594 external-priority patent/WO2008156783A2/en
Publication of JP2010531304A publication Critical patent/JP2010531304A/ja
Publication of JP2010531304A5 publication Critical patent/JP2010531304A5/ja
Pending legal-status Critical Current

Links

JP2010513237A 2007-06-18 2008-06-18 抗悪性腫瘍活性を有するpfkfb3阻害物質ファミリー Pending JP2010531304A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93603007P 2007-06-18 2007-06-18
PCT/US2008/007594 WO2008156783A2 (en) 2007-06-18 2008-06-18 Family of pfkfb3 inhibitors with anti-neoplastic activities

Publications (2)

Publication Number Publication Date
JP2010531304A JP2010531304A (ja) 2010-09-24
JP2010531304A5 true JP2010531304A5 (enExample) 2011-07-28

Family

ID=39735477

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010513237A Pending JP2010531304A (ja) 2007-06-18 2008-06-18 抗悪性腫瘍活性を有するpfkfb3阻害物質ファミリー

Country Status (5)

Country Link
US (1) US8088385B2 (enExample)
EP (1) EP2167058B1 (enExample)
JP (1) JP2010531304A (enExample)
AU (1) AU2008266856A1 (enExample)
WO (1) WO2008156783A2 (enExample)

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WO2011161201A1 (en) 2010-06-22 2011-12-29 Kancera Ab Bisarylsulfonamides useful as kinase inhibitors in the treatment of inflammation and cancer
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US9492418B2 (en) 2011-05-10 2016-11-15 Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College Inhibitors of PFKFB3 for cancer therapy
RU2477723C2 (ru) 2011-06-16 2013-03-20 Общество С Ограниченной Ответственностью "Фьюжн Фарма" Ингибиторы протеинкиназ (варианты), их применение для лечения онкологических заболеваний и фармацевтическая композиция на их основе
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KR102030609B1 (ko) 2011-09-02 2019-10-11 인사이트 홀딩스 코포레이션 Pi3k 억제제로서 헤테로시클릴아민
US10000449B2 (en) 2011-12-22 2018-06-19 Kancera Ab Bisarylsulfonamides useful in the treatment of inflammation and cancer
MX348147B (es) 2011-12-22 2017-05-30 Kancera Ab Biarilsulfonamidas utiles en el tratamiento de la inflamacion y cancer.
CA2868787A1 (en) * 2012-03-29 2013-10-03 Advanced Cancer Therapeutics, Llc Pfkfb3 inhibitor and methods of use as an anti-cancer therapeutic
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US8828998B2 (en) 2012-06-25 2014-09-09 Infinity Pharmaceuticals, Inc. Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors
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US9732097B2 (en) 2015-05-11 2017-08-15 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
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WO2017208174A2 (en) * 2016-05-31 2017-12-07 The Regents Of The University Of California Methods of treating disease with pfkfb3 inhibitors
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US7846915B2 (en) * 2004-10-20 2010-12-07 Resverlogix Corporation Stilbenes and chalcones for the prevention and treatment of cardiovascular diseases

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