JP2010522242A5 - - Google Patents
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- Publication number
- JP2010522242A5 JP2010522242A5 JP2010501112A JP2010501112A JP2010522242A5 JP 2010522242 A5 JP2010522242 A5 JP 2010522242A5 JP 2010501112 A JP2010501112 A JP 2010501112A JP 2010501112 A JP2010501112 A JP 2010501112A JP 2010522242 A5 JP2010522242 A5 JP 2010522242A5
- Authority
- JP
- Japan
- Prior art keywords
- disease
- tachyarrhythmia
- crohn
- pain
- bowel syndrome
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 208000011231 Crohn disease Diseases 0.000 claims 4
- 208000002193 Pain Diseases 0.000 claims 4
- 206010049447 Tachyarrhythmia Diseases 0.000 claims 4
- 208000001871 Tachycardia Diseases 0.000 claims 4
- 150000001875 compounds Chemical class 0.000 claims 4
- 239000003814 drug Substances 0.000 claims 4
- 208000002551 irritable bowel syndrome Diseases 0.000 claims 4
- 208000024891 symptom Diseases 0.000 claims 2
- 229940124597 therapeutic agent Drugs 0.000 claims 2
- 108010052164 Sodium Channels Proteins 0.000 claims 1
- 102000018674 Sodium Channels Human genes 0.000 claims 1
- 201000010099 disease Diseases 0.000 claims 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 239000012453 solvate Substances 0.000 claims 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US89673507P | 2007-03-23 | 2007-03-23 | |
| US60/896,735 | 2007-03-23 | ||
| US3532408P | 2008-03-10 | 2008-03-10 | |
| US61/035,324 | 2008-03-10 | ||
| PCT/US2008/057730 WO2008118758A1 (en) | 2007-03-23 | 2008-03-20 | Inhibitors of ion channels |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010522242A JP2010522242A (ja) | 2010-07-01 |
| JP2010522242A5 true JP2010522242A5 (enExample) | 2011-04-21 |
| JP5361857B2 JP5361857B2 (ja) | 2013-12-04 |
Family
ID=39788940
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010501112A Expired - Fee Related JP5361857B2 (ja) | 2007-03-23 | 2008-03-20 | イオンチャネルの阻害剤 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US8357711B2 (enExample) |
| EP (1) | EP1995241B1 (enExample) |
| JP (1) | JP5361857B2 (enExample) |
| AR (1) | AR065824A1 (enExample) |
| AT (1) | ATE461177T1 (enExample) |
| CA (1) | CA2681572C (enExample) |
| CL (1) | CL2008000835A1 (enExample) |
| DE (1) | DE602008000809D1 (enExample) |
| ES (1) | ES2340640T3 (enExample) |
| PA (1) | PA8773501A1 (enExample) |
| PE (1) | PE20090237A1 (enExample) |
| TW (1) | TW200845969A (enExample) |
| UY (1) | UY30978A1 (enExample) |
| WO (1) | WO2008118758A1 (enExample) |
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| WO2006060762A2 (en) | 2004-12-03 | 2006-06-08 | Arena Pharmaceuticals, Inc. | Pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto |
| GB0510139D0 (en) | 2005-05-18 | 2005-06-22 | Addex Pharmaceuticals Sa | Novel compounds B1 |
| GB0513702D0 (en) | 2005-07-04 | 2005-08-10 | Sterix Ltd | Compound |
| US7754717B2 (en) | 2005-08-15 | 2010-07-13 | Amgen Inc. | Bis-aryl amide compounds and methods of use |
| AU2006312083A1 (en) | 2005-11-03 | 2007-05-18 | Merck Sharp & Dohme Corp. | Histone deacetylase inhibitors with aryl-pyrazolyl motifs |
| CN101460491A (zh) | 2006-04-12 | 2009-06-17 | 惠氏公司 | 苯胺基嘧啶苯基和苯并噻吩类似物 |
-
2008
- 2008-03-20 DE DE602008000809T patent/DE602008000809D1/de active Active
- 2008-03-20 CL CL200800835A patent/CL2008000835A1/es unknown
- 2008-03-20 WO PCT/US2008/057730 patent/WO2008118758A1/en not_active Ceased
- 2008-03-20 ES ES08153165T patent/ES2340640T3/es active Active
- 2008-03-20 AT AT08153165T patent/ATE461177T1/de not_active IP Right Cessation
- 2008-03-20 CA CA2681572A patent/CA2681572C/en not_active Expired - Fee Related
- 2008-03-20 JP JP2010501112A patent/JP5361857B2/ja not_active Expired - Fee Related
- 2008-03-20 US US12/052,593 patent/US8357711B2/en not_active Expired - Fee Related
- 2008-03-20 EP EP08153165A patent/EP1995241B1/en active Active
- 2008-03-21 TW TW097110261A patent/TW200845969A/zh unknown
- 2008-03-24 PA PA20088773501A patent/PA8773501A1/es unknown
- 2008-03-24 PE PE2008000533A patent/PE20090237A1/es not_active Application Discontinuation
- 2008-03-24 UY UY30978A patent/UY30978A1/es not_active Application Discontinuation
- 2008-03-25 AR ARP080101215A patent/AR065824A1/es not_active Application Discontinuation
-
2012
- 2012-11-15 US US13/677,849 patent/US8741934B2/en not_active Expired - Fee Related
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