JP2010518173A5 - - Google Patents

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Publication number
JP2010518173A5
JP2010518173A5 JP2009549760A JP2009549760A JP2010518173A5 JP 2010518173 A5 JP2010518173 A5 JP 2010518173A5 JP 2009549760 A JP2009549760 A JP 2009549760A JP 2009549760 A JP2009549760 A JP 2009549760A JP 2010518173 A5 JP2010518173 A5 JP 2010518173A5
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JP
Japan
Prior art keywords
salt
cancer
salts
group
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009549760A
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English (en)
Japanese (ja)
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JP2010518173A (ja
JP5504460B2 (ja
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Publication date
Priority claimed from CNA2007100375572A external-priority patent/CN101245050A/zh
Application filed filed Critical
Publication of JP2010518173A publication Critical patent/JP2010518173A/ja
Publication of JP2010518173A5 publication Critical patent/JP2010518173A5/ja
Application granted granted Critical
Publication of JP5504460B2 publication Critical patent/JP5504460B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009549760A 2007-02-14 2008-02-04 4−フェニルアミノキナゾリン誘導体の塩形態 Active JP5504460B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN200710037557.2 2007-02-14
CNA2007100375572A CN101245050A (zh) 2007-02-14 2007-02-14 4-苯胺喹唑啉衍生物的盐
PCT/CN2008/000318 WO2008098485A1 (en) 2007-02-14 2008-02-04 The salts of 4-aniline quinazoline derivative

Publications (3)

Publication Number Publication Date
JP2010518173A JP2010518173A (ja) 2010-05-27
JP2010518173A5 true JP2010518173A5 (https=) 2011-04-07
JP5504460B2 JP5504460B2 (ja) 2014-05-28

Family

ID=39689656

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009549760A Active JP5504460B2 (ja) 2007-02-14 2008-02-04 4−フェニルアミノキナゾリン誘導体の塩形態

Country Status (8)

Country Link
US (1) US8349854B2 (https=)
EP (1) EP2116540B1 (https=)
JP (1) JP5504460B2 (https=)
KR (1) KR20100014947A (https=)
CN (3) CN101245050A (https=)
AU (1) AU2008215053B2 (https=)
CA (1) CA2677978C (https=)
WO (1) WO2008098485A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101347433B (zh) * 2007-07-20 2012-05-02 江苏艾力斯生物医药有限公司 4-苯胺喹唑啉衍生物的制药用途
CN101544609A (zh) * 2008-03-25 2009-09-30 上海艾力斯医药科技有限公司 4-苯胺喹唑啉衍生物的结晶形式
CN101584696A (zh) 2008-05-21 2009-11-25 上海艾力斯医药科技有限公司 包含喹唑啉衍生物的组合物及制备方法、用途
AU2016379292B2 (en) 2015-12-24 2021-03-25 Kyowa Kirin Co., Ltd. α, β unsaturated amide compound
CN106117182B (zh) * 2016-06-20 2019-08-30 中国药科大学 喹唑啉-n-苯乙基四氢异喹啉类化合物及其制备方法和应用
CN112225679A (zh) * 2020-10-13 2021-01-15 苏州亚科科技股份有限公司 一种3-(环己胺)-2-羟基-1-丙磺酸的制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ243082A (en) 1991-06-28 1995-02-24 Ici Plc 4-anilino-quinazoline derivatives; pharmaceutical compositions, preparatory processes, and use thereof
AU661533B2 (en) 1992-01-20 1995-07-27 Astrazeneca Ab Quinazoline derivatives
GB9314893D0 (en) 1993-07-19 1993-09-01 Zeneca Ltd Quinazoline derivatives
GB9510757D0 (en) * 1994-09-19 1995-07-19 Wellcome Found Therapeuticaly active compounds
MX9707453A (es) 1995-03-30 1997-12-31 Pfizer Derivados de quinazolina.
HU228446B1 (en) 1996-04-12 2013-03-28 Warner Lambert Co Kinazoline derivatives as irreversible inhibitors of protein-kinase, pharmaceutical compositions containing these compounds and use thereof
GB9800575D0 (en) * 1998-01-12 1998-03-11 Glaxo Group Ltd Heterocyclic compounds
RS49779B (sr) 1998-01-12 2008-06-05 Glaxo Group Limited, Biciklična heteroaromatična jedinjenja kao inhibitori protein tirozin kinaze
AU5391099A (en) 1998-07-30 2000-02-21 American Home Products Corporation Substituted quinazoline derivatives
PL204958B1 (pl) * 2000-06-30 2010-02-26 Glaxo Group Ltd Ditosylany związków chinazolinowych, środek farmaceutyczny i zastosowanie tych związków
KR100735639B1 (ko) * 2004-12-29 2007-07-04 한미약품 주식회사 암세포 성장 억제 효과를 갖는 퀴나졸린 유도체 및 이의제조방법
CN101003514A (zh) * 2006-01-20 2007-07-25 上海艾力斯医药科技有限公司 喹唑啉衍生物、其制备方法及用途

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